Known Bioactive Library: Microsource 1 - US Drug Collection · 2091 C20 Microsource 01500181...

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ICCB-L Plate ICCB-L Well Vendor Vendor ID Compound Name Bioactivity Source CAS 2091 A03 Microsource 00200046 GRISEOFULVIN antifungal, inhibits mitosis in metaphase Penicillium griseofulvum 126-07-8 2091 A04 Microsource 01500161 CARBINOXAMINE MALEATE antihistaminic synthetic 3505-38-2, 486-16-8 [carbinoxamine] 2091 A05 Microsource 00200331 SALSALATE analgesic synthetic 552-94-3 2091 A06 Microsource 01500162 CARISOPRODOL muscle relaxant (skeletal) synthetic 78-44-4 2091 A07 Microsource 00210369 GALLIC ACID antineoplastic, astringent, antibacterial insect galls 149-91-7 2091 A08 Microsource 01500163 CEFADROXIL antibacterial semisynthetic 66592-87-8, 50370-12- 2 [anhydrous], 119922- 89-9 [hemihydrate] 2091 A09 Microsource 00211468 DANTHRON cathartic Rheum palmatum, Xyris semifuscata 117-10-2 2091 A10 Microsource 01500164 CEFAZOLIN SODIUM antibacterial semisynthetic 27164-46-1, 25953-19- 9 [cefazolin] 2091 A11 Microsource 00300024 HYDROCORTISONE glucocorticoid, antiinflammatory adrenal glands 50-23-7 2091 A12 Microsource 01500165 CEFOTAXIME SODIUM antibacterial semisynthetic 64485-93-4, 63527-52- 6 [cefotaxime] 2091 A13 Microsource 00300029 DESOXYCORTICOSTERONE ACETATE mineralocorticoid adrenocortex 56-47-3 2091 A14 Microsource 01500166 CEPHALOTHIN SODIUM antibacterial semisynthetic 58-71-9, 153-61-7 [cephalothin] 2091 A15 Microsource 00300034 TESTOSTERONE PROPIONATE androgen, antineoplastic semisynthetic 57-85-2 2091 A16 Microsource 01500167 CEPHAPIRIN SODIUM antibacterial semisynthetic 24356-60-3, 21593-23- 7 [cephapirin] 2091 A17 Microsource 00300548 SPARTEINE SULFATE oxytocic Lupinus spp and other Leguminosae 6160-12-9, 299-39-8 [anhydrous], 90-39-1 [sparteine] 2091 A18 Microsource 01500168 CEPHRADINE antibacterial semisynthetic 38821-53-3 [anhydrous], 58456-863 [dihydrate], 31828- 50-9 [non- stoichiometric hydrate] 2091 A19 Microsource 00300607 RUTOSIDE (rutin) vascular protectant Ruta graveolens, widespread in plants 153-18-4 2091 A20 Microsource 01500169 CETYLPYRIDINIUM CHLORIDE antiinfective (topical) synthetic 6004-24-6, 123-03-5 [anhydrous] 2091 A21 Microsource 00300618 SALICYLANILIDE antipyretic, fungicide synthetic 87-17-2 2091 A22 Microsource 01500171 CHLORAMBUCIL antineoplastic, alkylating agent synthetic 305-03-3 2091 B03 Microsource 01500263 DOPAMINE HYDROCHLORIDE cardiotonic, antihypotensive synthetic 62-31-7, 51-61-6 [dopamine] 2091 B04 Microsource 01500375 MECHLORETHAMINE antineoplastic, alkylating agent synthetic 55-86-7, 51-75-2 [mechlorethamine] 2091 B05 Microsource 01500264 DOXEPIN HYDROCHLORIDE antidepressant synthetic 1229-29-4, 1668-19-5 [doxepin], 4698-39-9 [(//E//)-isomer], 25127- 31-5 [(//Z//)-isomer] 2091 B06 Microsource 01500376 MECLIZINE HYDROCHLORIDE antiemetic synthetic 31884-77-2, 1104-22- 9 [anhydrous], 569-65- 3 [meclizine] 2091 B07 Microsource 01500266 DOXYCYCLINE HYDROCHLORIDE antibacterial semisynthetic; GS- 3065 17086-28-1, 564-25-0 [anhydrous] 2091 B08 Microsource 01500377 MECLOFENAMATE SODIUM antiinflammatory, antipyretic synthetic 6385-02-0 2091 B09 Microsource 01500267 DOXYLAMINE SUCCINATE antihistaminic, hypnotic synthetic 562-10-7, 469-21-6 [doxylamine] 2091 B10 Microsource 01500379 MEDROXYPROGESTERONE ACETATE contraceptive semisynthetic 71-58-9, 520-85-4 [medroxyprogesterone ] 2091 B11 Microsource 01500268 DYCLONINE HYDROCHLORIDE anesthetic (topical) synthetic 536-43-6, 586-60-7 [dyclonine] 2091 B12 Microsource 01500380 MEDRYSONE glucocorticoid semisynthetic 2668-66-8 2091 B13 Microsource 01500269 DYPHYLLINE PDE inhibitor, bronchodilator, vasodilator synthetic 479-18-5 2091 B14 Microsource 01500381 MEGESTROL ACETATE progestogen, antineoplastic semisynthetic 595-33-5, 3562-63-8 [megestrol] 2091 B15 Microsource 01500270 TRISODIUM ETHYLENEDIAMINE TETRACETATE chelating agent, antioxidant synthetic 150-38-9 2091 B16 Microsource 01500382 MELPHALAN antineoplastic, alkylating agent synthetic 148-82-3 Known Bioactive Library: Microsource 1 - US Drug Collection Microsource1-US Drug Collection Page 1 of 24 Created 9/2015

Transcript of Known Bioactive Library: Microsource 1 - US Drug Collection · 2091 C20 Microsource 01500181...

Page 1: Known Bioactive Library: Microsource 1 - US Drug Collection · 2091 C20 Microsource 01500181 CHLOROTRIANISENE estrogen synthetic 569-57-3 2091 C21 Microsource 00330018 DICHLORVOS

ICCB-L Plate

ICCB-L Well

VendorVendor

IDCompound Name Bioactivity Source CAS

2091 A03 Microsource 00200046 GRISEOFULVINantifungal, inhibits mitosis in metaphase

Penicillium griseofulvum

126-07-8

2091 A04 Microsource 01500161 CARBINOXAMINE MALEATE antihistaminic synthetic3505-38-2, 486-16-8 [carbinoxamine]

2091 A05 Microsource 00200331 SALSALATE analgesic synthetic 552-94-3

2091 A06 Microsource 01500162 CARISOPRODOLmuscle relaxant (skeletal)

synthetic 78-44-4

2091 A07 Microsource 00210369 GALLIC ACIDantineoplastic, astringent, antibacterial

insect galls 149-91-7

2091 A08 Microsource 01500163 CEFADROXIL antibacterial semisynthetic66592-87-8, 50370-12-2 [anhydrous], 119922-89-9 [hemihydrate]

2091 A09 Microsource 00211468 DANTHRON catharticRheum palmatum, Xyris semifuscata

117-10-2

2091 A10 Microsource 01500164 CEFAZOLIN SODIUM antibacterial semisynthetic27164-46-1, 25953-19-9 [cefazolin]

2091 A11 Microsource 00300024 HYDROCORTISONEglucocorticoid, antiinflammatory

adrenal glands 50-23-7

2091 A12 Microsource 01500165 CEFOTAXIME SODIUM antibacterial semisynthetic64485-93-4, 63527-52-6 [cefotaxime]

2091 A13 Microsource 00300029 DESOXYCORTICOSTERONE ACETATE mineralocorticoid adrenocortex 56-47-3

2091 A14 Microsource 01500166 CEPHALOTHIN SODIUM antibacterial semisynthetic58-71-9, 153-61-7 [cephalothin]

2091 A15 Microsource 00300034 TESTOSTERONE PROPIONATE androgen, antineoplastic semisynthetic 57-85-2

2091 A16 Microsource 01500167 CEPHAPIRIN SODIUM antibacterial semisynthetic24356-60-3, 21593-23-7 [cephapirin]

2091 A17 Microsource 00300548 SPARTEINE SULFATE oxytocicLupinus spp and other Leguminosae

6160-12-9, 299-39-8 [anhydrous], 90-39-1 [sparteine]

2091 A18 Microsource 01500168 CEPHRADINE antibacterial semisynthetic

38821-53-3 [anhydrous], 58456-86-3 [dihydrate], 31828-50-9 [non-stoichiometric hydrate]

2091 A19 Microsource 00300607 RUTOSIDE (rutin) vascular protectantRuta graveolens, widespread in plants

153-18-4

2091 A20 Microsource 01500169 CETYLPYRIDINIUM CHLORIDE antiinfective (topical) synthetic6004-24-6, 123-03-5 [anhydrous]

2091 A21 Microsource 00300618 SALICYLANILIDE antipyretic, fungicide synthetic 87-17-2

2091 A22 Microsource 01500171 CHLORAMBUCILantineoplastic, alkylating agent

synthetic 305-03-3

2091 B03 Microsource 01500263 DOPAMINE HYDROCHLORIDEcardiotonic, antihypotensive

synthetic62-31-7, 51-61-6 [dopamine]

2091 B04 Microsource 01500375 MECHLORETHAMINEantineoplastic, alkylating agent

synthetic55-86-7, 51-75-2 [mechlorethamine]

2091 B05 Microsource 01500264 DOXEPIN HYDROCHLORIDE antidepressant synthetic

1229-29-4, 1668-19-5 [doxepin], 4698-39-9 [(//E//)-isomer], 25127-31-5 [(//Z//)-isomer]

2091 B06 Microsource 01500376 MECLIZINE HYDROCHLORIDE antiemetic synthetic31884-77-2, 1104-22-9 [anhydrous], 569-65-3 [meclizine]

2091 B07 Microsource 01500266 DOXYCYCLINE HYDROCHLORIDE antibacterialsemisynthetic; GS-3065

17086-28-1, 564-25-0 [anhydrous]

2091 B08 Microsource 01500377 MECLOFENAMATE SODIUMantiinflammatory, antipyretic

synthetic 6385-02-0

2091 B09 Microsource 01500267 DOXYLAMINE SUCCINATE antihistaminic, hypnotic synthetic562-10-7, 469-21-6 [doxylamine]

2091 B10 Microsource 01500379 MEDROXYPROGESTERONE ACETATE contraceptive semisynthetic71-58-9, 520-85-4 [medroxyprogesterone]

2091 B11 Microsource 01500268 DYCLONINE HYDROCHLORIDE anesthetic (topical) synthetic536-43-6, 586-60-7 [dyclonine]

2091 B12 Microsource 01500380 MEDRYSONE glucocorticoid semisynthetic 2668-66-8

2091 B13 Microsource 01500269 DYPHYLLINEPDE inhibitor, bronchodilator, vasodilator

synthetic 479-18-5

2091 B14 Microsource 01500381 MEGESTROL ACETATEprogestogen, antineoplastic

semisynthetic595-33-5, 3562-63-8 [megestrol]

2091 B15 Microsource 01500270TRISODIUM ETHYLENEDIAMINE TETRACETATE

chelating agent, antioxidant

synthetic 150-38-9

2091 B16 Microsource 01500382 MELPHALANantineoplastic, alkylating agent

synthetic 148-82-3

Known Bioactive Library: Microsource 1 - US Drug Collection

Microsource1-US Drug Collection Page 1 of 24 Created 9/2015

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ICCB-L Plate

ICCB-L Well

VendorVendor

IDCompound Name Bioactivity Source CAS

2091 B17 Microsource 01500272 EMETINEinhibits RNA, DNA and protein synthesis

Uragoga ipecacuanha

316-42-7, 483-18-1 [emetine]

2091 B18 Microsource 01500383 MEPENZOLATE BROMIDE anticholinergic synthetic76-90-4, 25990-43-6 [mepenzolate]

2091 B19 Microsource 01500276 ERGOCALCIFEROLantirachitic vitamin; LD50 (rat) 56 mg/kg po

irradiation of ergosterol

50-14-6

2091 B20 Microsource 01500387 MERCAPTOPURINEantineoplastic, purine antimetabolite

synthetic6112-76-1, 50-44-2 [anhydrous]

2091 B21 Microsource 01500277 ERGONOVINE MALEATE oxytocic, 5HT antagonistergot and Convolvulvaceae spp

129-51-1, 60-79-7 [ergonovine]

2091 B22 Microsource 01500388 MESTRANOLestrogen, with progesterone as oral contraceptive

semisynthetic 72-33-3

2091 C03 Microsource 00305025 PHENYL AMINOSALICYLATEantibacterial (tuberculostatic)

synthetic; NSC-40144

133-11-9

2091 C04 Microsource 01500172 CHLORAMPHENICOL PALMITATEantibacterial, antirickettsial

semisynthetic 530-43-8

2091 C05 Microsource 00307023 TESTOSTERONE androgen, antineoplasticmamallian male hormone

58-22-0

2091 C06 Microsource 01500173 CHLORAMPHENICOL HEMISUCCINATEantibacterial, antirickettsial, inhibits protein synthesis

semisynthetic982-57-0, 56-75-7 [chloramphenicol]

2091 C07 Microsource 00310006 HYDRASTININE HYDROCHLORIDEcardiotonic, uterine hemostatic

derivative of hydrastine (01501009)

4884-68-8, 6592-85-4 [hydrastinine]

2091 C08 Microsource 01500174 CHLORAMPHENICOLantibacterial, antirickettsial, inhibits protein synthesis

Streptomyces venezuelae

56-75-7

2091 C09 Microsource 00310035 SANGUINARINE SULFATEantineoplastic, antiplaque agent

Sanguinaria canadensis

5578-73-4

2091 C10 Microsource 01500175 CHLORCYCLIZINE HYDROCHLORIDE H1-antihistamine synthetic1620-21-9, 82-93-9 [base]

2091 C11 Microsource 00310039 alpha-TOCHOPHEROL vitamin Esoya, wheat germ and other plant oils

59-02-9

2091 C12 Microsource 01500177 CHLORHEXIDINEantibacterial (topical), disinfectant

synthetic3697-42-5, 55-56-1 [chlorhexidine]

2091 C13 Microsource 00310040 alpha-TOCHOPHERYL ACETATE vitamin E derivative 58-95-7

2091 C14 Microsource 01500178 CHLOROCRESOL antiinfectant synthetic 59-50-7

2091 C15 Microsource 00310050 QUININE ETHYL CARBONATE antimalarial semisynthetic 83-75-0

2091 C16 Microsource 01500179 CHLOROQUINE DIPHOSPHATEantimalarial, antiamebic, antirheumatic, intercalating agent

synthetic 54-05-7

2091 C17 Microsource 00330001 DACTINOMYCINantineoplastic, intercalating agent

Actinomyces spp 50-76-0

2091 C18 Microsource 01500180 CHLOROTHIAZIDE diuretic, antihypertensive synthetic 58-94-6

2091 C19 Microsource 00330002 MITOMYCIN C antineoplasticStreptomyces verticillatus

50-07-7

2091 C20 Microsource 01500181 CHLOROTRIANISENE estrogen synthetic 569-57-3

2091 C21 Microsource 00330018 DICHLORVOSinsecticide, cholinesterase inhibitor

synthetic 62-73-7

2091 C22 Microsource 01500182 CHLOROXYLENOLantibacterial, topical and urinary antiseptic

synthetic 88-04-0

2091 D03 Microsource 01500279 ERYTHROMYCIN ETHYLSUCCINATE antibacterial semisynthetic1264-62-6, 114-07-8 [erythromycin]

2091 D04 Microsource 01500390 METAPROTERENOL bronchodilator synthetic586-06-1, 5874-97-5 [metaproterenol sulfate]

2091 D05 Microsource 01500280 ERYTHROMYCIN antibacterialStreptomyces erythreus

114-07-8

2091 D06 Microsource 01500391 METHACHOLINE CHLORIDEcholinergic, diagnostic aid

synthetic62-51-1, 55-92-5 [methacholine]

2091 D07 Microsource 01500282 ESTRADIOL estrogen pregnancy urine 50-28-2

2091 D08 Microsource 01500394 METHENAMINE antibacterial (urinary) synthetic 100-97-0

2091 D09 Microsource 01500283 ESTRADIOL CYPIONATE estrogen semisynthetic 313-06-4

2091 D10 Microsource 01500395 METHICILLIN SODIUM antibacterial semisynthetic7246-14-2, 132-92-3 [anhydrous], 61-32-5 [methicillin]

2091 D11 Microsource 01500284 ESTRADIOL VALERATE estrogen semisynthetic 979-32-82091 D12 Microsource 01500396 METHIMAZOLE antihyperthyroid synthetic 60-56-0

2091 D13 Microsource 01500285 ESTRIOL estrogenmammalian hormone

50-27-1, 514-68-1 [as, succinate]

2091 D14 Microsource 01500397 METHOCARBAMOLmuscle relaxant (skeletal)

synthetic 532-03-6

Microsource1-US Drug Collection Page 2 of 24 Created 9/2015

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ICCB-L Plate

ICCB-L Well

VendorVendor

IDCompound Name Bioactivity Source CAS

2091 D15 Microsource 01500286 ESTRONE estrogenpregnacy urine, dates and Punica granatum seeds

53-16-7

2091 D16 Microsource 01500398 METHOTREXATE(+/-)antineoplastic, antirheumatic, folic acid antagonist

synthetic; AMETHOPTERIN

60388-53-6

2091 D17 Microsource 01500287 ETHACRYNIC ACID diuretic synthetic 58-54-8

2091 D18 Microsource 01500399 METHOXAMINE HYDROCHLORIDEalpha1 adrenoreceptor agonist, vasoconstrictor

synthetic61-16-5, 390-28-3 [methoxamine]

2091 D19 Microsource 01500288 ETHAMBUTOL HYDROCHLORIDEantibacterial (tuberculostatic)

synthetic1070-11-7, 74-55-5 [ethambutol]

2091 D20 Microsource 01500400 METHOXSALENantipsoriatic, pigmentation agent

amni visnaga 298-81-7

2091 D21 Microsource 01500291 ETHINYL ESTRADIOLestrogen, plus progestogen as oral contraceptive

semisynthetic 57-63-6

2091 D22 Microsource 01500401 METHSCOPOLAMINE BROMIDE anticholinergic semisynthetic 155-41-92091 E03 Microsource 00330062 TEMEFOS insecticide synthetic 3383-96-8

2091 E04 Microsource 01500183 CHLORPHENIRAMINE (S) MALEATE antihistaminic synthetic113-92-8, 132-22-9 [chlorpheniramine]

2091 E05 Microsource 00330071 LINDANE insecticidesynthetic; gamma-BHC

58-89-9

2091 E06 Microsource 01500184 CHLORPROMAZINE antiemetic, antipsychotic synthetic 50-53-3

2091 E07 Microsource 00330082 MITOTANEinsecticide, antineoplastic

synthetic 53-19-0

2091 E08 Microsource 01500185 CHLORPROPAMIDE antidiabetic synthetic 94-20-2

2091 E09 Microsource 00330086 DIBUTYL PHTHALATEplasticiser, suspect endocrine disruptor

synthetic 84-74-2

2091 E10 Microsource 01500186 CHLORTETRACYCLINE HYDROCHLORIDEantibacterial, antiamebic, Ca chelator, hepatotoxic; inhibits protein synthesis

Streptomyces aureofaciens

64-72-2

2091 E11 Microsource 01300027 IVERMECTIN antiparasitic semisynthetic 70288-86-7

2091 E12 Microsource 01500187 CHLORTHALIDONE diuretic, antihypertensive synthetic 77-36-1

2091 E13 Microsource 01300037 SODIUM NITROPRUSSIDE antihypertensive 13755-38-9

2091 E14 Microsource 01500188 CHLORZOXAZONEmuscle relaxant (skeletal)

synthetic 95-25-0

2091 E15 Microsource 01300038 SODIUM OXYBATE anestheticsynthetic; WY-3478, NSC-84223

502-85-2

2091 E16 Microsource 01500189 CICLOPIROX OLAMINE antifungal synthetic 41621-49-22091 E17 Microsource 01400151 ETHYL PARABEN antifungal synthetic 120-47-82091 E18 Microsource 01500190 CINOXACIN antibacterial synthetic 28657-80-9

2091 E19 Microsource 01400208 COUMARINantineoplastic, antiinflammatory, antihyperglycaemic

Coumarouna odorata, tonka beans, lavender oil

91-64-5

2091 E20 Microsource 01500191 CLEMASTINE antihistaminic synthetic 15686-51-82091 E21 Microsource 01600716 2,6-DI-t-BUTYL-4-METHYLPHENOL antioxidant synthetic; BHT 128-37-02091 E22 Microsource 01500192 CLIDINIUM BROMIDE anticholinergic synthetic 3485-62-9

2091 F03 Microsource 01500292 ETHIONAMIDEantibacterial, tuberculostatic

synthetic 536-33-4

2091 F04 Microsource 01500403 METHYLDOPA antihypertensive synthetic41372-08-1, 555-30-6 [anhydrous]

2091 F05 Microsource 01500293 ETHOPROPAZINE HYDROCHLORIDEantiparkinsonian, anticholinergic

synthetic1094-08-2, 522-00-9 [ethopropazine]

2091 F06 Microsource 01500406 METHYLPREDNISOLONE glucocorticoid semisynthetic 83-43-2

2091 F07 Microsource 01500295 EUCATROPINE HYDROCHLORIDEanticholinergic (opthalmic)

semisynthetic536-93-6, 100-91-4 [eucatropine]

2091 F08 Microsource 01500408 METHYLTHIOURACIL antithyroid agent synthetic 56-04-2

2091 F09 Microsource 01500296 EUGENOLanalgesic (topical), antiseptic, antifungal

common in plant essential oils

97-53-0

2091 F10 Microsource 01500410 METOCLOPRAMIDE HYDROCHLORIDE antiemetic synthetic54143-57-6, 7232-21-5 [anhydrous], 364-62-5 [metoclopramide]

2091 F11 Microsource 01500299 FLUDROCORTISONE ACETATE mineralocorticoid semisynthetic514-36-3, 127-31-1 [fludrocortisone]

2091 F12 Microsource 01500411 METOPROLOL TARTRATEantihypertensive, antianginal

synthetic56392-17-7, 37350-58-6 [metroprolol]

2091 F13 Microsource 01500300 FLUMETHAZONE PIVALATEglucocorticoid, antiinflammatory

semisynthetic2002-29-1, 2135-17-3 [flumethasone]

2091 F14 Microsource 01500412 METRONIDAZOLE antiprotozoal synthetic443-48-1, 69198-10-3 [metronidazole hydrochloride]

2091 F15 Microsource 01500302 FLUOCINOLONE ACETONIDEglucocorticoid, antiinflammatory

semisynthetic 67-73-2

2091 F16 Microsource 01500413 MICONAZOLE NITRATE antifungal (topical) synthetic22832-87-7, 22916-47-8 [miconazole]

2091 F17 Microsource 01500303 FLUOCINONIDEantiinflammatory, glucocorticoid

semisynthetic 356-12-7

2091 F18 Microsource 01500414 MINOCYCLINE HYDROCHLORIDE antibacterial semisynthetic13614-98-7, 10118-90-8 [minocycline]

Microsource1-US Drug Collection Page 3 of 24 Created 9/2015

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ICCB-L Plate

ICCB-L Well

VendorVendor

IDCompound Name Bioactivity Source CAS

2091 F19 Microsource 01500305 FLUOROURACILantineoplastic, pyrimidine antimetabolite

synthetic 51-21-8

2091 F20 Microsource 01500415 MINOXIDILantihypertensive, antialopecia agent

synthetic 38304-91-5

2091 F21 Microsource 01500308 FLURBIPROFENantiinflammatory, analgesic

synthetic 5104-49-4

2091 F22 Microsource 01500404 METHYLERGONOVINE MALEATE oxytocic semisynthetic57432-61-8, 7054-07-1 [replaced], 113-42-8 [methylergonovine]

2091 G03 Microsource 01500101 ACETAMINOPHEN analgesic, antipyretic synthetic 103-90-2

2091 G04 Microsource 01500193 CLINDAMYCIN HYDROCHLORIDEantibacterial, inhibits protein synthesis

semisynthetic; U-21251

21462-39-5, 58207-19-5 [monohydrate], 18323-44-9 [clindamycin]

2091 G05 Microsource 01500102 ACETAZOLAMIDEcarbonic anhydrase inhibitor, diuretic, antiglaucoma

synthetic 59-66-5

2091 G06 Microsource 01500196 CLOMIPHENE CITRATEgonad stimulating principle

synthetic50-41-9, 911-45-5 [clomiphene]

2091 G07 Microsource 01500103 ACETOHYDROXAMIC ACIDurease inhibitor, antiurolithic, antbacterial

synthetic 546-88-3

2091 G08 Microsource 01500198 CLONIDINE HYDROCHLORIDE antihypertensive synthetic4205-91-8, 4205-90-7 [clonidine]

2091 G09 Microsource 01500104 ACETYLCHOLINEantiarrhythmic, miotic, vasodilator (peripheral)

synthetic60-31-1, 51-84-3 [acetylcholine]

2091 G10 Microsource 01500200 CLOTRIMAZOLE antifungal synthetic 23593-75-12091 G11 Microsource 01500105 ACETYLCYSTEINE mucolytic synthetic 616-91-1

2091 G12 Microsource 01500201 CLOXACILLIN SODIUM antibacterial semisynthetic7081-44-9, 642-78-4 [anhydrous]

2091 G13 Microsource 01500107 ADENOSINEantiarrhythmic, cardiac depressant

widespread in living tissue

58-61-7

2091 G14 Microsource 01500202 CLOXYQUIN antibacterial, antifungal synthetic 130-16-5

2091 G15 Microsource 01500108 ALLOPURINOLantihyperuricemia, antigout, antiurolithic

synthetic 315-30-0

2091 G16 Microsource 01500205 COLCHICINEantimitotic, antigout agent

Colchicum autumnale

64-86-8

2091 G17 Microsource 01500109 ALVERINE CITRATE anticholinergic synthetic5560-59-8, 150-59-4 [alverine]

2091 G18 Microsource 01500206 COLISTIMETHATE SODIUM antibacterial Bacillus colistinus8068-28-8, 21362-08-3 [replaced]

2091 G19 Microsource 01500110 AMANTADINE HYDROCHLORIDE

antiviral, antiparkinsonian; treatment of drug-induced extrapyrimidal reactions

synthetic665-66-7, 768-94-5 [amantadine]

2091 G20 Microsource 01500207 CORTISONE ACETATE glucocorticoid semisynthetic50-04-4, 53-06-5 [cortisone]

2091 G21 Microsource 01500111 AMIKACIN SULFATE antibacterial semisynthetic39831-55-5, 37517-28-5 [amikacin]

2091 G22 Microsource 01500208 COTININE antidepressant Nicotiana tabacum486-56-6, 5695-98-7[fumarate]

2091 H03 Microsource 01500309 FURAZOLIDONE antibacterial NF-180; synthetic 67-45-82091 H04 Microsource 01500418 MOXALACTAM DISODIUM antibacterial semisynthetic 8031-09-2

2091 H05 Microsource 01500310 FUROSEMIDE diuretic, antihypertensive synthetic 54-31-9

2091 H06 Microsource 01500419 NADIDEalcohol and narcotic antagonist

synthetic 53-84-9

2091 H07 Microsource 01500311 FUSIDIC ACID antibacterial Fusidium spp 6990-06-3

2091 H08 Microsource 01500420 NAFCILLIN SODIUM antibacterial semisynthetic7177-50-6, 985-16-0 [anhydrous], 147-52-4 [nafcillin]

2091 H09 Microsource 01500312 GALLAMINE TRIETHIODIDEmuscle relaxant (skeletal)

synthetic65-29-2, 153-76-4 [gallamine]

2091 H10 Microsource 01500424 NAPHAZOLINE HYDROCHLORIDEadrenergic agonist, nasal decongestant

synthetic550-99-2, 835-31-4 [naphazoline]

2091 H11 Microsource 01500313 GEMFIBROZIL antihyperlipoproteinemic synthetic 25812-30-0

2091 H12 Microsource 01500425 NAPROXEN(+)antiinflammatory, analgesic, antipyretic

synthetic 22204-53-1

2091 H13 Microsource 01500314 GENTAMICIN SULFATE antibacterialMicromonospora spp

1405-41-0, 1403-66-3 [gentamicin]

2091 H14 Microsource 01500427 NEOMYCIN SULFATE antibacterialStreptomyces fradiae

1405-10-3, 1404-04-2 [neomycin]

2091 H15 Microsource 01500315 GENTIAN VIOLET antibacterial, anthelmintic synthetic 548-62-9

2091 H16 Microsource 01500433 NITROFURANTOIN antibacterial synthetic

67-20-9, 54-87-5 [nitrofurantoin sodium], 17140-81-7 [monohydrate]

2091 H17 Microsource 01500316 GLUCOSAMINE HYDROCHLORIDE antiarthritic

polysaccharides in bacteria, fungi, higher plants, invertebrates, vertebrates

3416-24-8

Microsource1-US Drug Collection Page 4 of 24 Created 9/2015

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ICCB-L Plate

ICCB-L Well

VendorVendor

IDCompound Name Bioactivity Source CAS

2091 H18 Microsource 01500428 NEOSTIGMINE BROMIDE cholinergic synthetic114-80-7, 59-99-4 [neostigmine]

2091 H19 Microsource 01500319 GRAMICIDIN antibacterial Bacillus brevis 1405-97-6

2091 H20 Microsource 01500431 NIFEDIPINEantianginal, antihypertensive

synthetic 21829-25-4

2091 H21 Microsource 01500321 GUAIFENESIN expectorant synthetic 93-14-1

2091 H22 Microsource 01500430 NIACINantihyperlipidemic, vitamin (enzyme cofactor)

widespread in the plant and fungal kingdom

59-67-6

2091 I03 Microsource 01500112 AMILORIDE HYDROCHLORIDENa+ channel inhibitor, diuretic

synthetic17440-83-4, 2016-88-8 [anhydrous], 2609-46-3 [amiloride]

2091 I04 Microsource 01500209 CRESOL antiinfectant coal tar 1319-77-32091 I05 Microsource 01500113 POTASSIUM p-AMINOBENZOATE ultraviolet screen synthetic 150-13-0 (acid)

2091 I06 Microsource 01500210 CROMOLYN SODIUM antiasthmatic, antiallergy synthetic15826-37-6, 16110-51-3 [cromolyn]

2091 I07 Microsource 01500114 AMINOCAPROIC ACID hemostatic synthetic 60-32-22091 I08 Microsource 01500211 CYCLIZINE H1 antihistamine synthetic 82-92-8

2091 I09 Microsource 01500115 AMINOGLUTETHIMIDEaromatase inhibitor, antineoplastic, testosterone suppressant

synthetic 125-84-8

2091 I10 Microsource 01500212 CYCLOPENTOLATE HYDROCHLORIDE mydriatic synthetic5870-29-1, 512-15-2 [cyclopentolate]

2091 I11 Microsource 01500116 AMINOSALICYLATE SODIUMantibacterial, tuberculostatic

synthetic 6018-19-5

2091 I12 Microsource 01500213 CYCLOPHOSPHAMIDE HYDRATEantineoplastic, alkylating agent

synthetic6055-19-2, 50-18-0 [anhydrous]

2091 I13 Microsource 01500117 AMITRIPTYLINE HYDROCHLORIDE antidepressant synthetic 549-18-8

2091 I14 Microsource 01500215 CYCLOSERINEantibacterial (tuberculostatic)

Streptomyces spp 68-41-7

2091 I15 Microsource 01500119 AMODIAQUINE DIHYDROCHLORIDE antimalarial synthetic6398-98-7, 69-44-3 [anhydrous], 86-42-0 [amodiaquine]

2091 I16 Microsource 01500216 CYPROTERONE ACETATE antiandrogen synthetic 427-51-0

2091 I17 Microsource 01500120 AMOXICILLIN antibacterial semisynthetic61336-70-7, 26787-78-0 [anhydrous]

2091 I18 Microsource 01500217 CYTARABINEantineoplastic, antiviral, antimetabolite

synthetic 147-94-4

2091 I19 Microsource 01500122 AMPHOTERICIN B antifungalStreptomycetes nodosus

1397-89-3

2091 I20 Microsource 01500218 DACARBAZINE antineoplastic synthetic 4342-03-4

2091 I21 Microsource 01500123 AMPICILLIN SODIUM antibacterial semisynthetic69-52-3, 69-53-4 [ampicillin]

2091 I22 Microsource 01500220 DANAZOLanterior pituitary suppressant

synthetic 17230-88-5

2091 J03 Microsource 01500322 GUANABENZ ACETATE antihypertensive synthetic 23256-50-02091 J04 Microsource 01500434 NITROFURAZONE antiinfective (topical) synthetic 59-87-0

2091 J05 Microsource 01500323 GUANETHIDINE SULFATEantihypertensive, mitotic agent

synthetic60-02-6, 55-65-2 [guanethidine]

2091 J06 Microsource 01500435 NITROMIDE antibacterial, coccidiostat synthetic 121-81-3

2091 J07 Microsource 01500324 HALAZONE antiinfectant synthetic 80-13-7

2091 J08 Microsource 01500436 NOREPINEPHRINEadrenergic agonist, antihypotensive

synthetic69815-49-2, 51-40-1 [anhydrous], 51-41-2 [norepinephrine]

2091 J09 Microsource 01500325 HALOPERIDOLantidyskinetic, antipsychotic

synthetic 52-86-8

2091 J10 Microsource 01500437 NORETHINDRONE progestogen synthetic 68-22-4

2091 J11 Microsource 01500327 HETACILLIN POTASSIUM antibacterial semisynthetic5321-32-4, 3511-16-8 [hetacillin]

2091 J12 Microsource 01500438 NORETHINDRONE ACETATEOral contraceptive (in combination with estrogen)

synthetic 51-98-9

2091 J13 Microsource 01500328 HEXACHLOROPHENE antiinfective (topical) synthetic 70-30-4

2091 J14 Microsource 01500439 NORETHYNODREL

progestogen, in combination with estrogen as oral contraceptive

synthetic 68-23-5

2091 J15 Microsource 01500330 HEXYLRESORCINOLanthelmintic, topical antiseptic

synthetic 136-77-6

2091 J16 Microsource 01500440 NORFLOXACIN antibacterial synthetic 70458-96-7

2091 J17 Microsource 01500331 HISTAMINE DIHYDROCHLORIDE

H receptor agonist, induces edema in mammalian tissues; gastric secretion stimulant

Claviceps purpurea, many plants and animals

51-45-6 [histamine]

2091 J18 Microsource 01500441 NORGESTREL progestogen synthetic 6533-00-2

2091 J19 Microsource 01500332 HOMATROPINE BROMIDEanticholinergic (opthalmic)

semisynthetic51-56-9, 87-00-3 [homatropine]

2091 J20 Microsource 01500442 NORTRIPTYLINE antidepressant synthetic894-71-3, 72-69-5 [nortriptyline]

2091 J21 Microsource 01500333 HOMATROPINE METHYLBROMIDEanticholinergic (opthalmic)

semisynthetic80-49-9, 87-00-3 [homatropine]

Microsource1-US Drug Collection Page 5 of 24 Created 9/2015

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ICCB-L Plate

ICCB-L Well

VendorVendor

IDCompound Name Bioactivity Source CAS

2091 J22 Microsource 01500443 NOSCAPINE HYDROCHLORIDE antitussiveCorydalis cava and Papaver spp

912-60-7, 128-62-1 [noscapine]

2091 K03 Microsource 01500124 AMPROLIUM coccidiostat synthetic 121-25-5

2091 K04 Microsource 01500222 DAPSONEantibacterial, leprostatic, dermatitis herpetiformis suppressant

synthetic 80-08-0

2091 K05 Microsource 01500126 ANTAZOLINE PHOSPHATE antihistaminic synthetic154-68-7, 91-75-8 [antazoline]

2091 K06 Microsource 01500223 DAUNORUBICIN antineoplastic

Streptomyces peucetius; FI-6339, NDC-0082-4155, RP-13057

20830-81-3

2091 K07 Microsource 01500127 ANTHRALIN antipsoriatic synthetic 480-22-8, 1143-38-0

2091 K08 Microsource 01500224 DEFEROXAMINE MESYLATE chelating agent (Fe & Al) Strptomyces pilosus138-14-7, 70-51-9 [deferoxamine]

2091 K09 Microsource 01500128 ANTIPYRINE analgesic synthetic 60-80-02091 K10 Microsource 01500225 SODIUM DEHYDROCHOLATE choleretic semisynthetic 145-41-5

2091 K11 Microsource 01500129 APOMORPHINE HYDROCHLORIDE emetic synthetic41372-20-7, 314-19-2 [anhydrous], 58-00-4 [apomorphine]

2091 K12 Microsource 01500226 DEMECLOCYCLINE HYDROCHLORIDE antibacterialStreptomyces aureofaiens

127-33-3

2091 K13 Microsource 01500130 ASPIRINanalgesic, antipyretic, antiinflammatory

synthetic 50-78-2

2091 K14 Microsource 01500227 DESIPRAMINE HYDROCHLORIDE antidepressant synthetic58-28-6, 50-47-5 [desipramine]

2091 K15 Microsource 01500131 ATROPINE SULFATE anticholinergic, mydriaticAtropa and Datura spp

51-55-8, 5908-99-6 [atropine sulfate], 55-48-1 [anhydrous]

2091 K16 Microsource 01500230 DEXAMETHASONE glucocorticoid semisynthetic 50-02-22091 K17 Microsource 01500132 AUROTHIOGLUCOSE antirheumatic synthetic 12192-57-3

2091 K18 Microsource 01500232 DEXAMETHASONE SODIUM PHOSPHATEglucocorticoid, antiinflammatory

semisynthetic

2392-39-4, 312-93-6 [dexamethasone 21-(dihydrogen phosphate)]

2091 K19 Microsource 01500133 AZATHIOPRINEimmunosuppressant, antineoplastic, antirheumatic

synthetic 446-86-6

2091 K20 Microsource 01500233 DEXTROMETHORPHAN HYDROBROMIDE antitussive synthetic6700-34-1, 125-69-9 [anhydrous], 125-71-3 [dextromethorphan]

2091 K21 Microsource 01500134 BACITRACIN antibacterialBacillus licheniformis and B subtilis

1405-87-4

2091 K22 Microsource 01500235 DIBENZOTHIOPHENE keratolytic synthetic 132-65-0

2091 L03 Microsource 01500334 HYDRALAZINE HYDROCHLORIDE antihypertensive semisynthetic304-20-1, 86-54-4 [hydralazine]

2091 L04 Microsource 01500444 NOVOBIOCIN SODIUM antibacterialStreptomyces niveus and S griseus

1476-53-5, 303-81-1 [novobiocin]

2091 L05 Microsource 01500335 HYDROCHLOROTHIAZIDE diuretic semisynthetic 58-93-52091 L06 Microsource 01500445 NYLIDRIN HYDROCHLORIDE vasodilator (peripheral) synthetic 849-55-8

2091 L07 Microsource 01500338 HYDROCORTISONE ACETATEglucocorticoid, antiinflammatory

semisynthetic 50-03-3

2091 L08 Microsource 01500446 NYSTATINantifungal, binds to membrane sterols

Streptomyces noursei

114-90-9

2091 L09 Microsource 01500339 HYDROCORTISONE HEMISUCCINATE glucocorticoid semisynthetic83784-20-7, 2203-97-6 [anhydrous]

2091 L10 Microsource 01500447 ORPHENADRINE CITRATEmuscle relaxant (skeletal), antihistaminic

synthetic4682-36-4, 83-98-7 [orphenadrine]

2091 L11 Microsource 01500340HYDROCORTISONE PHOSPHATE TRIETHYLAMINE

glucocorticoid semisynthetic3863-59-0 [cortisol 21-(dihydrogen phosphate)]

2091 L12 Microsource 01500448 OXACILLIN SODIUM antibacterial semisynthetic7240-38-2, 1173-88-2 [anhydrous], 66-79-5 [oxacillin]

2091 L13 Microsource 01500341 HYDROFLUMETHIAZIDE antihypertensive, diuretic synthetic 135-09-1

2091 L14 Microsource 01500450 OXIDOPAMINE HYDROCHLORIDEadrenergic agonist (opthalmic)

synthetic 1199-18-4

2091 L15 Microsource 01500343 HYDROXYPROGESTERONE CAPROATE progestogen semisynthetic630-56-8, 68-96-2 [hydroxyprogesterone]

2091 L16 Microsource 01500451 OXYBENZONE ultraviolet screen synthetic 131-57-7

2091 L17 Microsource 01500344 HYDROXYUREAantineoplastic, inhibits ribonucleoside diphosphate reductase

synthetic 127-07-1

2091 L18 Microsource 01500453 OXYMETAZOLINE HYDROCHLORIDEadrenergic agonist, nasal decongestant

synthetic2315-02-8, 1491-59-4 [oxymetazoline]

2091 L19 Microsource 01500345 HYDROXYZINE PAMOATE anxiolytic, antihistaminic synthetic10246-75-0, 68-88-2 [hydroxyzine]

2091 L20 Microsource 01500455 OXYPHENBUTAZONE antiinflammatory synthetic7081-38-1, 129-20-4 [anhydrous]

Microsource1-US Drug Collection Page 6 of 24 Created 9/2015

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ICCB-L Plate

ICCB-L Well

VendorVendor

IDCompound Name Bioactivity Source CAS

2091 L21 Microsource 01500346 HYOSCYAMINE anticholinergic, analgesicAtropa, Datura and Hyoscyamus spp

101-31-5

2091 L22 Microsource 01500456 OXYQUINOLINE HEMISULFATE antiinfectant synthetic 148-24-3

2091 M03 Microsource 01500135 BACLOFENmuscle relaxant (skeletal)

synthetic 1134-47-0

2091 M04 Microsource 01500236 DIBUCAINE HYDROCHLORIDE anesthetic (local) synthetic61-12-1, 85-79-0 [dibucaine]

2091 M05 Microsource 01500136 BECLOMETHASONE DIPROPIONATEantiasthmatic, topical antiinflammatory

synthetic5534-09-8, 4419-39-0 [beclomethasone]

2091 M06 Microsource 01500237 DICLOFENAC SODIUM antiinflammatory synthetic 15307-79-6

2091 M07 Microsource 01500137 BENSERAZIDE HYDROCHLORIDE decarboxylase inhibitorcomponent of Madopa (Hoffmann-LaRoche)

322-35-0

2091 M08 Microsource 01500238 DICLOXACILLIN SODIUM antibacterial semisynthetic13412-64-1, 343-55-5 [anhydrous], 3116-76-5 [dicloxacillin]

2091 M09 Microsource 01500138 BENZETHONIUM CHLORIDE antiinfective (topical) synthetic 121-54-02091 M10 Microsource 01500239 DICUMAROL anticoagulant synthetic 66-76-22091 M11 Microsource 01500139 BENZOCAINE anesthetic (topical) synthetic 94-09-7

2091 M12 Microsource 01500240 DICYCLOMINE HYDROCHLORIDE anticholinergic synthetic67-92-5, 77-19-0 [dicyclomine]

2091 M13 Microsource 01500141 BENZTHIAZIDE diuretic, antihypertensive synthetic 91-33-8

2091 M14 Microsource 01500241 DIENESTROL estrogen synthetic84-17-3, 13029-44-2 [//E,E//]

2091 M15 Microsource 01500142 BENZTROPINE anticholinergic synthetic132-17-2, 86-13-5 [benztropine]

2091 M16 Microsource 01500242 DIETHYLCARBAMAZINE CITRATE anthelmintic synthetic1642-54-2, 90-89-1 [diethylcarbamazine]

2091 M17 Microsource 01500143 beta-CAROTENE provitamin Aprovitamin A; widespread in plants and animals

7235-40-7

2091 M18 Microsource 01500244 DIETHYLSTILBESTROL estrogen synthetic 56-53-1

2091 M19 Microsource 01500146 BETHANECHOL CHLORIDE cholinergic synthetic590-63-6, 674-38-4 [bethanechol]

2091 M20 Microsource 01500245 DIFLUNISALanalgesic, antiinflammatory

synthetic 22494-42-4

2091 M21 Microsource 01505430 FLUROTHYLcentral stimulant, convulsant

synthetic; SK&F-6539

333-36-8

2091 M22 Microsource 01500246 DIGITOXIN inotropic, cardiotonic Digitalis spp 71-63-6

2091 N03 Microsource 01500347 IBUPROFEN antiinflammatory synthetic15687-27-1, 58560-75-1 [(+/-) mixture]

2091 N04 Microsource 01500457 OXYTETRACYCLINE antibacterialStreptomyces rimosus

6153-64-6, 79-57-2 [anhydrous]

2091 N05 Microsource 01500348 IMIPRAMINE HYDROCHLORIDE antidepressant synthetic113-52-0, 50-49-7 [imipramine]

2091 N06 Microsource 01500459 PAPAVERINE HYDROCHLORIDEmuscle relaxant (smooth), cerebral vasodilator

Papaver somniferum, Rauwolfia serpentina

61-25-6, 58-74-2 [papaverine]

2091 N07 Microsource 01500349 INDAPAMIDE diuretic, antihypertensive synthetic 26807-65-8

2091 N08 Microsource 01500460 PARACHLOROPHENOLtopical antibacterial (topical)

synthetic 106-48-9

2091 N09 Microsource 01500350 INDOMETHACINantiinflammatory, antipyretic, analgesic

synthetic 53-86-1

2091 N10 Microsource 01500462 PARGYLINE HYDROCHLORIDE antihypertensive synthetic306-07-0, 555-57-7 [pargyline]

2091 N11 Microsource 01500351 INDOPROFENanalgesic, antiinflammatory

synthetic 31842-01-0

2091 N12 Microsource 01500465 PENICILLIN G POTASSIUM antibacterial Penicillium spp69-57-8, 61-33-6 [penicillin, G]

2091 N13 Microsource 01500352 INOSITOL growth factorlipotropic polyol widely distributed in plants and animals

87-89-8

2091 N14 Microsource 01500467 PENICILLIN V POTASSIUM antibacterial semisynthetic132-98-9, 87-08-1 [penicillin, V]

2091 N15 Microsource 01500353 IODOQUINOL antiamebic synthetic 83-73-82091 N16 Microsource 01500472 PHENACEMIDE anticonvulsant synthetic 63-98-9

2091 N17 Microsource 01500354 IPRATROPIUM BROMIDEbronchodilator, antiarrhythmic

synthetic66985-17-9, 22254-24-6 [anhydrous]

2091 N18 Microsource 01500473 PHENAZOPYRIDINE HYDROCHLORIDE analgesic synthetic136-40-3, 94-78-0 [phenazopyridine]

2091 N19 Microsource 01500355 ISONIAZIDantibacterial, tuberculostatic

synthetic 54-85-3

2091 N20 Microsource 01500476 PHENELZINE SULFATE antidepressant synthetic156-51-4, 51-71-8 [phenelzine]

2091 N21 Microsource 01500356 ISOPROPAMIDE IODIDE anticholinergic synthetic71-81-8, 7492-32-2 [isopropamide]

2091 N22 Microsource 01500477 PHENINDIONE anticoagulant synthetic 83-12-52091 O03 Microsource 01500147 BISACODYL cathartic synthetic 603-50-9

2091 O04 Microsource 01500247 DIGOXIN cardiac stimulantDigitalis lanata or D. orientalis Lam., Scrophulariaceae

20830-75-5

Microsource1-US Drug Collection Page 7 of 24 Created 9/2015

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ICCB-L Plate

ICCB-L Well

VendorVendor

IDCompound Name Bioactivity Source CAS

2091 O05 Microsource 01500148 BITHIONATE SODIUM anthelmintic, antiseptic synthetic 97-18-7

2091 O06 Microsource 01500249 DIHYDROSTREPTOMYCIN SULFATEantibacterial, tuberculostatic

Streptomyces humidus

5490-27-7, 128-46-1 [dihydrostreptomycin]

2091 O07 Microsource 01500151 BROMOCRIPTINE MESYLATEprolactin inhibitor, antiparkinsonian

semisynthetic22260-51-1, 25614-03-3 [bromocriptine]

2091 O08 Microsource 01500251 DIMENHYDRINATE antiemetic synthetic 523-87-5

2091 O09 Microsource 01500152 BUSULFANantineoplastic, alkylating agent

synthetic 55-98-1

2091 O10 Microsource 01500253 DIMETHADIONE anticonvulsant synthetic 695-53-4

2091 O11 Microsource 01500155 CAFFEINE CNS stimulantCofea, Theobroma, Camelia and Cola spp

58-08-2, 5743-12-4 [monohydrate]

2091 O12 Microsource 01500255 DIOXYBENZONE ultraviolet screen synthetic 131-53-3

2091 O13 Microsource 01500156 CAMPHOR (1R)analgesic, antiinfective, antipruritic

Cinnamomum camphora

464-49-3; 76-22-2

2091 O14 Microsource 01500256 DIPHENHYDRAMINE HYDROCHLORIDE antihistaminic synthetic 147-24-0

2091 O15 Microsource 01500157 CAPREOMYCIN SULFATEantibacterial, tuberculostatic

Streptomyces capreolis

1405-37-4, 11003-38-6 [capreomycin]

2091 O16 Microsource 01500258 DIPHENYLPYRALINE HYDROCHLORIDE antihistaminic synthetic132-18-3 147-20-6 [diphenylpyraline]

2091 O17 Microsource 01500158 CARBACHOL cholinergic, miotic synthetic 51-83-22091 O18 Microsource 01500259 DIPYRIDAMOLE coronary vasodilator synthetic 58-32-2

2091 O19 Microsource 01500159 CARBAMAZEPINE analgesic, anticonvulsant synthetic 298-46-4

2091 O20 Microsource 01500260 PYRITHIONE ZINCantibacterial, antifungal, antiseborrheic

synthetic 13463-41-7

2091 O21 Microsource 01500160 CARBENICILLIN DISODIUM antibacterial semisynthetic4800-94-6, 4697-36-3 [carbenicillin]

2091 O22 Microsource 01500262 DISULFIRAM alcohol antagonist synthetic 97-77-8

2091 P03 Microsource 01500357 ISOPROTERENOL HYDROCHLORIDE bronchodilator synthetic51-30-9, 7683-59-2 [isoproterenol]

2091 P04 Microsource 01500478 PHENIRAMINE MALEATE antihistaminic synthetic132-20-7, 86-21-5 [pheniramine]

2091 P05 Microsource 01500358 ISOSORBIDE DINITRATE antianginal semisynthetic 87-33-22091 P06 Microsource 01500480 PHENOLPHTHALEIN cathartic synthetic 77-09-8

2091 P07 Microsource 01500359 ISOXSUPRINE HYDROCHLORIDE vasodilator synthetic579-56-6, 395-28-8 [isoxsuprine]

2091 P08 Microsource 01500482 PHENYLBUTAZONE antiinflammatory synthetic 50-33-9

2091 P09 Microsource 01500360 KANAMYCIN A SULFATE antibacterialStreptomyces kanamyceticus

25389-94-0, 133-92-6 [replaced], 59-01-8 [kanamycin]

2091 P10 Microsource 01500483 PHENYLEPHRINE HYDROCHLORIDE mydriatic, decongestant synthetic61-76-7, 59-42-7 [phenylephrine]

2091 P11 Microsource 01500362 KETOCONAZOLE antifungal synthetic 65277-42-1

2091 P12 Microsource 01500484PHENYLPROPANOLAMINE HYDROCHLORIDE

vasoconstrictor, decongestant, anorexic

synthetic 154-41-6

2091 P13 Microsource 01500365 LEVONORDEFRIN vasoconstrictor synthetic829-74-3, 18829-78-2 [replaced]

2091 P14 Microsource 01500485 PHENYTOIN SODIUManticonvulsant, antieleptic

synthetic630-93-3, 57-41-0 [phenytoin]

2091 P15 Microsource 01500372 MAFENIDE HYDROCHLORIDE antibacterial synthetic 138-39-6

2091 P16 Microsource 01500486 PHYSOSTIGMINE SALICYLATEcholinergic, anticholinesterase, miotic

Physostigma venenosum

57-64-7, 57-47-6 [physostigmine]

2091 P17 Microsource 01500373 MAPROTILINE HYDROCHLORIDE antidepressant synthetic10347-81-6, 10262-69-8 (maprotiline)

2091 P18 Microsource 01500487 PILOCARPINE NITRATEantiglaucoma agent, miotic

Pilocarpus spp148-72-1, 92-13-7 [pilocarpine]

2091 P19 Microsource 01500374 MECAMYLAMINE HYDROCHLORIDE antihypertensive synthetic826-39-1, 60-40-2 [mecamylamine]

2091 P20 Microsource 01500488 PINDOLOL

antihypertensive, antianginal, antiarrhythmic, antiglaucoma agent

synthetic 13523-86-9

2091 P21 Microsource 01500364 LEUCOVORIN CALCIUMantianemic, antidote to folic acid antagonists

synthetic 1492-18-8

2091 P22 Microsource 01500489 PIPERACILLIN SODIUM antibacterial semisynthetic59703-84-3, 66258-76-2 [piperacillin], 61477-96-1 [anhydrous]

2092 A03 Microsource 01500490 PIPERAZINE anthelmintic synthetic110-85-0, 144-29-6 [anhydrous], 41372-10-5 [piperazine citrate]

2092 A04 Microsource 01500592 TRIHEXYPHENIDYL HYDROCHLORIDEanticholinergic, antiparkinsonian

synthetic 52-49-3

2092 A05 Microsource 01500491 PIROXICAM antiinflammatory synthetic 36322-90-4

2092 A06 Microsource 01500593 TRIMEPRAZINE TARTRATE antipruritic synthetic4330-99-8, 41375-66-0 [replaced], 84-96-8 [trimeprazine]

2092 A07 Microsource 01500492 POLYMYXIN B SULFATE antibacterial Bacillus polymyxa1405-20-5, 1404-26-8 [polymyxin B]

Microsource1-US Drug Collection Page 8 of 24 Created 9/2015

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VendorVendor

IDCompound Name Bioactivity Source CAS

2092 A08 Microsource 01500594 TRIMETHOBENZAMIDE HYDROCHLORIDE antiemetic synthetic554-92-7, 138-56-7 [trimethobenzamide]

2092 A09 Microsource 01500494 PRAZIQUANTEL anthelmintic synthetic 55268-74-12092 A10 Microsource 01500595 TRIMETHOPRIM antibacterial synthetic 738-70-5

2092 A11 Microsource 01500495 PRAZOSIN HYDROCHLORIDE antihypertensive synthetic19237-84-4, 19216-56-9 [prazosin]

2092 A12 Microsource 01500596 TRIOXSALENmelanizing agent, antipsoriatic

synthetic 3902-71-4

2092 A13 Microsource 01500496 PREDNISOLONE glucocorticoid semisynthetic50-24-8 [anhydrous], 52438-85-4 [sesquihydrate]

2092 A14 Microsource 01500597 TRIPELENNAMINE CITRATE antihistaminic synthetic6138-56-3, 91-81-6 [tripelennamine]

2092 A15 Microsource 01500497 PREDNISOLONE ACETATE glucocorticoid semisynthetic 52-21-1

2092 A16 Microsource 01500598 TRIPROLIDINE HYDROCHLORIDE antihistaminic synthetic6138-79-0, 550-70-9 [anhydrous], 486-12-4 [triprolidine]

2092 A17 Microsource 01500499 PREDNISONE glucocorticoid semisynthetic 53-03-2

2092 A18 Microsource 01500599 TROPICAMIDEanticholinergic (opthalmic)

synthetic 1508-75-4

2092 A19 Microsource 01500500 PRIMAQUINE DIPHOSPHATE antimalarial synthetic63-45-6, 90-34-6 [primaquine]

2092 A20 Microsource 01500600 TRYPTOPHANantidepressant, nutrient; LD50(rat) 1634 mg/kg ip

many plants, animal protein

73-22-3 ['L']

2092 A21 Microsource 01500501 PRIMIDONE anticonvulsant synthetic 125-33-7

2092 A22 Microsource 01500601 TUAMINOHEPTANE SULFATE adrenergic agonist synthetic6411-75-2, 123-82-0 [tuaminoheptane]

2092 B03 Microsource 01501008 FENBUFEN antiinflammatory synthetic 36330-85-52092 B04 Microsource 01502040 CEFMETAZOLE SODIUM antibacterial semisynthetic 56796-39-52092 B05 Microsource 01501010 FENOFIBRATE antihyperlipidemic synthetic 49562-28-9

2092 B06 Microsource 01502041 CEFAMANDOLE NAFATE antibacterial semisynthetic42540-40-9, 34444-01-4 [cefamandole]

2092 B07 Microsource 01501011 FENOPROFEN antiinflammatory synthetic 31879-05-7

2092 B08 Microsource 01502042 CEFOPERAZONE SODIUM antibacterial semisynthetic62893-20-3, 62893-19-0 [cefoperazone]

2092 B09 Microsource 01501015 FLUFENAMIC ACIDantiinflammatory, analgesic

synthetic 530-78-9

2092 B10 Microsource 01502044 OFLOXACIN antibacterial synthetic 82419-36-12092 B11 Microsource 01501016 FENBENDAZOLE anthelmintic synthetic 43210-67-92092 B12 Microsource 01502046 BEZAFIBRATE antihyperlipidemic synthetic 41859-67-0

2092 B13 Microsource 01501021 FENSPIRIDE HYDROCHLORIDEantiinflammatory, bronchodilator

synthetic5053-08-7, 5053-06-5 [fenspiride]

2092 B14 Microsource 01502047 LIOTHYRONINE (L- isomer) SODIUM thyroid hormone synthetic; L-isomer55-06-1, 6893-02-3 [liothyronine]

2092 B15 Microsource 01501110 MEBENDAZOLE anthelmintic synthetic 31431-39-7

2092 B16 Microsource 01502006 CARPROFENantiinflammatory, analgesic

synthetic 53716-49-7

2092 B17 Microsource 01501103 MEFENAMIC ACIDantiinflammatory, analgesic

synthetic 61-68-7

2092 B18 Microsource 01502053 ALRESTATINaldose reductase inhibitor

synthetic; AY-22284A

51411-04-2, 51876-97-2 [alrestatin sodium]

2092 B19 Microsource 01501104 METHACYCLINE HYDROCHLORIDE antibacterial semisynthetic3963-95-9, 914-00-1 [methacycline]

2092 B20 Microsource 01502084 PROADIFEN HYDROCHLORIDEcytochrome P450 inhibitor, Ca antagonist

synthetic; SKF-525A 78997-40-7

2092 B21 Microsource 01501105 PUROMYCIN HYDROCHLORIDEantineoplastic, antiprotozoal

Streptomyces alboniger

58-58-2, 53-79-2 [puromycin]

2092 B22 Microsource 01502106 CARBOPLATINantineoplastic, convulsant

synthetic 41575-94-4

2092 C03 Microsource 01500502 PROBENECID uricosuric synthetic 57-66-9

2092 C04 Microsource 01500602 TUBOCURARINE CHLORIDEmuscle relaxant (skeletal)

Chondodendron spp

6989-98-6, 57-94-3 [anhydrous], 41354-45-4 [replaced], 57-95-4 [tubocurarine]

2092 C05 Microsource 01500503 PROCAINAMIDE HYDROCHLORIDE antiarrhythmic synthetic614-39-1, 51-06-9 [procainamide]

2092 C06 Microsource 01500603 TYROTHRICINtopical antibacterial (topical)

Bacillus aneurinolyticus; mixture of gramicidins & tyrocidines (tyrocidine A shown)

1404-88-2

2092 C07 Microsource 01500504 PROCAINE HYDROCHLORIDE anesthetic (local) synthetic51-05-8, 59-46-1 [procaine]

2092 C08 Microsource 01500604 UREA diuretic synthetic 57-13-6

2092 C09 Microsource 01500505 PROCHLORPERAZINE EDISYLATEantiemetic, antipsychotic, treatment of vertigo

synthetic

1257-78-9, 84-02-6 [prochlorperazine maleate], 58-38-8 [prochlorperazine]

2092 C10 Microsource 01500605 URSODIOLanticholelithogenic; LD50(rat) 890 mg/kg ip

bear bile 128-13-2

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VendorVendor

IDCompound Name Bioactivity Source CAS

2092 C11 Microsource 01500507 PROCYCLIDINE HYDROCHLORIDE anticholinergic synthetic1508-76-5, 77-37-2 [procyclidine]

2092 C12 Microsource 01500606 VALPROATE SODIUM anticonvulsant synthetic1069-66-5, 99-66-1 [valproic acid]

2092 C13 Microsource 01500508 PROGESTERONE progestogen semisynthetic 57-83-0

2092 C14 Microsource 01500607 VANCOMYCIN HYDROCHLORIDE antibacterialStreptomyces orientalis

1404-93-9, 1404-90-6 [vancomycin]

2092 C15 Microsource 01500509 PROMAZINE HYDROCHLORIDE antipsychotic synthetic53-60-1, 58-40-2 [promazine]

2092 C16 Microsource 01500609 VIDARABINE antiviral synthetic24356-66-9, 5536-17-4 [anhydrous]

2092 C17 Microsource 01500510 PROMETHAZINE HYDROCHLORIDE antihistaminic synthetic58-33-3, 60-87-7 [promethazine]

2092 C18 Microsource 01500611 VINBLASTINE SULFATEantineoplastic, spindle poison

Vinca rosea143-67-9, 865-21-4 [vinblastine]

2092 C19 Microsource 01500511 PROPANTHELINE BROMIDE anticholinergic synthetic50-34-0, 298-50-0 [propantheline]

2092 C20 Microsource 01500613 WARFARINanticoagulant, rodenticide

synthetic

81-81-2, 2610-86-8 [warfarin potassium], 129-06-6 [warfarin sodium]

2092 C21 Microsource 01500514 DEXPROPRANOLOL HYDROCHLORIDEantihypertensive, antianginal, antiarrhythmic

synthetic 13071-11-9

2092 C22 Microsource 01500614 XYLOMETAZOLINE HYDROCHLORIDEadrenergic agonist, nasal decongestant

synthetic1218-35-5, 526-36-3 [xylometazoline]

2092 D03 Microsource 01501108 MEFEXAMIDE stimulant (central) synthetic 1227-61-8

2092 D04 Microsource 01502107 CISPLATINantineoplastic, convulsant

synthetic 15663-27-1

2092 D05 Microsource 01501109 PROBUCOL antihyperlipidemic synthetic 23288-49-5

2092 D06 Microsource 01502109 ZIDOVUDINE [AZT]RT transferase inhibitor, antiviral

synthetic 30516-87-1

2092 D07 Microsource 01501115 NALBUPHINE HYDROCHLORIDEanalgesic, narcotic antagonist

synthetic23277-43-2, 20594-83-6 [nalbuphine]

2092 D08 Microsource 01502111 AZACITIDINEantineoplastic, pyrimidine antimetabolite

synthetic; U-18496; NSC-102816

320-67-2

2092 D09 Microsource 01501117 MEBEVERINE HYDROCHLORIDE muscle relaxant (smooth) synthetic2753-45-9, 3625-06-7 [mebeverine]

2092 D10 Microsource 01502112 CYCLOHEXIMIDE protein synthesis inhibitor synthetic 66-81-9

2092 D11 Microsource 01501118 MECLOCYCLINE SULFOSALICYLATE antibacterialsemisynthetic; GS-2989, NSC-78502

73816-42-9, 2013-58-3 [meclocycline]

2092 D12 Microsource 01502113 AZASERINEantineoplastic, amino acid antagonist

Streptomyces fragilis 115-02-6

2092 D13 Microsource 01501119 PROGLUMIDE anticholinergic synthetic 6620-60-62092 D14 Microsource 01502127 TINIDAZOLE antiprotozoal synthetic 19387-91-8

2092 D15 Microsource 01501120 MINAPRINE HYDROCHLORIDE psychotropic synthetic25953-17-7, 25905-77-5 [minaprine]

2092 D16 Microsource 01502150 CARBIDOPAdecarboxylase inhibitor, antiparkinsonism

synthetic38821-49-7, 28860-95-9 [anhydrous]

2092 D17 Microsource 01501121 MEMANTINE HYDROCHLORIDEmuscle relaxant (skeletal)

synthetic 19982-08-2

2092 D18 Microsource 01502195 PIRACETAM antinauseant synthetic 7491-74-92092 D19 Microsource 01501127 ATENOLOL beta adrenergic blocker synthetic 29122-68-72092 D20 Microsource 01502196 ETHOSUXIMIDE anticonvulsant synthetic 77-67-8

2092 D21 Microsource 01501128 CAPSAICINanalgesic (topical), depletes Substance P, neurotoxic

Capsicum spp 404-86-4

2092 D22 Microsource 01502197 PIPERIDOLATE HYDROCHLORIDE antispasmodic synthetic129-77-1, 82-98-4 [piperidolate]

2092 E03 Microsource 01500515 PROPYLTHIOURACIL antihyperthyroid synthetic 51-52-5

2092 E04 Microsource 01500615 ZOMEPIRAC SODIUManalgesic, antiinflammatory

synthetic64092-49-5, 64092-48-4 [anhydrous], 33369-31-2 [zomepirac]

2092 E05 Microsource 01500516 PSEUDOEPHEDRINE HYDROCHLORIDE decongestant synthetic345-78-8, 90-82-4 [pseudoephedrine]

2092 E06 Microsource 01500616 ACETARSOLantiprotozoal; diethylamine salt as antiphilitic

synthetic 97-44-9

2092 E07 Microsource 01500517 PYRANTEL PAMOATE anthelmintic synthetic22204-24-6, 15686-83-6 [pyrantel]

2092 E08 Microsource 01500618 ACRIFLAVINIUM HYDROCHLORIDEantiinfective, intercalating agent

synthetic 8018-07-3

2092 E09 Microsource 01500518 PYRAZINAMIDEantibacterial, tuberculostatic

synthetic 98-96-4

2092 E10 Microsource 01500621 AMINOPYRINE antipyretic, analgesic synthetic83-07-8, 747-30-8 [aminophenazone cyclamate]

2092 E11 Microsource 01500519 PYRILAMINE MALEATE antihistaminic synthetic59-33-6, 91-84-9 [pyrilamine]

2092 E12 Microsource 01500637 MERBROMIN antibacterial synthetic 129-16-82092 E13 Microsource 01500520 PYRIMETHAMINE antimalarial synthetic 58-14-0

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VendorVendor

IDCompound Name Bioactivity Source CAS

2092 E14 Microsource 01500642 PHENACETIN analgesic, antipyretic synthetic 62-44-22092 E15 Microsource 01500521 PYRVINIUM PAMOATE anthelmintic synthetic 3546-41-6

2092 E16 Microsource 01500643 PHENETHICILLIN POTASSIUM antibacterial semisynthetic132-93-4, 147-55-7 [phenethicillin]

2092 E17 Microsource 01500522 QUINACRINE HYDROCHLORIDEanthelmintic, antimalarial, intercalating agent

synthetic6151-30-0, 69-05-6 [anhydrous], 83-89-6 [quinacrine]

2092 E18 Microsource 01500644 PHENYLMERCURIC ACETATE antifungal synthetic 62-38-4

2092 E19 Microsource 01500523 QUINIDINE GLUCONATEantiarrhythmic, antimalarial

Cinchona spp7054-25-3, 6591-63-5 [quinidine sulfate], 56-54-2 [quinidine]

2092 E20 Microsource 01500646 SULFANILAMIDE antibacterial synthetic 63-74-1

2092 E21 Microsource 01500524 QUININE SULFATEantimalarial, skeletal muscle relaxant

Cinchona spp6119-70-6, 804-63-7 [anhydrous], 130-95-0 [quinine]

2092 E22 Microsource 01500648 AZELAIC ACIDantiacne, antiproliferative agent

rancid fats and Lycopodium spp

123-99-9

2092 F03 Microsource 01501129 CARBETAPENTANE CITRATE antitussive synthetic23142-01-0, 77-23-6 [carbetapentane]

2092 F04 Microsource 01502198 ANISINDIONE anticoagulant synthetic 117-37-3

2092 F05 Microsource 01501130 FAMPRIDINEK channel blocker; multiple sclerosis therapy

synthetic 504-24-5

2092 F06 Microsource 01502202 CYCLOSPORINE immunosuppressantTolypocladium inflatum

59865-13-3

2092 F07 Microsource 01501133 NICERGOLINE vasodilator synthetic 27848-84-6

2092 F08 Microsource 01502203 TROLEANDOMYCIN antibacterialsemisynthetic; TAO, NSC-108166

2751-09-9

2092 F09 Microsource 01501134 PIMOZIDE antipsychotic synthetic 2062-78-42092 F10 Microsource 01502230 ASCORBIC ACID antiscorbutic, antiviral Vitamin C 50-81-7

2092 F11 Microsource 01501137 NEFOPAM analgesic synthetic23327-57-3, 13669-70-0 [nefopam]

2092 F12 Microsource 01502254 MENADIONE prothrombogenic agentAsplenium and Juglans spp.

58-27-5

2092 F13 Microsource 01501138 PIRENZEPINE HYDROCHLORIDE antiulcer synthetic29868-97-1, 28797-61-7 [pirenzepine]

2092 F14 Microsource 01502255 SALICIN analgesic, antipyretic Salix spp 138-52-3

2092 F15 Microsource 01501139 PRAMOXINE HYDROCHLORIDE anesthetic (topical) synthetic637-58-1, 140-65-8 [pramoxine]

2092 F16 Microsource 01502258 MONENSIN SODIUM (monensin A is shown) antibacterialStreptomyces cinnamonensis

22373-78-0, 17090-79-8 (monensin)

2092 F17 Microsource 01501140 MEPHENESINmuscle relaxant (skeletal)

synthetic 59-47-2

2092 F18 Microsource 01503001 BENZOIC ACID antifungal synthetic 65-85-02092 F19 Microsource 01501142 SULFACHLORPYRIDAZINE antibacterial synthetic 80-32-02092 F20 Microsource 01503002 BENZYL BENZOATE scabicide synthetic 120-51-42092 F21 Microsource 01501144 SULFADIMETHOXINE antibacterial synthetic 122-11-22092 F22 Microsource 01503004 BENZOYL PEROXIDE keratolytic synthetic; NSC-675 94-36-0

2092 G03 Microsource 01500525 RACEPHEDRINE HYDROCHLORIDEbronchodilator, decongestant

synthetic134-71-4, 90-81-3 [racephedrine]

2092 G04 Microsource 01500649 THEOBROMINEdiuretic, bronchodilator, cardiotonic

Camelia, Theobroma, Cola spp

83-67-0

2092 G05 Microsource 01500526 RESERPINE antihypertensive Rauwolfia serpentina 50-55-5

2092 G06 Microsource 01500651 STRYCHNINE central stimulantStrychnos nux-vomica and other Strychnos spp

57-24-9

2092 G07 Microsource 01500527 RESORCINOL keratolytic, antiseborheic coal tar 108-46-3

2092 G08 Microsource 01500663 YOHIMBINE HYDROCHLORIDEalpha adrenergic blocker, mydriatic, antidepressant

Corynanthe spp 65-19-0

2092 G09 Microsource 01500529 RIFAMPINantibacterial (tuberculostatic)

semisynthetic; L-5103, Ba-41166/E, NSC-113926

13292-46-1

2092 G10 Microsource 01500665 ACEBUTOLOL HYDROCHLORIDEantihypertensive, antianginal, antiarrhythmic

synthetic34381-68-5, 37517-30-9 [acebutolol]

2092 G11 Microsource 01500530 ROXARSONE antibacterial synthetic 121-19-7

2092 G12 Microsource 01500655 ACONITINEanesthetic (gastric), antipyretic, and cardiotoxin

Aconitum spp 302-27-2

2092 G13 Microsource 01500531 SALICYL ALCOHOLanesthetic (local), antiinflammatory

Populus sieboldii 90-01-7

2092 G14 Microsource 01500667 ADENOSINE PHOSPHATEvasodilator, neuromodulator

widespread in living tissue

61-19-8

2092 G15 Microsource 01500532 SALICYLAMIDE analgesic synthetic 65-45-2

2092 G16 Microsource 01500668 KETOTIFEN FUMARATE antiasthmatic synthetic34580-14-8, 34580-13-7 [ketotifen]

2092 G17 Microsource 01500533 SODIUM SALICYLATE keratolytic synthetic 54-21-7

2092 G18 Microsource 01500670 BETAHISTINE HYDROCHLORIDE vasodilator synthetic5579-84-0, 5638-76-6 [betahistine]

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IDCompound Name Bioactivity Source CAS

2092 G19 Microsource 01500534 SCOPOLAMINE HYDROBROMIDEanticholinergic, treatment of motion sickness

Scopolia, Datura, Atropa spp

6533-68-2, 114-49-8 [anhydrous], 51-34-3 [scopolamine]

2092 G20 Microsource 01500673 MOLSIDOMINE antianginal synthetic 25717-80-0

2092 G21 Microsource 01500536 SISOMICIN SULFATEantibacterial, binds to ribosomes

Micromonospora myoensis

53179-09-2, 32385-11-8 [sisomicin]

2092 G22 Microsource 01500674 MYCOPHENOLIC ACID antineoplasticPenicillium brevicompactum and other Penicillium spp

24280-93-1

2092 H03 Microsource 01501145 SULFAQUINOXALINE SODIUM antibacterial synthetic 59-40-5

2092 H04 Microsource 01503007 BETAINE HYDROCHLORIDEantiarteriosclerotic, hypolipaemic, hepatoprotectant

widespread in fungi and plants

590-46-5, 141-58-2 [replaced], 107-43-7 [betaine]

2092 H05 Microsource 01501146 SULFAGUANIDINE antibacterial synthetic 57-67-0

2092 H06 Microsource 01502260 ABAMECTINantiparisitic (avermectin A1a shown)

Streptomyces avermitilis

65195-55-3

2092 H07 Microsource 01501147 SULFAMONOMETHOXINE antibacterial synthetic 1220-83-32092 H08 Microsource 01503009 BIOTIN vitamin B complex Vitamin B complex 58-85-5

2092 H09 Microsource 01501148 SULCONAZOLE NITRATE antifungal synthetic61318-91-0, 61318-90-9 [sulconazole]

2092 H10 Microsource 01503014 AKLOMIDEantiprotozoal, coccidiostat

synthetic 3011-89-0

2092 H11 Microsource 01501149 RITODRINE HYDROCHLORIDE muscle relaxant (smooth) synthetic23239-51-2, 26652-09-5 [ritodrine]

2092 H12 Microsource 01503038 NICOTINYL ALCOHOL TARTRATE vasodilator synthetic 100-55-0

2092 H13 Microsource 01501150 SULPIRIDEdopamine receptor antagonist, antipsychotic

synthetic 15676-16-1

2092 H14 Microsource 01503059 FLOXURIDINEantineoplastic, antimetabolite

synthetic 50-91-9

2092 H15 Microsource 01501151 RANITIDINE H2 antihistamine synthetic 66357-35-52092 H16 Microsource 01503065 ALTRETAMINE antineoplastic synthetic 645-05-62092 H17 Microsource 01501152 SPIPERONE antipsychotic synthetic; R-5147 749-02-0

2092 H18 Microsource 01503069 AMINOHIPPURIC ACID renal function diagnosis synthetic61-78-9, 94-16-6 [aminohippurate sodium]

2092 H19 Microsource 01501153 SULOCTIDIL peripheral vasodilator synthetic 54063-56-82092 H20 Microsource 01503070 MEFLOQUINE antimalarial synthetic 53230-10-72092 H21 Microsource 01501154 RONIDAZOLE antiprotozoal synthetic 7681-76-7

2092 H22 Microsource 01503073 ADIPHENINE HYDROCHLORIDE muscle relaxant (smooth) synthetic50-42-0, 64-95-9 [adiphenine]

2092 I03 Microsource 01500538 SPECTINOMYCIN HYDROCHLORIDE antibacterialStreptomyces spectabilis

22189-32-8, 21736-83-4 [anhydrous], 1695-77-8 [spectinomycin]

2092 I04 Microsource 01500675 OLEANDOMYCIN PHOSPHATE antibacterialStreptomyces antibioticus

3922-90-5 (base)

2092 I05 Microsource 01500539 SPIRONOLACTONE diuretic synthetic 52-01-7

2092 I06 Microsource 01500676 OUABAINantiarrhythmic, cardiotonic, hypertensive, Na/K ATPase inhibitor

Acokanthera and Strophanthus spp

11018-89-6, 630-60-4 [anhydrous]

2092 I07 Microsource 01500541 STREPTOMYCIN SULFATEantibacterial (tuberculostatic)

Streptomyces griseus

3810-74-0, 57-92-1 [streptomycin]

2092 I08 Microsource 01500677 ALBUTEROL (+/-) bronchodilator, tocolytic synthetic 18559-94-9

2092 I09 Microsource 01500543 STREPTOZOSINantineoplastic, alkylating agent

synthetic 18883-66-4

2092 I10 Microsource 01500680 ARECOLINE HYDROBROMIDEanthelmintic (Cestodes), hypotensive, cathartic

betel nuts (Arica catechu)

300-08-3, 63-75-2 [arecoline]

2092 I11 Microsource 01500544 SULFABENZAMIDE antibacterial synthetic 127-71-92092 I12 Microsource 01500682 CAPTOPRIL antihypertensive synthetic 62571-86-2

2092 I13 Microsource 01500545 SULFACETAMIDE antibacterial synthetic

144-80-9, 127-56-0 [anhydrous], 6209-17-2 [sulfacetamide sodium]

2092 I14 Microsource 01500684 CIMETIDINE antiulcer synthetic 51481-61-92092 I15 Microsource 01500546 SULFADIAZINE antibacterial synthetic 68-35-92092 I16 Microsource 01500685 CLOZAPINE antipsychotic synthetic 5786-21-02092 I17 Microsource 01500547 SULFAMERAZINE antibacterial synthetic 127-79-7

2092 I18 Microsource 01500687 HYDRASTINE (1R, 9S)antihypertensive, sedative, antibacterial

Corydalis spp 118-08-1

2092 I19 Microsource 01500548 SULFAMETHAZINE antibacterial synthetic 57-68-1

2092 I20 Microsource 01500689 LIDOCAINE HYDROCHLORIDEanesthetic (local), antiarrhythmic

synthetic6108-05-0, 73-78-9 [anhydrous], 137-58-6 [lidocaine]

2092 I21 Microsource 01500549 SULFAMETHIZOLE antibacterial synthetic 144-82-1

2092 I22 Microsource 01500691 PHENTOLAMINE HYDROCHLORIDE antihypertensive synthetic73-05-2, 50-60-2 [phentolamine]

2092 J03 Microsource 01501155 SULFAMETER antibacterial synthetic 651-06-9

2092 J04 Microsource 01503076 QUINAPRIL HYDROCHLORIDEantihypertensive, ACE inhibitor

synthetic82586-55-8, 85441-61-8 [quinapril]

2092 J05 Microsource 01501156 SULFAMETHOXYPYRIDAZINE antibacterial synthetic 80-35-3

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IDCompound Name Bioactivity Source CAS

2092 J06 Microsource 01503083 AMIPRILOSEimmunomodulator, antiinflammatory

semisynthetic56824-20-5, 60414-06-4 [amiprilose hydrochloride]

2092 J07 Microsource 01501161 SUPROFEN antiinflammatory synthetic 40828-46-42092 J08 Microsource 01503086 TIAPRIDE HYDROCHLORIDE neuroleptic synthetic 51012-32-92092 J09 Microsource 01501171 SACCHARIN sweetener synthetic 81-07-22092 J10 Microsource 01503092 GLUCONOLACTONE chelating agent synthetic 90-80-22092 J11 Microsource 01501173 ACETANILIDE analgesic, antipyretic synthetic 103-84-42092 J12 Microsource 01503101 AZLOCILLIN SODIUM antibacterial semisynthetic 37091-66-02092 J13 Microsource 01501175 FLURANDRENOLIDE antiinflammatory semisynthetic 1524-88-5

2092 J14 Microsource 01503102 BACAMPICILLIN HYDROCHLORIDE antibacterial semisynthetic37661-08-8, 50972-17-3 [bacampicillin]

2092 J15 Microsource 01501176 ERYTHROMYCIN ESTOLATE antibacterialStreptomyces erythreus

134-36-1, 114-07-8 [erythromycin]

2092 J16 Microsource 01503104 BENDROFLUMETHIAZIDE diuretic, antihypertensive synthetic 73-48-3

2092 J17 Microsource 01501179 ESTRADIOL PROPIONATE estrogen semisynthetic 113-38-2

2092 J18 Microsource 01503106 BEPRIDIL HYDROCHLORIDE antiarrhythmicsynthetic; CERM-1978

74764-40-2

2092 J19 Microsource 01501182 ESTRADIOL BENZOATE estrogen semisynthetic 50-50-0

2092 J20 Microsource 01503107 BROMHEXINE HYDROCHLORIDE expectorant synthetic611-75-6, 3572-43-8 [bromhexine]

2092 J21 Microsource 01501184 ESTRADIOL ACETATE estrogen semisynthetic 4245-41-4

2092 J22 Microsource 01503110 CARMUSTINEantineoplastic, alkylating agent

synthetic 154-93-8

2092 K03 Microsource 01500550 SULFAMETHOXAZOLEantibacterial, antipneumocystis

synthetic 723-46-6

2092 K04 Microsource 01500756 NALIDIXIC ACID antibacterial synthetic389-08-2, 3374-05-8 [anhydrous], 15769-77-4 [nalidixate sodium]

2092 K05 Microsource 01500551 SULFAPYRIDINE antibacterial synthetic 144-83-22092 K06 Microsource 01500767 BUTAMBEN anesthetic (local) synthetic 94-25-7

2092 K07 Microsource 01500552 SULFASALAZINEanticolitis and Crohn's disease

synthetic 599-79-1

2092 K08 Microsource 01500771 CEFACLOR antibacterial semisynthetic70356-03-5, 53994-73-3 [anhydrous]

2092 K09 Microsource 01500553 SULFATHIAZOLE antibacterial synthetic 72-14-0

2092 K10 Microsource 01500772 IODIPAMIDE radioopaque agentsynthetic; L-isomer: spectrum

606-17-7, 2618-26-0 [iodipamide sodium]

2092 K11 Microsource 01500554 SULFINPYRAZONE uricosuric synthetic 57-96-5

2092 K12 Microsource 01500774 LEVOTHYROXINEantihypercholesterimic, thyromimetic

thyroid gland 51-48-9

2092 K13 Microsource 01500555 SULFISOXAZOLE antibacterial synthetic 127-69-52092 K14 Microsource 01500778 LIOTHYRONINE thyroid hormone blocker semisynthetic 6893-02-32092 K15 Microsource 01500556 SULINDAC antiinflammatory synthetic 38194-50-2

2092 K16 Microsource 01500801 ALLANTOIN wound healing agentallantoic fluid; widely distributed in plants

97-59-6

2092 K17 Microsource 01500557 TAMOXIFEN CITRATEestrogen antagonist, antineoplastic

synthetic54965-24-1, 10540-29-1 [tamoxifen]

2092 K18 Microsource 01500804 ALTHIAZIDE diuretic synthetic 5588-16-9

2092 K19 Microsource 01500558 TERBUTALINE HEMISULFATEbetaadrenergic agonist, bronchodilator

synthetic23031-32-5, 23031-25-6 [terbutaline]

2092 K20 Microsource 01500807 ADENINE Vitamin B4 widespread in nature 73-24-5

2092 K21 Microsource 01500564 TETRACAINE HYDROCHLORIDE anesthetic (local) synthetic136-47-0, 94-24-6 [tetracaine]

2092 K22 Microsource 01500810 AMINACRINE local antiseptic synthetic90-45-9, 134-50-9 [aminacrine hydrochloride]

2092 L03 Microsource 01501185 ECONAZOLE NITRATE antifungal SQ-13050; synthetic68797-31-9, 27220-47-9 [econazole]

2092 L04 Microsource 01503111 CEFTRIAXONE SODIUM TRIHYDRATE antibacterialsemisynthetic; RO-13-9904

104376-79-6, 73384-59-5 [ceftriaxone]

2092 L05 Microsource 01501187 FLUNISOLIDE antiinflammatory semisynthetic77326-96-6, 3385-03-3

2092 L06 Microsource 01503115 VINPOCETINEcerebral vasodilator, antimotion

vincamine Vinca minor

42971-09-5

2092 L07 Microsource 01501200 XYLAZINE analgesic synthetic23076-35-9, 7361-61-7 [xylazine]

2092 L08 Microsource 01503117 TRIMIPRAMINE MALEATE antidepressant synthetic521-78-8, 739-71-9 [trimipramine]

2092 L09 Microsource 01501201 TOLAZAMIDE antidiabetic synthetic 1156-19-0

2092 L10 Microsource 01503118 TRIFLUPROMAZINE HYDROCHLORIDE antipsychotic synthetic1098-60-8, 146-54-3 [triflupromazine]

2092 L11 Microsource 01501202 GALANTHAMINE HYDROBROMIDEanticholinesterase, analgesic, antiAlzheimer

Galanthus, Narcissus and other Lillaceae

357-70-0, 1953-04-4 [hydrobromide]

2092 L12 Microsource 01503121 TRAZODONE HYDROCHLORIDE antidepressant synthetic25332-39-2, 19794-93-5 [trazodone]

2092 L13 Microsource 01501203 RETINOL vitamin Afish & liver oils, eggs, milk

68-26-8

Microsource1-US Drug Collection Page 13 of 24 Created 9/2015

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IDCompound Name Bioactivity Source CAS

2092 L14 Microsource 01503134 MENTHOL(-)analgesic (topical), antipruritic agent

Mentha piperita and other Mentha spp

1490-04-6

2092 L15 Microsource 01501205 LANATOSIDE C cardiotoniccardiotonc Digitalis lanata

17575-22-3

2092 L16 Microsource 01503135 THONZYLAMINE HYDROCHLORIDE antihistamine synthetic63-56-9, 91-85-0 [thonzylamine]

2092 L17 Microsource 01501214 ENALAPRIL MALEATEACE inhibitor, antihypertensive

synthetic76095-16-4, 75847-73-3 [enalapril]

2092 L18 Microsource 01503136 THIAMPHENICOL antibacterial synthetic 15318-45-32092 L19 Microsource 01501215 KETOPROFEN antiinflammatory synthetic 22071-15-42092 L20 Microsource 01503142 TENOXICAM antiinflammatory synthetic 59804-37-4

2092 L21 Microsource 01501217 LISINOPRIL ACE inhibitor synthetic83915-83-7, 76547-98-3 [anhydrous]

2092 L22 Microsource 01503200 CETRIMONIUM BROMIDE antiinfectant synthetic57-09-0, 6899-10-1 [cetrimonium]

2092 M03 Microsource 01500566 TETRACYCLINE HYDROCHLORIDEantibacterial, antiamebic, antirickettsial

Streptomyces spp64-75-5, 60-54-8 [tetracycline]

2092 M04 Microsource 01500812 BEKANAMYCIN SULFATE antibacterial

semisynthetic; Streptomyces kanamyceticus; NK-1006

4696-76-8 (base)

2092 M05 Microsource 01500568 THEOPHYLLINE bronchodilatorCamelia, thea, Paullinia cupana

5967-84-0, 58-55-9 [anhydrous]

2092 M06 Microsource 01500822 BRUCINE central stimulantStrychnos nux-vomica

4845-99-2, 357-57-3 [brucine]

2092 M07 Microsource 01500570 THIABENDAZOLE anthelmintic synthetic 148-79-8

2092 M08 Microsource 01500828 CANRENOIC ACID, POTASSIUM SALTaldosterone antagonist, diuretic

semisynthetic2181-04-6, 4138-96-9 [canrenoic acid]

2092 M09 Microsource 01500572 THIMEROSAL antiinfective, preservative synthetic 54-64-8

2092 M10 Microsource 01500837 CHENODIOLanticholithogenic, antilipemic agent

human bile 474-25-9

2092 M11 Microsource 01500573 THIOGUANINEantineoplastic, purine antimetabolite

synthetic154-42-7, 5580-03-0 [hemihydrate]

2092 M12 Microsource 01500838 CHOLECALCIFEROL vitamin D3 fish oils 67-97-0

2092 M13 Microsource 01500575 THIORIDAZINE HYDROCHLORIDE antipsychotic synthetic130-61-0, 50-52-2 [thioridazine]

2092 M14 Microsource 01500839 CINCHONIDINE antimalarial Cinchona spp 485-71-2

2092 M15 Microsource 01500576 THIOTHIXENE antipsychotic synthetic5591-45-7, 3313-26-6 [//Z//]

2092 M16 Microsource 01500841 CINCHONINE antimalarial Cinchona spp 118-10-5

2092 M17 Microsource 01500579 TOBRAMYCINantibacterial, inhibits protein synthesis

Streptomyces spp 32986-56-4

2092 M18 Microsource 01500844 COENZYME B12 vitaminVitamin B12; cyanocobalamin

13870-90-1

2092 M19 Microsource 01500580 TOLAZOLINE HYDROCHLORIDE adrenergic blocker synthetic59-97-2, 59-98-3 [tolazoline]

2092 M20 Microsource 01500847 CHOLESTEROL emulsifying agentcommon animal sterol

57-88-5

2092 M21 Microsource 01500581 TOLBUTAMIDE antidiabetic synthetic 64-77-7

2092 M22 Microsource 01500873 PIPERINE analeptic, antibacterialblack pepper (Piper nigrum L.)

94-62-2

2092 N03 Microsource 01502004 BUMETANIDE diuretic synthetic 28395-03-12092 N04 Microsource 01503202 CHLOROXINE chelating agent synthetic 773-76-2

2092 N05 Microsource 01502005 CARBENOXOLONE SODIUMantiinflammatory, antisecretory, antiulcer

semisynthetic7421-40-1, 5697-56-3 [carbenoxolone]

2092 N06 Microsource 01503203 CHLORPROTHIXENE HYDROCHLORIDE antipsychotic synthetic 113-59-72092 N07 Microsource 01502013 ISOTRETINON antiacne, antineoplastic semisynthetic 4759-48-22092 N08 Microsource 01503204 CINNARAZINE H1 antihistamine synthetic 298-57-7

2092 N09 Microsource 01502014 MESNA mucolytic synthetic

19767-45-4, 3375-50-6 [2-mercaptoethanesulfonic, acid]

2092 N10 Microsource 01503207 CYCLOBENZAPRINE HYDROCHLORIDEmuscle relaxant (skeletal)

synthetic6202-23-9, 303-53-7 [cyclobenzaprine]

2092 N11 Microsource 01502016 TRETINON keratolytic semisynthetic 302-79-4

2092 N12 Microsource 01503209 DANTROLENE SODIUMmuscle relaxant (skeletal)

synthetic24868-20-0, 14663-23-1 [anhydrous], 7261-97-4 [dantrolene]

2092 N13 Microsource 01502018 BRETYLIUM TOSYLATEinhibitor of norepinephrine release

synthetic61-75-6, 59-41-6 [bretylium]

2092 N14 Microsource 01503210 BETAMETHASONE 17,21-DIPROPIONATEglucocorticoid, antiinflammatory

semisynthetic 5593-20-4

2092 N15 Microsource 01502019 FOSCARNET SODIUM antiviral synthetic 63585-09-1

2092 N16 Microsource 01503212 DOBUTAMINE HYDROCHLORIDE cardiotonic synthetic49745-95-1, 34368-04-2 [dobutamine]

2092 N17 Microsource 01502020 FOLIC ACID hematopoietic vitaminliver, kidney, green plants and fungi

59-30-3

2092 N18 Microsource 01503214 EDOXUDINE antiviralsynthetic; EDU; EUDR; ORF-15817; RWJ-15817

15176-29-1

2092 N19 Microsource 01502021 PHTHALYLSULFATHIAZOLE antibacterial synthetic 85-73-4

Microsource1-US Drug Collection Page 14 of 24 Created 9/2015

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VendorVendor

IDCompound Name Bioactivity Source CAS

2092 N20 Microsource 01503215 ENOXACIN antibacterial synthetic 74011-58-82092 N21 Microsource 01502025 SUCCINYLSULFATHIAZOLE antibacterial synthetic 116-43-8

2092 N22 Microsource 01503221 ETHISTERONE progestogen synthetic; NSC-9565 434-03-7

2092 O03 Microsource 01500582 TOLMETIN SODIUM antiinflammatory synthetic64490-92-2, 26171-23-3 [tolmetin]

2092 O04 Microsource 01500903 ETOPOSIDE antineoplastic semisynthetic 33419-42-0

2092 O05 Microsource 01500583 TOLNAFTATE antifungalsynthetic; SCH-10144

2398-96-1

2092 O06 Microsource 01500907 DEHYDROCHOLIC ACID cholereticderivative of cholic acid

81-23-2

2092 O07 Microsource 01500584 TRANYLCYPROMINE SULFATEantidepressant, MAO inhibitor

synthetic13492-01-8, 7081-36-9 [replaced], 155-09-9 [tranylcypromine]

2092 O08 Microsource 01500992 FLUMEQUINE antibacterial synthetic 42835-25-62092 O09 Microsource 01500585 TRIACETIN antifungal (topical) synthetic 102-76-1

2092 O10 Microsource 01500993 FLUNARIZINE HYDROCHLORIDE vasodilator synthetic30484-77-6, 52468-60-7 [flunarazine]

2092 O11 Microsource 01500586 TRIAMCINOLONE glucocorticoid semisynthetic 124-94-72092 O12 Microsource 01500994 FLUPHENAZINE HYDROCHLORIDE H1 antihistamine synthetic 146-56-52092 O13 Microsource 01500587 TRIAMCINOLONE ACETONIDE antiinflammatory semisynthetic 76-25-52092 O14 Microsource 01500995 FLUTAMIDE antiandrogen synthetic 13311-84-72092 O15 Microsource 01500588 TRIAMCINOLONE DIACETATE antiinflammatory semisynthetic 67-78-72092 O16 Microsource 01501002 DROPERIDOL neuroleptic synthetic 548-73-22092 O17 Microsource 01500589 TRIAMTERENE diuretic semisynthetic 396-01-02092 O18 Microsource 01501003 FAMOTIDINE H2 antihistamine synthetic 76824-35-6

2092 O19 Microsource 01500590 TRICHLORMETHIAZIDE diuretic, antihypertensive synthetic 133-67-5

2092 O20 Microsource 01501005 ETODOLAC antiinflammatory synthetic 41340-25-4

2092 O21 Microsource 01500591 TRIFLUOPERAZINE HYDROCHLORIDE antipsychotic synthetic440-17-5, 117-89-5 [trifluoperazine]

2092 O22 Microsource 01501007 FENOTEROL HYDROBROMIDE betaadrenergic agonist synthetic 13392-18-22092 P03 Microsource 01502026 TRANEXAMIC ACID hemostatic synthetic 1197-18-8

2092 P04 Microsource 01503223 PARAROSANILINE PAMOATEanthelmintic, antischistosomal

synthetic7232-51-1, 569-61-9 [pararosaniline]

2092 P05 Microsource 01502028 CEPHALEXIN antibacterial semisynthetic23325-78-2, 15686-71-2 [anhydrous]

2092 P06 Microsource 01503227 PERHEXILINE MALEATE coronary vasodilator synthetic6724-53-4, 6621-47-2 [perhexiline]

2092 P07 Microsource 01502029 CEFSULODIN SODIUM antibacterial semisynthetic52152-93-9, 62587-73-9 [cefsulodin]

2092 P08 Microsource 01503229 METHAPYRILENE HYDROCHLORIDE H1 antihistamine synthetic135-23-9, 91-80-5 [methapyrilene]

2092 P09 Microsource 01502030 OXOLINIC ACID antibacterial synthetic 14698-29-42092 P10 Microsource 01503239 HYCANTHONE anthelmintic, hepatotoxic synthetic 3105-97-3

2092 P11 Microsource 01502031 CEFOXITIN SODIUM antibacterial semisynthetic66309-69-1, 61622-34-2 [cefotiam]

2092 P12 Microsource 01503234 BETA-PROPIOLACTONE antiinfectivesynthetic; NSC-21626

57-57-8

2092 P13 Microsource 01502032 SURAMINantiprotozoal, trypanocidal, antiviral

synthetic; Bayer-205, 309F

129-46-4, 145-63-1 [suramin]

2092 P14 Microsource 01503240 PYRIDOSTIGMINE BROMIDE cholinergic synthetic101-26-8, 155-97-5 [pyridostigmine]

2092 P15 Microsource 01502033 CEFUROXIME SODIUM antibacterial semisynthetic 56238-63-22092 P16 Microsource 01503242 ISOXICAM antiinflammatory synthetic 34552-84-6

2092 P17 Microsource 01502037 LOMEFLOXACIN HYDROCHLORIDE antibacterial synthetic98079-52-8, 98079-51-7 (lomefloxacin)

2092 P18 Microsource 01503243 LABETALOL HYDROCHLORIDE adrenergic blocker synthetic32780-64-6, 36894-69-6 [labetalol]

2092 P19 Microsource 01502038 CEFAMANDOLE SODIUM antibacterial semisynthetic 34444-01-4

2092 P20 Microsource 01503245 LEVAMISOLE HYDROCHLORIDE immunomodulator synthetic16595-80-5, 14769-73-4 [levamisole]

2092 P21 Microsource 01502039 FOSFOMYCIN CALCIUM antibacterial Streptomyces spp26472-47-9, 23112-90-5(acid)

2092 P22 Microsource 01503250 MEPHENTERMINE SULFATE vasoconstrictor synthetic1212-72-2, 6190-60-9 [dihydrate], 100-92-5 [mephentermine]

2093 A03 Microsource 01503251 METARAMINOL BITARTRATE antihypotensive synthetic 33402-03-8

2093 A04 Microsource 01504142 ACETRIAZOIC ACID X-ray contrast medium synthetic85-36-9, 129-63-5 [acetrizoate sodium]

2093 A05 Microsource 01503252 METHAZOLAMIDEcarbonic anhydrase inhibitor

synthetic 554-57-4

2093 A06 Microsource 01504144 DIRITHROMYCIN antibacterial semisynthetic 62013-04-1

2093 A07 Microsource 01503253 METHYLBENZETHONIUM CHLORIDE antiinfective synthetic1320-44-1, 25155-18-4 [anhydrous]

2093 A08 Microsource 01504148 MEPIVACAINE HYDROCHLORIDE anesthetic (local) synthetic1722-62-9, 96-88-8 [mepivacaine]

2093 A09 Microsource 01503255METHYLPREDNISOLONE SODIUM SUCCINATE

glucocorticoid, antiinflammatory

semisynthetic 2375-03-3

2093 A10 Microsource 01504152 NILUTAMIDE antiandrogen synthetic 63612-50-0

2093 A11 Microsource 01503256 AMSACRINEantineoplastic, immune suppressive

synthetic 51264-14-3

2093 A12 Microsource 01504171 VENLAFAXINE antidepressant synthetic99300-78-4, 93413-69-5 [venlafaxine]

Microsource1-US Drug Collection Page 15 of 24 Created 9/2015

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VendorVendor

IDCompound Name Bioactivity Source CAS

2093 A13 Microsource 01503257 MIDODRINE HYDROCHLORIDEantihypertensive, vasoconstrictor

synthetic3092-17-9, 42794-76-3 [midodrine]

2093 A14 Microsource 01504172 CITALOPRAMantidepressant, 5HT reuptake inhibitor

synthetic 59729-33-8

2093 A15 Microsource 01503260 NADOLOL betaadrenergic blocker synthetic 42200-33-92093 A16 Microsource 01504173 FLUOXETINE antidepressant synthetic 54910-89-3

2093 A17 Microsource 01503262 NALTREXONE HYDROCHLORIDE morphine antagonist synthetic16676-29-2, 16590-41-3 [naltrexone]

2093 A18 Microsource 01504174 BUPROPION antidepressant synthetic31677-93-7, 34911-55-2 [bupropion]

2093 A19 Microsource 01503263 CYCLOTHIAZIDE diuretic synthetic 2259-96-3

2093 A20 Microsource 01504175 CEFUROXIME AXETIL antibacterial synthetic64544-07-6, 55268-75-2 [cefuroxime]

2093 A21 Microsource 01503265 NICLOSAMIDE anthelmintic, teniacide synthetic; BAY-2353 50-65-7

2093 A22 Microsource 01504179 FEXOFENADINE HYDROCHLORIDEnonsedating H1-antihistamine

synthetic 138452-21-8

2093 B03 Microsource 01505305 PEFLOXACINE MESYLATEantibacterial, antiproliferative

synthetic 149676-40-4

2093 B04 Microsource 01505622 RALOXIFENE HYDROCHLORIDE antiestrogen synthetic-LY-156758 82640-04-8

2093 B05 Microsource 01505306 ASPARTAME sweetener synthetic 22839-47-02093 B06 Microsource 01505636 ZIMELIDINE DIHYDROCHLORIDE antidepressant synthetic; H-102/09 61129-30-4

2093 B07 Microsource 01505308 CHLOROPHYLLIDE Cu COMPLEX Na SALT antineoplasticwater soluble derivative of chlorophyll

15611-43-5

2093 B08 Microsource 01505637 CEFPODOXIME PROXETIL antibacterialsemisynthetic; U-76252, CS-807

87239-81-4

2093 B09 Microsource 01505309 BIFONAZOLEantifungal, calmodulin antagonist

synthetic 60628-96-8

2093 B10 Microsource 01505650 AMINOPENTAMIDEantispasmodic, antiemetic

synthetic; NND-1962 119793-66-7

2093 B11 Microsource 01505312 TYLOSIN TARTRATE antibacterialStreptomyces fradiae

1405-54-5, 1401-69-0(base)

2093 B12 Microsource 01505652 ARSANILIC ACID antibacterial synthetic; AS-101 98-50-02093 B13 Microsource 01505314 SARAFLOXACIN HYDROCHLORIDE antibacterial synthetic 91296-87-6

2093 B14 Microsource 01505656 PANTHENOLvitamin B5 precursor, radioprotectant

various plants 16485-10-2

2093 B15 Microsource 01505319 CLOPIDOL coccidiostat, antiplatelet synthetic 2971-90-62093 B16 Microsource 01505660 PHENTERMINE anorexic synthetic 122-09-8

2093 B17 Microsource 01505321 RIFAXIMINantibacterial, RNA synthesis inhibitor

semisynthetic 80621-81-4

2093 B18 Microsource 01505665 PHTHALYSULFATHIAZOLE antibacterial synthetic 85-73-42093 B19 Microsource 01505327 CHLORMADINONE ACETATE progestin, antiandrogen semisynthetic 302-22-72093 B20 Microsource 01505668 RONNEL insecticide synthetic 299-84-32093 B21 Microsource 01505330 OXICONAZOLE NITRATE antifungal synthetic 64211-46-7

2093 B22 Microsource 01505672 VINCRISTINE SULFATE antineoplasticVinca rosea; 37231, NSC-67574

2068-78-2

2093 C03 Microsource 01503267 NOMIFENSINE MALEATEantidepressant, dopamine uptake inhibitor

synthetic32795-47-4, 24526-64-5 [nomifensine]

2093 C04 Microsource 01504190 AVOBENZONE sunscreen synthetic 70356-09-1

2093 C05 Microsource 01503269 PERGOLIDE MESYLATEdopamine receptor agonist

semisynthetic66104-23-2, 66104-22-1 [pergolide]

2093 C06 Microsource 01504184 AMINOLEVULINIC ACID HYDROCHLORIDE antineoplastic synthetic 5451-09-2

2093 C07 Microsource 01503270 PRILOCAINE HYDROCHLORIDE anesthetic (local) synthetic1786-81-8, 721-50-6 [prilocaine]

2093 C08 Microsource 01504188 PIRENPERONE 5HT2 receptor antagonist synthetic 75444-65-4

2093 C09 Microsource 01503273 HYDROCORTISONE BUTYRATEglucocorticoid, antiinflammatory

semisynthetic 13609-67-1

2093 C10 Microsource 01504210 ATOVAQUONEantipneumocystic, antimalarial

synthetic 95233-18-4

2093 C11 Microsource 01503276 ROXITHROMYCIN antibacterialsemisynthetic; RU-28965, RU-965

80214-83-1

2093 C12 Microsource 01504211 CHLOROGUANIDE HYDROCHLORIDE antimalarial synthetic 637-32-1

2093 C13 Microsource 01503278 MITOXANTHRONE HYDROCHLORIDE antineoplastic semisynthetic70476-82-3, 65271-80-9 [mitoxantrone]

2093 C14 Microsource 01504214 TRIMETOZINE sedative, neurosedative synthetic 635-41-62093 C15 Microsource 01503279 OXETHAZAINE anesthetic (local) synthetic 126-27-2

2093 C16 Microsource 01504216 ZOXAZOLAMINEmuscle relaxant, antirrheumatic

synthetic 61-80-3

2093 C17 Microsource 01503298 DIPYRONE analgesic, antipyretic synthetic5907-38-0, 68-89-3 [anhydrous]

2093 C18 Microsource 01504218 ACRISORCIN antifungal synthetic 7527-91-52093 C19 Microsource 01503301 SULFANILATE ZINC antibacterial synthetic 31884-76-1

2093 C20 Microsource 01504226 CYSTEAMINE HYDROCHLORIDEantiurolithic, depigmentation, radiation protectant

cysteamine; CL-9148

60-23-1

2093 C21 Microsource 01503304 URETHANE antineoplastic, cytotoxic synthetic; NSC-746 51-79-6

2093 C22 Microsource 01504229 METAXALONEmuscle relaxant (skeletal)

synthetic 1665-48-1

Microsource1-US Drug Collection Page 16 of 24 Created 9/2015

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VendorVendor

IDCompound Name Bioactivity Source CAS

2093 D03 Microsource 01505332 AZAPERONEtranquilizer, neuroleptic, alpha adrenergic blocker

synthetic; R-1929 1649-18-9

2093 D04 Microsource 01505673 TROGLITAZONE antidiabeticsynthetic; CS-045, CI-991, GR-92132X

97322-87-7

2093 D05 Microsource 01505340 AZELASTINE HYDROCHLORIDE

H1 antihistamine (nonsedating); leucotriene synthesis blocker

synthetic 58581-89-8

2093 D06 Microsource 01505675 TRIENTINE HYDROCHLORIDE chelating agent synthetic; MK-0681 38260-01-4

2093 D07 Microsource 01505347 RIBOFLAVINVitamin B2; Vitamin cofactor; LD50(rat) 560 mg/kg ip

retina, whey and urine

83-88-5

2093 D08 Microsource 01505677 TICLOPIDINE HYDROCHLORIDE PAF inhibitorsynthetic; 53-32C, 4-C-32

53885-35-1

2093 D09 Microsource 01505354 FIPRONILGABA Cl channel agonist, antiparasitic

synthetic; RM-1601, MB-46030

120068-37-3

2093 D10 Microsource 01505466 TRIMETHADIONE anticonvulsant synthetic 127-48-0

2093 D11 Microsource 01505356 DECOQUINATE coccidiostatsynthetic; M&B-15497, HC-1528

18507-89-6

2093 D12 Microsource 01505778 BEPHENIUM HYDROXYNAPTHOATE anthelmintic synthetic 3818-50-62093 D13 Microsource 01505360 CEFDITORIN PIVOXIL antibacterial semisynthetic 117467-28-42093 D14 Microsource 01505780 DIPERODON HYDROCHLORIDE analgesic, anesthetic synthetic 537-12-2

2093 D15 Microsource 01505361 MODAFINIL analepticsynthetic; CRL-40476, CEP-1538

68693-11-8

2093 D16 Microsource 01505781 SELEGILINE HYDROCHLORIDEantidepressant, MAO inhibitor, antiparkinsonian

synthetic 14611-52-0

2093 D17 Microsource 01505364 CEFPROZIL antibacterialsemisynthetic; BMY-28100-03-800

121123-17-9

2093 D18 Microsource 01505782 CEFTAZIDIME antibacterial semisynthetic 72558-82-82093 D19 Microsource 01505371 CETIRIZINE HYDROCHLORIDE H1 antihistamine synthetic 83881-52-1

2093 D20 Microsource 01505801 TOPIRAMATE

anticonvulsant, antimigraine, GABA-A agonist, AMP/kinate glutamate receptor antagonist, carbonic anhydrase inhibitor

synthetic; RWJ-17021

97240-79-4

2093 D21 Microsource 01505366 RANOLAZINE antianginal, antiischemicsynthetic; RS-43285-003; CVT-303

95635-55-5

2093 D22 Microsource 01505802 GEMIFLOXACIN MESYLATE antibacterial synthetic 204519-65-32093 E03 Microsource 01503322 THIRAM antifungal synthetic 137-26-8

2093 E04 Microsource 01504235 ROFECOXIBCOX2 inhibitor, antiinflammatory, antiarthritic

synthetic 162011-90-7

2093 E05 Microsource 01503324 THIOTEPAantineoplastic, alkylating agent

synthetic 52-24-4

2093 E06 Microsource 01504236 SIMVASTATINantihyperlipidemic, HMGCoA reductase inhibitor

synthetic 79902-63-9

2093 E07 Microsource 01503330 TETROQUINONE keratolytic synthetic 319-89-12093 E08 Microsource 01504237 HYDROQUINONE antioxidant synthetic 123-31-9

2093 E09 Microsource 01503339 SULFANITRAN antibacterialsynthetic; NSC-77120

122-16-7

2093 E10 Microsource 01504243 OXCARBAZEPINE antipsychotic synthetic 28721-07-5

2093 E11 Microsource 01503393 PIPOBROMANantineoplastic, alkylating agent

synthetic 54-91-1

2093 E12 Microsource 01504257 CARVEDILOL beta-adrenergic blocker synthetic 72956-09-3

2093 E13 Microsource 01503412 ETANIDAZOLEantineoplastic, hypoxic cell radiosensitizer

synthetic 22668-01-5

2093 E14 Microsource 01504258 NATEGLINIDE antidiabetic synthetic 105816-04-4

2093 E15 Microsource 01503419 NAFRONYL OXALATE vasodilator synthetic3200-06-4, 31329-57-4 [nafronyl]

2093 E16 Microsource 01504259 IRBESARTANangiotensin 2 receptor antagonist

synthetic 138402-11-6

2093 E17 Microsource 01503420 QUIPAZINE MALEATE antidepressant, oxytocic synthetic5786-68-5, 4774-24-7 [quipazine]

2093 E18 Microsource 01504260 LEVOFLOXACIN antibacterial synthetic 138199-71-02093 E19 Microsource 01503421 RITANSERIN antiserotonin synthetic 87051-43-2

2093 E20 Microsource 01504261 CANDESARTAN CILEXTILangiotensin 1 receptor antagonist

synthetic 139481-59-7

2093 E21 Microsource 01503422 SEMUSTINE antineoplastic synthetic 13909-09-6

2093 E22 Microsource 01504268 LOSARTANantihypertensive, AT1 angiotensin II antagonist

synthetic124750-99-8, 114798-26-4 [losartan]

2093 F03 Microsource 01505374 VARDENAFIL HYDROCHLORIDEerectile dysfunction, PD5 inhibitor

synthetic 224789-15-5

2093 F04 Microsource 01505803 PRAVASTATIN SODIUMantihyperlipidemic, HMGCoA reductase inhibitor

CS-514; SQ-31000 81131-70-6

2093 F05 Microsource 01505376 ACEDAPSONE antimalarial, leprostaticsynthetic; CI-556, CN-1883, DADDS, PAM-MAR-1165

77-46-3

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VendorVendor

IDCompound Name Bioactivity Source CAS

2093 F06 Microsource 01505805 GABAPENTIN anticonvulsantsynthetic; CI-945; GOE-3450

60142-96-3

2093 F07 Microsource 01505384 METHYLDOPATE HYDROCHLORIDE antihypertensive synthetic 2508-79-4

2093 F08 Microsource 01505814 METFORMIN HYDROCHLORIDE antidiabetic synthetic; LA-60231115-70-4, 657-24-9(metformin)

2093 F09 Microsource 01505385 ATOMOXETINE HYDROCHLORIDEnorepinephrine reuptake inhibitor

synthetic; LY-139603

82248-59-7

2093 F10 Microsource 01505816 PREGABALIN anticonvulsant synthetic; CI-1008 148553-50-8

2093 F11 Microsource 01505387 DULOXETINE HYDROCHLORIDE antidepressantsynthetic; LY-248686

136434-34-9

2093 F12 Microsource 01505817 RAMELTEONmelatonin receptor agonist

synthetic; TAK-375; M-II

196597-26-9

2093 F13 Microsource 01505389 TRAMADOL HYDROCHLORIDE analgesicsynthetic; U-26225A, CG-315E

36282-47-0

2093 F14 Microsource 01505818 PANTOPRAZOLEproton pump inhibitor, gastric acid release inhibitor, antiulcer

synthetic; SK&F-96022, BY-1023

102625-70-7

2093 F15 Microsource 01505390 NISOLDIPINE vasodilator (coronary) synthetic; bayk-5552 63675-72-9

2093 F16 Microsource 01505819 ELETRIPTAN HYDROBROMIDE5-HT agonist, anti-migrane

synthetic; UK-116044-04

177834-92-3, 143322-58-1(base)

2093 F17 Microsource 01505392 TERBINAFINE HYDROCHLORIDE antifungal synthetic, SF-86-32778628-80-5, 91161-71-6(base)

2093 F18 Microsource 01505820 TOPOTECAN HYDROCHLORIDEantineoplastic; topoisomerase I inhibitor

semisynthetic 119413-54-6

2093 F19 Microsource 01505393 DESLORATIDINE H1-antihistaminesynthetic; SCH-34117

100643-71-8

2093 F20 Microsource 01505831 SITAGLIPTINDPP4 inhibitor, antidiabetic

synthetic

2093 F21 Microsource 01505396 FLUORESCEIN corneal trama indicator synthetic 2321-07-5

2093 F22 Microsource 01505851 ARIPIPRAZOLEantipsychotic, 5HT2A antagonist

synthetic; OPC-14597, OPC-31

129722-12-9

2093 G03 Microsource 01503423 SPIRAMYCIN antibacterialStreptomyces ambofaciens

8025-81-8

2093 G04 Microsource 01504269 LITHIUM CITRATE antidepressant synthetic6080-58-6, 919-16-4 [anhydrous]

2093 G05 Microsource 01503428 CHOLINE CHLORIDEcholeretic, lipotropic, hepatoprotectant

widespread in the plant and animal kingdoms

67-48-1, 62-49-7 [choline]

2093 G06 Microsource 01504272 GATIFLOXACIN antibacterialsynthetic; BMS-206584-01, AM-1155

160738-57-8

2093 G07 Microsource 01503429 CLOFIBRATE antihyperlipidemic synthetic 637-07-0

2093 G08 Microsource 01504273 MIGLITOLalpha-glucosidase inhibitor, antidiabetic

synthetic; BAYm-1099

72432-03-2

2093 G09 Microsource 01503500 RESORCINOL MONOACETATEantiseborrheic, antipruritic

synthetic 102-29-4

2093 G10 Microsource 01504300 ORLISTATreversible lipase inhibitor, antiobesity

synthetic 96829-58-2

2093 G11 Microsource 01503600 NIMODIPINE vasodilator synthetic 66085-59-42093 G12 Microsource 01504303 MOXIFLOXACIN HYDROCHLORIDE antibacterial synthetic 186826-86-8

2093 G13 Microsource 01503604 RETINYL PALMITATEprovitamin, antixerophthalamic

semisynthetic; Vitamin A palmitate

79-81-2

2093 G14 Microsource 01504401 PIOGLITAZONE HYDROCHLORIDE antidiabetic synthetic111025-46-8 (pioglitazone)

2093 G15 Microsource 01503607 THALIDOMIDE hypnotic synthetic 50-35-1

2093 G16 Microsource 01504402 TOLTERODINE TARTRATEmuscarinic receptor antagonist

synthetic 124937-51-5

2093 G17 Microsource 01503609 NITRENDIPINE antihypertensive synthetic 84845-75-0

2093 G18 Microsource 01504403 DONEPEZIL HYDROCHLORIDEacetylcholinesterase inhibitor (reversible), cognitive enhancer

synthetic; E-2020, BNAG

142057-77-0

2093 G19 Microsource 01503610 BENZALKONIUM CHLORIDE antiinfective (topical) synthetic 8001-54-5

2093 G20 Microsource 01505003 PIZOTYLINE MALATE5HT antagonist, antimigraine

synthetic; PIZOTIFEN; BC-105

5189-11-7

2093 G21 Microsource 01503611 PENTOXIFYLLINEPDE inhibitor, bronchodilator, vasodilator

synthetic 6493-05-6

2093 G22 Microsource 01505020 HOMOSALATE UV screen, analgesic synthetic 118-56-9

2093 H03 Microsource 01505397 NIACINAMIDEVitamin B3; enzyme cofactor; anti-pellagra

widespread in plants, yeasts, fungi

98-92-0

2093 H04 Microsource 01505881 DIZOCILPINE MALEATE neuroprotective synthetic; MK-801 77086-22-72093 H05 Microsource 01505398 PHENYLETHYL ALCOHOL antimicrobial synthetic 60-12-8

2093 H06 Microsource 01505906 ZILEUTON 5-lipoxygenase inhibitorsynthetic; Abbott-64077

111406-87-2

2093 H07 Microsource 01505399 OXYBUTYNIN CHLORIDE anticholinergicsynthetic; MJ-4309-1, 5058

1508-65-2

2093 H08 Microsource 01505907 METHYLPHENIDATE HYDROCHLORIDE CNS stimulant synthetic298-59-9, 113-45-1(base)

2093 H09 Microsource 01505410 BENURESTAT urease inhibitor synthetic; EU-2826 38274-54-3

2093 H10 Microsource 01505943 RABEPRAZOLE SODIUMgastric acid secretion inhibitor

synthetic; LY-307640, E-3810

117976-90-6

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ICCB-L Well

VendorVendor

IDCompound Name Bioactivity Source CAS

2093 H11 Microsource 01505411 BENZOXIQUINE antiinfective synthetic; NSC-3951 86-75-9

2093 H12 Microsource 01505944 RISEDRONATE SODIUM HYDRATE calcium regulator synthetic; NE-58095 115436-72-1

2093 H13 Microsource 01505412 BISMUTH SUBSALICYLATEantidiarrheal, antacid, antiulcer

synthetic 14882-18-9

2093 H14 Microsource 01505950 SUCRALFATE SODIUM (10% w/v in DMSO) antiulcer semisynthetic 54182-58-0 (free acid)

2093 H15 Microsource 01505413 BENZOYLPASantibacterial, tuberculostatic

synthetic 13898-58-3

2093 H16 Microsource 01505953 SUCRALOSE sweetener semisynthetic 56038-13-22093 H17 Microsource 01505414 BROMINDIONE anticoagulant synthetic 1146-98-1

2093 H18 Microsource 01505955 COLISTIN SULFATE antibacterialBacillus polymyxa colistinus; polymyxin E

1264-72-8

2093 H19 Microsource 01505417 CAPOBENIC ACID antiarrhythmic synthetic; C-3 21434-91-3

2093 H20 Microsource 01505957 ARSENIC TRIOXIDEantineoplastic, antileukemia

mineral 1327-53-3

2093 H21 Microsource 01505425 ACETOHEXAMIDE antidiabetic synthetic; 33006 968-81-02093 H22 Microsource 01505958 CLONAZEPAM anticonvulsant, sedative synthetic 1622-61-32093 I03 Microsource 01503614 CIPROFLOXACIN antibacterial, fungicide synthetic 85721-33-1

2093 I04 Microsource 01505024 OLANZAPINE antipsychoticsynthetic; LY-170053

132539-06-1

2093 I05 Microsource 01503650 NABUMETONE antiinflammatory synthetic 42924-53-8

2093 I06 Microsource 01505111 THIOSTREPTON antibacterialStreptomyces aureus

1393-48-2

2093 I07 Microsource 01503678 CELECOXIBantiarthritic, cyclooxygenase2 inhibitor

synthetic; SC-58635 169590-42-5

2093 I08 Microsource 01505112 TILMICOSIN antibacterial semisynthetic 108050-54-0

2093 I09 Microsource 01503705 ANETHOLEexpectorant, gastric stimulant, insecticide

anise, fennel and other plant oils

4180-23-8

2093 I10 Microsource 01505113 FLUNIXIN MEGLUMINEanalgesic, antiinflammatory

synthetic; SCH-14714

42461-84-7

2093 I11 Microsource 01503708 TERFENADINEH1 antihistamine, nonsedating

synthetic 50679-08-8

2093 I12 Microsource 01505114 CLIOQUINOL antiseptic, antiamebic synthetic 130-26-7

2093 I13 Microsource 01503710 CLOPIDOGREL SULFATEplatelet aggregation inhibitor

synthetic 113665-84-2

2093 I14 Microsource 01505115 CLORSULON antiparasitic, fasciolicide synthetic; MK-401 60200-06-8

2093 I15 Microsource 01503712 LORATADINE H1 antihistamine synthetic 79794-75-52093 I16 Microsource 01505116 ESTROPIPATE estrogen semisynthetic 7280-37-72093 I17 Microsource 01503720 SELAMECTIN antiparasitic, antimite semisynthetic 165108-07-62093 I18 Microsource 01505124 CLAVULANATE LITHIUM beta-lactamase inhibitor semisynthetic 58001-44-8(acid)

2093 I19 Microsource 01503722 ATORVASTATIN CALCIUMantihyperlipidemic, HMGCoA reductase inhibitor

synthetic134523-03-8, 134523-00-5 [atorvastatin]

2093 I20 Microsource 01505166 ALENDRONATE SODIUM

bone resorption inhibitor, farnesyldiphosphate synthetase inhibitor, antimetastatic

synthesis 121268-17-5

2093 I21 Microsource 01503721 ENROFLOXACIN antibacterial synthetic 93106-60-6

2093 I22 Microsource 01505172 ACARBOSE

alpha-glucosidase & saccharase inhibitor, antidiabetes, antihyperlipidaemia, antiobesity

Actinoplanes spp 56180-94-0

2093 J03 Microsource 01505426 ETHOXZOLAMIDEcarbonic anhydrase inhibitor, antiulcer, antiglaucoma

synthetic 452-35-7

2093 J04 Microsource 01505971 BENZBROMARONE uricosuricsynthetic; MJ-10061, L-2214

117976-90-6

2093 J05 Microsource 01505429 FLUCYTOSINE antifungalsynthetic; RO-2-9915

2022-85-7

2093 J06 Microsource 01505972 BROMPERIDOL antipsychotic synthetic; R-11333 10457-90-6

2093 J07 Microsource 01505432 FOMEPIZOLE HYDROCHLORIDEalcohol dehydrogenase inhibitor

synthetic; 4-MP 56010-888

2093 J08 Microsource 01505973 CYPROHEPTADINE HYDROCHLORIDEH1-antihistamine, antipruritic

synthetic 41354-29-4

2093 J09 Microsource 01505433 GLIPIZIDE antidiabeticsynthetic; CP-28720, K-4024

29094-61-9

2093 J10 Microsource 01505974 CLOFAZIMINEantibacterial, antilepretic, antituberculosis

synthetiNSC-141046c; G-30320

2030-63-9

2093 J11 Microsource 01505436 D-LACTITOL MONOHYDRATEsweetener, treatment of portoencephalopathy

semisynthetic 81025-04-9, 585-86-4

2093 J12 Microsource 01505975 BENZYDAMINE HYDROCHLORIDEanalgesic, antipyretic, antiinflammatory

synthetic; AF-864 132-69-4

2093 J13 Microsource 01505437 LEVOCARNITINEcofactor for fatty acid metabolism, replenisher in arterial disease

semisynthetic 541-15-1

Microsource1-US Drug Collection Page 19 of 24 Created 9/2015

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ICCB-L Well

VendorVendor

IDCompound Name Bioactivity Source CAS

2093 J14 Microsource 01505976 DOXAZOSIN MESYLATE antihypertensivesynthetic; UK-33274-27

77883-43-3

2093 J15 Microsource 01505438 HYDROCORTISONE VALERATEantiinflammatory, glucocorticoid

semisynthetic 57524-89-7

2093 J16 Microsource 01505977 ISOETHARINE MESYLATE bronchodilator synthetic 7279-75-6

2093 J17 Microsource 01505440 LOBENDAZOLE anthelminticsynthetic; SK&F-24529; NSC-42044

6306-71-4

2093 J18 Microsource 01505978 FLORFENICOL antibacterialsynthetic; SCH-25298

76639-94-6

2093 J19 Microsource 01505444 METHYLENE BLUEantimethemoglobinemic, cyanide antidote

synthetic 7220-79-3

2093 J20 Microsource 01505979 ETHYNODIOL DIACETATE progestinsemisynthetic; SC-11800

297-76-7

2093 J21 Microsource 01505445 METHYLATROPINE NITRATE anticholinergic semisynthetic 52-88-0

2093 J22 Microsource 01505981 ORNIDAZOLE antiinfectivesynthetic; 16773-42-5

16773-42-5

2093 K03 Microsource 01503801 NAPROXOLantinflammatory, analgesic, antipyretic

synthetic 26159-36-4

2093 K04 Microsource 01505178 ROPINIROLEdopamine receptor agonist, antiParkinsonian

synthetic; SK&F-101468

91374-21-9

2093 K05 Microsource 01503804 COLFORSINadenylate cyclase activator, antiglaucoma, hypotensive, vasodilator

Coleus forskohlii; HL-362; L-75-1362B

66575-29-9

2093 K06 Microsource 01505187 QUETIAPINE

antipsychotic: 5HT antagonist, dopamine antagonist, H1-antihistamine, alpha adrenergic blocker

synthetic; ICI-204636, ZD-5077, ZM-204639

111974-69-7

2093 K07 Microsource 01503807 ISOSORBIDE MONONITRATE antianginalsemisynthetic; BM-22145, IS-5-MN, AHR-4698

16051-77-7

2093 K08 Microsource 01505189 RIZATRIPTAN BENZOATE5HT-1B/1D agonist, antimigraine

synthetic; MK-0462 (benzoate)

144034-80-0

2093 K09 Microsource 01503816 AMCINONIDEglucocorticoid, antiinflammatory

synthetic 51022-69-6

2093 K10 Microsource 01505200 BENAZEPRIL HYDROCHLORIDEACE inhibitor, antihypertensive

synthetic 86541-74-4

2093 K11 Microsource 01503818 BUPIVACAINE HYDROCHLORIDE anesthetic (local) synthetic

14252-80-3, 2180-92-9 [bupivacaine], 18010-40-7 [anhydrous]

2093 K12 Microsource 01505201 FAMCICLOVIR antiviral synthetic 104227-87-42093 K13 Microsource 01503903 ALBENDAZOLE anthelmintic synthetic 54965-21-8

2093 K14 Microsource 01505203 EZETIMIBE sterol absorption inhibitor synthetic 163222-33-1

2093 K15 Microsource 01503908 PACLITAXEL antineoplastic Taxus breviofolia 33069-62-4

2093 K16 Microsource 01505205 OLMESARTAN MEDOXOMILAngiotensin II inhibitor prodrug, antihypertensive

synthetic 144689-63-4

2093 K17 Microsource 01503914 BUTACAINE anesthetic (local) synthetic149-15-5, 149-16-6 [butacaine]

2093 K18 Microsource 01505207 CEFTIBUTEN antibacterial semisynthetic 97519-39-6

2093 K19 Microsource 01503918 CLOBETASOL PROPIONATEglucocorticoid, antiinflammatory

synthetic25122-46-7, 25122-41-2 [clobetasol]

2093 K20 Microsource 01505208 CEFDINIR antibacterialsemisynthetic; CL-983, FK-482

91832-40-5

2093 K21 Microsource 01503919 CLOPAMIDE diuretic synthetic 636-54-4

2093 K22 Microsource 01505209 VALSARTANAngiotensin II inhibitor, antihypertensive

synthetic; CGP-48933

137862-53-4

2093 L03 Microsource 01505449 PRALIDOXIME CHLORIDE cholesterase agonist synthetis; 2-PAM 51-15-0

2093 L04 Microsource 01505982 OXANTEL PAMOATE anthelminticsynthetic; CP-14445-16

68813-55-8

2093 L05 Microsource 01505450 PREDNISOLONE HEMISUCCINATEantiinflammatory, glucocorticoid

semisynthetic 2920-86-7

2093 L06 Microsource 01505983 PHENFORMIN HYDROCHLORIDE antidiabetic synthetic 834-28-6

2093 L07 Microsource 01505453 PYRIDOXINEvitamin B6, enzyme cofactor

rice husks, wheat germ, yeast

65-23-6

2093 L08 Microsource 01505984 PROTRYPTYLINE HYDROCHLORIDE antidepressant synthetic; MK-240 1225-55-42093 L09 Microsource 01505460 RIMANTADINE HYDROCHLORIDE antiviral synthetic; EXP-126 1501-84-42093 L10 Microsource 01505986 NIALAMIDE MAO inhibitor 51-12-72093 L11 Microsource 01505461 SULFISOXAZOLE ACETYL antibacterial synthetic 80-74-0

2093 L12 Microsource 01505987 DENATONIUM BENZOATEdenaturing agent, bitter principle

synthetic 3734-33-6

2093 L13 Microsource 01505463 TAURINE

neuroprotectant, inhibitory neurotransmitter, GABA agonist

widespread in animal tissue

107-35-7

2093 L14 Microsource 01505993 MESALAMINE antiinflammatory synthetic; 5-ASA 89-57-6

2093 L15 Microsource 01505464 THIAMINEvitamin B1, enzyme cofactor

rice husks, wheat germ, yeast

67-03-8

2093 L16 Microsource 02300061 CLOMIPRAMINE HYDROCHLORIDE antidepressant synthetic17321-77-6, 303-49-1 [clomipramine]

2093 L17 Microsource 01505465 TRICLOSAN antiinfective synthetic; CH-3565 3380-34-5

Microsource1-US Drug Collection Page 20 of 24 Created 9/2015

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VendorVendor

IDCompound Name Bioactivity Source CAS

2093 L18 Microsource 02300094 ASTEMIZOLEH1 antihistamine (nonsedating)

synthetic 68844-77-9

2093 L19 Microsource 01505467 ZINC UNDECYLENATE antifungal synthetic 557-08-4

2093 L20 Microsource 02300154 ACECAINIDE HYDROCHLORIDE antiarrhythmic synthetic34118-92-8, 32795-44-1 [acecainide]

2093 L21 Microsource 01505468 UNDECYLENIC ACID antifungal semisynthetic 112-38-9

2093 L22 Microsource 02300173 BUSPIRONE HYDROCHLORIDE5HT1a receptor agonist, anxiolytic

synthetic33386-08-2, 36505-84-7 [buspirone]

2093 M03 Microsource 01503923 IOPANIC ACID radioopaque agent synthetic 96-83-3

2093 M04 Microsource 01505210 SIBUTRAMINE HYDROCHLORIDE

anorexic, antidepressant, uptake inhibitor (5HT, norepinephrine, dopamine)

synthetic84485-00-7; 106650-56-0 (base); 125494-59-9 (hydrate)

2093 M05 Microsource 01503925 KETOROLAC TROMETHAMINE antiinflammatory synthetic74103-07-4, 74103-06-3 [ketorolac]

2093 M06 Microsource 01505212 PERINDOPRIL ERBUMINEantihypertensive, ACE inhibitor

synthetic; S9490-3, McN-A2833-109

107133-36-8; 82834-16-0 (perindopril)

2093 M07 Microsource 01503926 LANSOPRAZOLE antiulcer synthetic 103577-45-3

2093 M08 Microsource 01505213 ROSUVASTATIN CALCIUM antihyperlipidemic synthetic287714-14-4, 147098-20-2(Ca salt)

2093 M09 Microsource 01503929 MEXILETINE HYDROCHLORIDE antiarrhythmic synthetic; KO-11735370-01-4, 31828-71-4 [mexiletine]

2093 M10 Microsource 01505214 RAMIPRILantihypertensive, ACE inhibitor

synthetic; HOE-498 87333-19-5

2093 M11 Microsource 01503931 MORANTEL CITRATE anthelmintic synthetic26155-31-7, 20574-50-9 [morantel]

2093 M12 Microsource 01505222 DERACOXIBantiinflammatory, antiarthritic, COX-2 inhibitor

synthetic 169590-41-4

2093 M13 Microsource 01503932 OXYPHENCYCLIMINE HYDROCHLORIDE anticholinergic synthetic125-52-0, 125-53-1 [oxyphencyclimine]

2093 M14 Microsource 01505230 CILOSTAZOLphosphodiesterase inhibitor

synthetic 73963-72-1

2093 M15 Microsource 01503934 PERPHENAZINE antipsychotic synthetic 58-39-9

2093 M16 Microsource 01505244 CITICOLINE

cognition enhancer, phosphocholine cytidyltransferase activator

cytidine-5'-diphosphocholine

987-78-0

2093 M17 Microsource 01503935 PROPAFENONE HYDROCHLORIDE antiarrhythmic synthetic34183-22-7, 54063-53-5 [propafenone]

2093 M18 Microsource 01505248 CANRENONEaldosterone antagonist; antifibrogenic

synthetic 976-71-6

2093 M19 Microsource 01503968 TACROLIMUSimmune suppressant, antifungal

Streptomyces tsukubaensis

109581-93-3, 104987-11-3 [anhydrous]

2093 M20 Microsource 01505249 APRAMYCINantibacterial; LD50(iv) 280mg/kg(mouse)

Streptomyces tenebrarius, Saccharomyces porispora hiltus

37321-09-8

2093 M21 Microsource 01503975 FLUCONAZOLE antifungal synthetic 86386-73-4

2093 M22 Microsource 01505261 TELMISARTANantihypertensive, angiotensin II blocker

synthetic; BIBR-277 SE

144701-48-4

2093 N03 Microsource 01505470CLINDAMYCIN PALMITATE HYDROCHLORIDE

antibacterial, inhibits protein synthesis

semisynthetic; U-25179E

25507--04-4

2093 N04 Microsource 02300205 LEVODOPA antiparkinsonianVicia faba seedlings, Sarothamnus spp, & other palnts

59-92-7

2093 N05 Microsource 01505474 CEFONICID SODIUM antibacterialsemisynthetic; SK&F-D-75073-Z

71420-79-6

2093 N06 Microsource 02300104 TACRINE HYDROCHLORIDEanticholinesterase, cognitive adjuvant, K channel blocker

synthetic; CL-970 1684-40-8

2093 N07 Microsource 01505480 IFOSFAMIDE antineoplasticsynthetic; MJF-9325, Z-4942, NSC-109724

3778-73-2

2093 N08 Microsource 02300161 AMOXAPINEantidepressant, inhibits norepinephrine uptake

synthetic 14028-44-5

2093 N09 Microsource 01505482 NETILMICIN SULFATE antibacterialsemisynthetic; SCH-20569

56391-56-1

2093 N10 Microsource 02300165 AMIODARONE HYDROCHLORIDEadrenergic agonist, coronary vasodilator, Ca channel blocker

synthetic 1951-25-3

2093 N11 Microsource 01505483 DOXORUBICIN antineoplastic semisynthetic 23214-92-8

2093 N12 Microsource 02300206 DIAZOXIDEantihypertensive, diuretic, activates K channels and AMPA receptors

synthetic; SCH-6783; NSC-64198

364-98-7

2093 N13 Microsource 01505492 METHYSERGIDE MALEATEvasoconstrictor, antimigraine

semisynthetic 129-49-7

2093 N14 Microsource 02300214 DILTIAZEM HYDROCHLORIDECa channel blocker, coronary vasodilator

synthetic33286-22-5, 42399-41-7 [diltiazem]

2093 N15 Microsource 01505498 ACEPROMAZINE MALEATE sedative synthetic 3598-37-6

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VendorVendor

IDCompound Name Bioactivity Source CAS

2093 N16 Microsource 02300219 EDROPHONIUM CHLORIDEacetylcholinesterase inhibitor

synthetic116-38-1, 312-48-1 [edrophonium]

2093 N17 Microsource 01505514 BIPERIDENanticholinergic, antiparkinsonian

synthetic 514-65-8

2093 N18 Microsource 02300176 PHENOXYBENZAMINE HYDROCHLORIDE alpha adrenergic blocker synthetic63-92-3, 59-96-1 [phenoxybenzamine]

2093 N19 Microsource 01505530 DEXCHLORPHENIRAMINE MALEATE antihistamine synthetic 2438-32-6

2093 N20 Microsource 02300242 LOXAPINE SUCCINATE antipsychotic synthetic27833-64-3, 1977-10-2 [loxapine]

2093 N21 Microsource 01505532 DILOXANIDE FUROATE amoebicide synthetic 3736-81-0

2093 N22 Microsource 02300212 DOMPERIDONEantiemetic, dopamine antagonist

synthetic; R-33812 57808-66-9

2093 O03 Microsource 01503977 LOVASTATINantihyperlipidemic, HMGCoA reductase inhibitor

Aspergillus spp; mevinolin

75330-75-5

2093 O04 Microsource 01505262 SERTRALINE HYDROCHLORIDEantidepressant, 5HT uptake inhibitor

synthetic79559-97-0; 79617-96-2(base)

2093 O05 Microsource 01503978 HYDROXYCHLOROQUINE SULFATEantimalarial, lupus suppressant

synthetic747-36-4, 118-42-3 [hydroxychloroquine]

2093 O06 Microsource 01505263 ALFLUZOSINalpha(1)-adrenergic blocker

synthetic; SL-77499 81403-80-7

2093 O07 Microsource 01503985 BROMPHENIRAMINE MALEATE H1 antihistamine synthetic980-71-2, 86-22-6 [brompheniramine]

2093 O08 Microsource 01505267 OXAPROZIN antiinflammatory synthetic; WY-21743 21256-18-8

2093 O09 Microsource 01504008 SIROLIMUSimmunosuppressant, antineoplastic; rapamycin

Streptomyces hygroscopicus

53123-88-9

2093 O10 Microsource 01505270 PROPRANOLOL HYDROCHLORIDE (+/-)antihypertensive, antianginal, antiarrhythmic

synthetic318-98-9, 525-66-6 [propranolol]

2093 O11 Microsource 01504085 PAROXETINE HYDROCHLORIDE antidepressant synthetic 61869-08-72093 O12 Microsource 01505271 CROTAMITON antipruritic, scabicide synthetic 483-63-6

2093 O13 Microsource 01504088ETHYLNOREPINEPHRINE HYDROCHLORIDE

bronchodilator synthetic3198-07-0, 536-24-3 [ethylnorepinephrine]

2093 O14 Microsource 01505281 ZOLMITRIPTANantimigraine, 5HT[1B/1D] agonist

synthetic 139264-17-8

2093 O15 Microsource 01504094 TENIPOSIDE antineoplastic semisynthetic 29767-20-22093 O16 Microsource 01505296 OXFENDAZOLE anthelmintic synthetic 53716-50-0

2093 O17 Microsource 01504099 SILDENAFILerectile dysfunction therapy

synthetic 139755-83-2

2093 O18 Microsource 01505299 AMITRAZ scabicide synthetic; U-36059 33089-61-1

2093 O19 Microsource 01504078 SENNOSIDE A catharticCassia & Rheum spp

81-27-6

2093 O20 Microsource 01505294 CARBADOX antibacterial synthetic 6804-07-5

2093 O21 Microsource 01504105 TANNIC ACIDnonspecific enzyme/receptor blocker

principal constituent of tree galls, esp Quercus spp;

1401-55-4

2093 O22 Microsource 01505292 NONOXYNOL-9spermatocide, contraceptive

synthetic 26027-38-3

2093 P03 Microsource 01505537 ETIDRONATE DISODIUM bone resorption inhibitor synthetic 7414-83-72093 P04 Microsource 02300229 GLYBURIDE antihyperglycemic synthetic 10238-21-82093 P05 Microsource 01505551 LEVOBUNOLOL HYDROCHLORIDE beta-adrenergic blocker synthetic 17912-14-7

2093 P06 Microsource 02300259 NICOTINE DITARTRATEnicotinyl acetylchloline receptor agonist, ectoparasiticide

Nicotiana tabacum 65-31-6

2093 P07 Microsource 01505560 NATAMYCIN antibacterialSteptomyces natalensis; CL-12625, A-5283

7681-93-8

2093 P08 Microsource 02300292 MIANSERIN HYDROCHLORIDE 5HT antagonist synthetic21535-47-7, 24219-97-4 [mianserin]

2093 P09 Microsource 01505562 NORGESTIMATE progestin semisynthetic 35189-28-7

2093 P10 Microsource 02300309 VESAMICOL HYDROCHLORIDEacetylcholine transport blocker (vesicular)

synthetic 120447-62-3

2093 P11 Microsource 01505581 TIOCONAZOLE antifungal synthetic; UK-20349 65899-73-2

2093 P12 Microsource 02300307 VERAPAMIL HYDROCHLORIDE

adrenegic blocker, Ca channel blocker, coronary vasodilator, antiarrhythmic

synthetic152-11-4, 52-53-9 [verapamil]

2093 P13 Microsource 01505584 ERGOTAMINE TARTRATE analgesic, antimigraine Claviceps purpurea 379-79-3

2093 P14 Microsource 02300325 METOLAZONE diuretic, antihypertensive synthetic 17560-51-9

2093 P15 Microsource 01505590 ANAGRELIDE HYDROCHLORIDE antithrombotic synthetic; BL-4162a 58579-51-4

2093 P16 Microsource 02300332 PODOFILOX

antineoplastic, inhibits microtubule assembly, and human DNA topoisomerase II; antimitotic agent

Podophylum peltatum; podophylotoxin

518-28-5

2093 P17 Microsource 01505599 ETOMIDATE sedative synthetic 33125-97-2

2093 P18 Microsource 02300347 PENTYLENETETRAZOLanaleptic, circulation stimulant

synthetic 54-95-5

2093 P19 Microsource 01505600 FELBAMATEanticonvulsant, antiepileptic

synthetic; W-554 25451-15-4

Microsource1-US Drug Collection Page 22 of 24 Created 9/2015

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ICCB-L Plate

ICCB-L Well

VendorVendor

IDCompound Name Bioactivity Source CAS

2093 P20 Microsource 01505715 PANTOTHENIC ACID(d) Na salt vitamin B5 rice bran, queen bee jelly

63409-48-3

2093 P21 Microsource 01505610 LAMOTRIGINE anticonvulsant synthetic; BW-430C 84057-84-1

2093 P22 Microsource 01505729 DOCOSANOL antiviral Pygeum africanum 661-19-82094 A03 Microsource 01505742 ASCORBYL PALMITATE antioxidant semisynthetic 137-66-62094 A05 Microsource 01505753 GLYCOPYRROLATE anticholinergic synthetic; AHR-504 596-51-02094 A07 Microsource 01505759 OXTRIPHYLLINE bronchodilator synthetic 4499-40-52094 A09 Microsource 01505760 OCTISALATE sunscreen synthetic 118-60-52094 A11 Microsource 01505777 DIATRIZOIC ACID radiopaque agent synthetic 117-96-4

2094 A13 Microsource 01505880 DIFLORASONE DIACETATEantiinflammatory, glucocorticoid

semisynthetic; U-34865

33564-31-7

2094 A15 Microsource 01505985 NIZATIDINE antiulcer, H2 antagonistsynthetic; LY-139037

76963-41-2

2094 A17 Microsource 01505991 DECAMETHONIUM BROMIDE neuromuscular blocker synthetic 541-22-0

2094 A19 Microsource 01505994 ETHAMIVANCNS & respiratory stimulant

synthetic; NCS-406087

304-84-7

2094 A21 Microsource 01505995 BUTYL PARABEN antifungal, preservative synthetic 94-26-8

2094 C03 Microsource 01505996 AZTREONAM antibacterial synthetic; SQ-26776 78110-38-0

2094 C05 Microsource 01506009 METHIMAZOLE thyroid inhibitor synthetic 60-56-0

2094 C07 Microsource 01506035 REPAGLINIDE antidiabeticsynthetic; AG-EE-623-ZW

135062-02-1

2094 C09 Microsource 01506053 TYLOXAPOLpolymeric nonionic detergent

synthetic 25301-02-4

2094 C11 Microsource 01506066 DEBRISOQUIN SULFATE anti-hypertensivesynthetic; RO-5-3307/1

581-88-4

2094 C13 Microsource 01506067 ENILCONAZOLE antifungal synthetic; R-23979 35554-44-0

2094 C15 Microsource 01506074 JOSAMYCIN antibacterialsemisynthetic; EN-141

56689-45-3

2094 C17 Microsource 01506084 PROSCILLARIDIN cardiotonicScilla spp; A-32686, 2936

466-06-8

2094 C19 Microsource 01506086 SULFADOXINE antibacterialsynthetic; RO-4-4393

2447-57-6

2094 C21 Microsource 01506069 FINASTERIDEanti-androgen, alpha-reductase inhibitor

synthetic; MK=909 98319-26-7

2094 E03 Microsource 01506082 PENTETIC ACIDchelating agent, diagnostic aid

synthetic; DTPA 67-43-6

2094 E05 Microsource 01506043 SOTALOL HYDROCHLORIDE beta-adrenergic agonist synthetic; MJ-1999 959-24-0

2094 E07 Microsource 01506029 PEPSTATIN Aaspartyl protease inhibitor

Actinomyces spp 26305-03-3

2094 E09 Microsource 01505420 DEXPANTHENOL cholinergic semisynthetic 81-13-02094 E11 Microsource 01601020 DIETHYLTOLUAMIDE insect repellant synthetic; DEET 134-62-32094 E13 Microsource 01505202 AMLODIPINE BESYLATE Ca channel blocker synthetic 111470-99-6

2094 E15 Microsource 01503692 BLEOMYCIN (bleomycin B2 shown) antineoplastic[Bleocin (TM) 3.5% Cu]; Streptomyces verticillis

9041-93-4, 11056-06-7 [bleomycin]

2094 E17 Microsource 01505022 PROPOFOL anesthetic synthetic; ICI-35868 2078-54-8

2094 E19 Microsource 01503216 FILIPIN antifungalStreptomyces filipinensis

480-49-9

2094 E21 Microsource 01900006 PENTOBARBITAL anesthetic synthetic 76-74-4

2094 G03 Microsource 01900005 THIOPENTAL SODIUM anesthetic synthetic71-73-8, 76-75-5 [thiopental]

2094 G05 Microsource 01900002 THIAMYLAL SODIUM anesthetic synthetic337-47-3, 77-27-0 [thiamylal]

2094 G07 Microsource 01505348 RILUZOLEanticonvulsant, glutamate release inhibitor, anti-ALS

synthetic 1744-22-5

2094 G09 Microsource 01505485 PHYTONADIONE vitamin semisynthetic 84-80-0

2094 G11 Microsource 01505905COLESEVALAM HYDROCHLORIDE (high mol wt copolymer @10mg/ml)

antihyperlipidemic, cholesterol sequestrant

synthetic; GT-31-104 182815-44-7

2094 G13 Microsource 01503266 NOCODAZOLE antineoplastic, antimitotic synthetic; R-17934 31430-18-9

2094 G15 Microsource 01500363 LACTULOSE laxative synthetic 4618-18-2

2094 G17 Microsource 01500567 TETRAHYDROZOLINE HYDROCHLORIDEadrenergic agonist, nasal decongestant

synthetic522-48-5, 84-22-0 [tetrahydrozoline]

2094 G19 Microsource 01500464 PENICILLAMINEchelating agent (Cu), antirheumatic

semisynthetic 52-67-5

2094 G21 Microsource 02300270 PINACIDILK channel agonist, antihypertensive

synthetic85371-64-8, 60560-33-0 [anhydrous]

2094 I03 Microsource 01505346 KETANSERIN TARTRATE5HT2/5HT1C seritonin antagonist

synthetic; R4146883846-83-7, 74050-98-9(base)

2094 I05 Microsource 01500304 FLUOROMETHOLONEglucocorticoid, antiinflammatory

semisynthetic 426-13-1

2094 I07 Microsource 01506014 METYRAPONE diagnostic aid synthetic 54-36-4

2094 I09 Microsource 01500274 ADRENALINE BITARTRATEadrenergic agonist, bronchodilator, antiglaucoma agent

Portulaca grandiflora 51-42-3

2094 I11 Microsource 01504150 MELOXICAM SODIUM antiinflammatory synthetic 71125-38-7

Microsource1-US Drug Collection Page 23 of 24 Created 9/2015

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ICCB-L Plate

ICCB-L Well

VendorVendor

IDCompound Name Bioactivity Source CAS

2094 I13 Microsource 01500813 BUDESONIDE antiinflammatory semisynthetic

51333-22-3 [11(gr b), 16(gr a)] 51372-29-3 [(11(gr b), 16(gr a)[//R//])] 51372-28-2 [(11(gr b), 16(gr a)[//S//])]

2094 I15 Microsource 01500275 EQUILIN estrogen pregnant mare urine 474-86-2

2094 I17 Microsource 02300009 TILORONE antiviral synthetic27591-69-1, 27591-97-5 [tilorone]

2094 I19 Microsource 01505012 EXEMESTANEantineoplastic, aromatase inhibitor

synthetic; PNU-155971, FCE-24304

107868-30-4

2094 I21 Microsource 01505333 TRANILASTantiallergic, mast cell degranulation inhibitor, angiogenesis blocker

synthetic; MK-341 53902-12-8

2094 K03 Microsource 01503232 PROCATEROL HYDROCHLORIDEbeta-adrenergic agonist, bronchodilator

synthetic59828-07-8, 72332-33-3 [procaterol], 60443-17-6 [replaced]

2094 K05 Microsource 01500248 DIHYDROERGOTAMINE MESYLATEvasoconstrictor, antimigraine

semisynthetic 6190-39-2

2094 K07 Microsource 01503078 ANIRACETAM cognitive enhancer synthetic 72432-10-1

2094 K09 Microsource 02300241 LOPERAMIDE HYDROCHLORIDE Ca channel blocker synthetic34552-83-5, 53179-11-6 [loperamide]

2094 K11 Microsource 01500422 NALOXONE HYDROCHLORIDE narcotic antagonist synthetic357-08-4, 51481-60-8 [dihydrate], 465-65-6 [naloxone]

2094 K13 Microsource 01501196 FLUMETHASONE antiinflammatory semisynthetic 2135-17-32094 K15 Microsource 01500261 DISOPYRAMIDE PHOSPHATE antiarrhythmic synthetic 3737-09-52094 K17 Microsource 01505434 HALOTHANE anesthetic synthesis 151-67-72094 K19 Microsource 01300030 OMEGA-3-ACID ESTERS (EPA shown) hypolipidemic semisynthetic; K-85 86227-47-6

2094 K21 Microsource 01300028 MANNITOLdiuretic, sweetener, diagnostic aid

manna and seaweeds; exudates of olive and plane trees

69-65-8

2094 M03 Microsource 01505426 ETHOXZOLAMIDEcarbonic anhydrase inhibitor, antiulcer, antiglaucoma

synthetic 452-35-7

2094 M05 Microsource 01504231 CLARITHROMYCIN antibacterialStreptomyces erythreus

81103-11-9

2094 M07 Microsource 01500368 LINCOMYCIN HYDROCHLORIDE antibacterial

Streptomyces lincolnensis, S espinosus, S variabilis

7179-49-9, 859-18-7 [anhydrous], 154-21-2 [lincomycin]

2094 M09 Microsource 01503373 OXIBENDAZOLE anthelmintic synthetic 20559-55-1

2094 M11 Microsource 01503679 AZITHROMYCIN antibacterial semisynthetic83905-01-5, 117772-70-0 [dihydrate]

2094 M13 Microsource 01505447 OCTODRINEvasoconstrictor, anesthetic (local)

synthetic; SK&F-51 543-82-8

2094 M15 Microsource 01505956 NITROGLYCERIN vasodilator (coronary)synthetic; SDM-7, SDM-17, SDM-20, SDM-26, SDM-27

55-63-0

2094 M17 Microsource 01505265 TELITHROMYCIN antibacterialsemisynthetic; HMR-3647

191114-48-4

2094 M19 Microsource 01300039 SODIUM PHENYLACETATE antihyperammonemic synthetic 114-70-5

2094 M21 Microsource 01502036 VIGABATRIN anticonvulsantsynthetic; MDL-71754

60643-86-9

2094 O03 Microsource 01505688 PROPARACAINE HYDROCHLORIDE local anesthetic synthetic 575-06-98

2094 O05 Microsource 01505707 TEICOPLANIN [A(2-1) shown] antibacterialActinoplanes teichomyceticus; MDL-507

61036-62-2

2094 O07 Microsource 01504183 TRIFLURIDINE antiviral (opthalmic) synthetic 70-00-82094 O09 Microsource 01503938 RIBAVIRIN antiviral synthetic 36791-04-52094 O11 Microsource 01505705 FLUDARABINE PHOSPHATE antineoplastic synthetic; 75607-67-92094 O13 Microsource 01504263 ROSIGLITAZONE antidiabetic synthetic 122320-73-4

2094 O15 Microsource 01505684 ROLITETRACYCLINE antibacterialsemisynthetic; SQ-15659

751-97-3

2094 O17 Microsource 01505703 ALTRENOGEST progestinantineoplasticsynthetic; RU-2267, A-35957

850-52-2

2094 O19 Microsource 01505704 BISOPROLOL FUMARATEbeta-blocker, antihypertensive

synthetic; CL-297939

104344-23-2

2094 O21 Microsource 01503432 MEPARTRICIN antifungal, antiprotozoalStreptomyces aureofaciens

11121-32-7

Microsource1-US Drug Collection Page 24 of 24 Created 9/2015