ChemInform Abstract: Microwave-Assisted Three-Component Coupling-Addition-SNAr (CASNAR) Sequences to...

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ChemInform 2010, 41, issue 21 © 2010 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim www.cheminform.wiley-vch.de Thiopyran derivatives R 0370 DOI: 10.1002/chin.201021142 Microwave-Assisted Three-Component Coupling-Addition-S N Ar (CASNAR) Se- quences to Annelated 4H-Thiopyran-4-ones. — A diversity of fused thiopyranones, e.g. (III), (V), (IX) or (XI), is synthesized by Sonogashira coupling of o-halo-(het)aroyl chlorides with terminal alkynes followed by microwave-assisted cyclization with sodi- um sulfide. — (WILLY, B.; FRANK, W.; MUELLER*, T. J. J.; Org. Biomol. Chem. 8 (2010) 1, 90-95; Inst. Org. Chem. Makromol. Chem., Heinrich-Heine-Univ., D-40225 Duesseldorf, Germany; Eng.) — Mischke 21- 142

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Thiopyran derivativesR 0370 DOI: 10.1002/chin.201021142

Microwave-Assisted Three-Component Coupling-Addition-SNAr (CASNAR) Se-quences to Annelated 4H-Thiopyran-4-ones. — A diversity of fused thiopyranones, e.g. (III), (V), (IX) or (XI), is synthesized by Sonogashira coupling of o-halo-(het)aroyl chlorides with terminal alkynes followed by microwave-assisted cyclization with sodi-um sulfide. — (WILLY, B.; FRANK, W.; MUELLER*, T. J. J.; Org. Biomol. Chem. 8 (2010) 1, 90-95; Inst. Org. Chem. Makromol. Chem., Heinrich-Heine-Univ., D-40225 Duesseldorf, Germany; Eng.) — Mischke

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ChemInform 2010, 41, issue 21 © 2010 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim