A full list of publications is available for download as PDF document.
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DIETER ENDERS VERÖFFENTLICHUNGEN 1) D. Seebach, D. Enders, Angew. Chem. 1972, 84, 350 - 351; Angew. Chem. Int. Ed. Engl. 1972, 11, 301 - 302. C-C-Verknüpfungen in α-Stellung zum Stickstoff sekun- därer Amine. Lithium-dimethylnitrosamin. 2) D. Enders, Diplomarbeit, Universität Gießen, 1972. C-C-Verknüpfungen in α-Stel- lung zum Stickstoff sekundärer Amine. Lithium-dimethylnitrosamin. 3) D. Seebach, D. Enders, Angew. Chem. 1972, 84, 1186 - 1187; Angew. Chem. Int. Ed. Engl. 1972, 11, 1101 - 1102. Metallierung am primären, sekundären und tertiären C-Atom offenkettiger und cyclischer Nitrosamine. 4) D. Seebach, D. Enders, Angew. Chem. 1972, 84, 1187; Angew. Chem. Int. Ed. Engl. 1972, 11, 1102 - 1103. Reaktion metallierter Nitrosamine mit Nitrilen. Eine neue Methode zur Darstellung von v-Triazolen. 5) D. Seebach, D. Enders, B. Renger, W. Bruegel, Angew. Chem. 1973, 85, 504; Angew. Chem. Int. Ed. Engl. 1973, 12, 495. Isolierung und Identifizierung von v- Tetrazinderivaten aus dem Zerfall von Nitrosamin-Anionen. 6) D. Enders, D. Seebach, Angew. Chem. 1973, 85, 1104; Angew. Chem. Int. Ed. Engl. 1973, 12, 1014. Nucleophile Thioacylierung mit Lösungen von Dimethylthiocarba- moyllithium. 7) D. Enders, Dissertation Universität Gießen, 1974. Nucleophile α-sekundäre Aminoalkylierung über metallierte Nitrosamine. 8) D. Enders, M. Kolb, Chemie für Labor und Betrieb 1974, 25, 337 - 346. Die Wood- ward-Hoffmann-Regeln. Eine einfache Einführung I. 9) D. Enders, M. Kolb, Chemie für Labor und Betrieb 1974, 25, 392 - 399. Die Wood- ward-Hoffmann-Regeln. Eine einfache Einführung II. 10) D. Seebach, D. Enders, J. Med. Chem. 1974, 17, 1225 - 1227. Synthesis of α- Heterosubstituted Nitrosamines - Novel Test Substances for Cancer and Mutagenesis Research? 22.01.18
Transcript of A full list of publications is available for download as PDF document.
DIETER ENDERS
VERÖFFENTLICHUNGEN
1) D. Seebach, D. Enders, Angew. Chem. 1972, 84, 350 - 351; Angew. Chem. Int. Ed.
Engl. 1972, 11, 301 - 302. C-C-Verknüpfungen in α-Stellung zum Stickstoff sekun-
därer Amine. Lithium-dimethylnitrosamin.
2) D. Enders, Diplomarbeit, Universität Gießen, 1972. C-C-Verknüpfungen in α-Stel-
lung zum Stickstoff sekundärer Amine. Lithium-dimethylnitrosamin.
3) D. Seebach, D. Enders, Angew. Chem. 1972, 84, 1186 - 1187; Angew. Chem. Int.
Ed. Engl. 1972, 11, 1101 - 1102. Metallierung am primären, sekundären und
tertiären C-Atom offenkettiger und cyclischer Nitrosamine.
4) D. Seebach, D. Enders, Angew. Chem. 1972, 84, 1187; Angew. Chem. Int. Ed. Engl.
1972, 11, 1102 - 1103. Reaktion metallierter Nitrosamine mit Nitrilen. Eine neue
Methode zur Darstellung von v-Triazolen.
5) D. Seebach, D. Enders, B. Renger, W. Bruegel, Angew. Chem. 1973, 85, 504;
Angew. Chem. Int. Ed. Engl. 1973, 12, 495. Isolierung und Identifizierung von v-
Tetrazinderivaten aus dem Zerfall von Nitrosamin-Anionen.
6) D. Enders, D. Seebach, Angew. Chem. 1973, 85, 1104; Angew. Chem. Int. Ed. Engl.
1973, 12, 1014. Nucleophile Thioacylierung mit Lösungen von Dimethylthiocarba-
moyllithium.
7) D. Enders, Dissertation Universität Gießen, 1974. Nucleophile α-sekundäre
Aminoalkylierung über metallierte Nitrosamine.
8) D. Enders, M. Kolb, Chemie für Labor und Betrieb 1974, 25, 337 - 346. Die Wood-
ward-Hoffmann-Regeln. Eine einfache Einführung I.
9) D. Enders, M. Kolb, Chemie für Labor und Betrieb 1974, 25, 392 - 399. Die Wood-
ward-Hoffmann-Regeln. Eine einfache Einführung II.
10) D. Seebach, D. Enders, J. Med. Chem. 1974, 17, 1225 - 1227. Synthesis of α-
Heterosubstituted Nitrosamines - Novel Test Substances for Cancer and
Mutagenesis Research?
22.01.18
2
11a) D. Seebach, D. Enders, Angew. Chem. 1975, 87, 1 - 18; Angew. Chem. Int. Ed.
Engl. 1975, 14, 15 - 32. Umpolung der Reaktivität von Aminen. Nucleophile α-
sekundäre Aminoalkylierung über metallierte Nitrosamine.
b) D. Seebach, D. Enders, in New Synthetic Methods, Vol. 2, Verlag Chemie
Weinheim, 1975, Umpolung of Amine Reactivity, Nucleophilic α- (secondary
Amino)-Alkylation via Metalated Nitrosamines.
12) D. Seebach, D. Enders, Chem. Ber. 1975, 108, 1293 - 1320. Lithiierte Methylnitros-
amine. Nucleophile α-sekundäre Aminomethylierung.
13) P. Bischof, R. Gleiter, R. Dach, D. Enders, D. Seebach, Tetrahedron 1975, 31, 1415
- 1417. Zur Wechselwirkung einsamer Elektronenpaare in ∆2-Tetrazenen.
Photoelektronenspektroskopische Untersuchungen.
14) E. J. Corey, D. Enders, Tetrahedron Lett. 1976, 3 - 6. Applications of N,N-
Dimethylhydrazones to Synthesis. Use in Efficient, Positionally and
Stereochemically Selective C-C-Bond Formation; Oxidative Hydrolysis of Carbonyl
Compounds.
15) E. J. Corey, D. Enders, Tetrahedron Lett. 1976, 11 - 14. Synthetic Routes to
Polyfunctional Molecules via Metalated N,N-Dimethyl-Hydrazones.
16) E. J. Corey, D. Enders, M. G. Bock, Tetrahedron Lett. 1976, 7 - 10 . A Simple and
Highly Effective Route to α,β-Unsaturated Aldehydes.
17) D. Seebach, W. Lubosch, D. Enders, Chem. Ber. 1976, 109, 1309 - 1323.
Nucleophile Thioacylierung mit Thiocarbamoyllithium-Derivaten von sekundären
Aminen.
18) D. Enders, T. Hassel, R. Pieter, B. Renger, D. Seebach, Synthesis 1976, 548 - 550.
Reductive Denitrosation of Nitrosamines to Secondary Amines with
Hydrogen/Raney Nickel.
19) D. Enders, H. Eichenauer, Angew. Chem. 1976, 88, 579 - 580; Angew. Chem. Int.
Ed. Engl. 1976, 15, 549 - 550. Asymmetrische Synthese von α-substituierten
Ketonen durch Metallierung und Alkylierung chiraler Hydrazone.
20) D. Enders, H. Eichenauer, Tetrahedron Lett. 1977, 191 - 194. Enantioselective
Alkylation of Aldehydes via Metalated Chiral Hydrazones.
3
21) D. Seebach, D. Enders, B. Renger, Chem. Ber. 1977, 110, 1852 - 1865. Lithiierung
und elektrophile Substitution an α-Methylengruppen von Nitrosaminen.
Umpolung der Reaktivität sekundärer Amine.
22) D. Seebach, D. Enders, R. Dach, R. Pieter, Chem. Ber. 1977, 110, 1879 - 1886.
Reaktion metallierter Nitrosamine mit Nitrilen. Eine neue Methode zur
Darstellung von v-Triazolen.
23) D. Enders, R. Pieter, Chemie für Labor und Betrieb 1977, 28, 503 - 504. Routine-
Dünnschichtchromatographie - ganz einfach.
24) E. Friedrich, W. Lutz, H. Eichenauer, D. Enders, Synthesis 1977, 893 - 894. Mild
Cleavage of N,N-Dimethylhydrazones with Singlet Oxygen.
25) E. J. Corey, D. Enders, Chem. Ber. 1978, 111, 1337 - 1361. Herstellung und
synthetische Verwendung von metallierten Dimethylhydrazonen. Regio- und
stereoselektive Alkylierung von Carbonylverbindungen.
26) E. J. Corey, D. Enders, Chem. Ber. 1978, 111, 1362 - 1383. Synthesewege zu poly-
funktionellen Molekülen über metallierte Dimethylhydrazone.
27) H. Eichenauer, E. Friedrich, W. Lutz, D. Enders, Angew. Chem. 1978, 90, 219 -
220; Angew. Chem. Int. Ed. Engl. 1978, 17, 206 - 207. Regiospezifische und
enantioselektive Aldol-Reaktionen.
28) D. Enders, P. Weuster, Tetrahedron Lett. 1978, 2853 - 2856. Regiospezifische Acy-
lierung von Ketonen zu 1,3-Diketonen über metallierte Dimethylhydrazone.
29) D. Seebach, R. Dach, D. Enders, B. Renger, M. Jansen, G. Brachtel, Helv. Chim.
Acta 1978, 61, 1622 - 1647. 1,4,5,6-Tetrahydro-v-tetrazin-Derivate.
30) H. Ahlbrecht, E. O. Düber, D. Enders, H. Eichenauer, P. Weuster, Tetrahedron
Lett. 1978, 3691 - 3694. NMR-spektroskopische Untersuchungen an
deprotonierten Iminen und Hydrazonen.
31) D. Enders, R. Pieter, B. Renger, D. Seebach, Org. Synth. 1978, 58, 113 - 121.
Nucleophilic α-secondary Aminoalkylation: 2-(Diphenyl-hydroxy-methyl)-
pyrrolidine.
32) D. Enders, H. Eichenauer, Angew. Chem. 1979, 91, 425 - 427; Angew. Chem. Int.
Ed. Engl. 1979, 18, 397 - 398. Asymmetrische Synthese von Ameisen-Alarm-
pheromonen. Alkylierung von acyclischen Ketonen mit praktisch vollständiger
asymmetrischer Induktion.
4
33) D. Enders, Habilitationsschrift, Universität Gießen, 1979. Enantioselektive C-C-
Verknüpfungen über metallierte chirale Hydrazone.
34) P. Rademacher, H.-U. Pfeffer, D. Enders, H. Eichenauer, P. Weuster, J. Chem.
Res. (S) 1979, 222 - 223; J. Chem. Res. (M) 1979, 2501 - 2536.
Photoelektronenspektren und Konformationsverhalten von Hydrazonen.
35) D. Enders, H. Eichenauer, Chem. Ber. 1979, 112, 2933 - 2960. Asymmetrische Syn-
thesen via metallierte chirale Hydrazone. Enantioselektive Alkyierung von
cyclischen Ketonen und Aldehyden.
36) K. G. Davenport, H. Eichenauer, D. Enders, M. Newcomb, D.E. Bergbreiter, J.
Am. Chem. Soc. 1979, 101, 5654 - 5659. Stereoselective Formation and
Electrophilic Substitution of Aldehyde Hydrazone Lithio Anions.
37) D. Enders, H. Eichenauer, R. Pieter, Chem. Ber. 1979, 112, 3703 - 3714. Enantio-
selektive Synthese von (–)-(R)- und (+)-(S)-[6]-Gingerol. Gewürzprinzip des
Ingwers.
38) H. Ahlbrecht, G. Bonnet, D. Enders, G. Zimmermann, Tetrahedron Lett. 1980, 21,
3175 - 3178. Chiral Homoenolate Equivalents I. Asymmetric Synthesis of β-Sub-
stituted Aldehydes via Metalated Chiral Allylamines.
39) D. Enders, in 30 Jahre Fonds der Chemischen Industrie 1950 - 1980, Verband der
Chemischen Industrie, 1980, S. 83 - 90. Neue Methoden zur enantioselektiven C-
C-Verknüpfung.
40) D. Enders, H. Lotter, Angew. Chem. 1981, 93, 831 - 832; Angew. Chem. Int. Ed.
Engl. 1981, 20, 795 - 796. Synthese von enantiomerenreinen (R)- und (S)-α-
Hydroxyketonen und vicinalen Diolen; asymmetrische nucleophile
Carbamoylierung.
41) D. Enders, Chemtech. 1981, 11, 504 - 513. Asymmetric C-C-Bond Formation.
42) D. Enders, H. Lotter, Tetrahedron Lett. 1982, 23, 639 - 642. C-C-Connective
Synthesis of α-Dialkylamino-ketones from Aldehydes and Secondary Amines.
43) D. Enders, in Current Trends in Organic Synthesis, H. Nozaki (Ed.), Pergamon
Press, Oxford, 1983, 151 - 168. Regio-, Diastereo-, and Enantioselective C-C-
Coupling Reactions Using Metalated Hydrazones, Formamides, Allylamines and
Aminonitriles.
5
44) D. Enders, in Perspectives in Organic Synthesis, H. Nozaki (Ed.), Kagaku - Zokan
(Kyoto) 1983, 99, 95 - 100. Regioselective Alkylations of Carbonyl Compounds via
Mono- and Polymetalated Dimethylhydrazones.
45) D. Enders, U. Baus, Liebigs Ann. Chem. 1983, 1439 - 1445. Asymmetrische
Synthese beider Enantiomere von (E)-4,6-Dimethyl-6-octen-3-on - Abwehrsubstanz
der Weberknechte Leiobunum vittatum und L. calcar (Opiliones).
46) D. Enders, K. Papadopoulos, Tetrahedron Lett. 1983, 24, 4967 - 4970. Asymmetric
Synthesis of β-Substituted δ-Ketoesters via Michael-Additions of SAMP-/RAMP-
Hydrazones to α / β-Unsaturated Esters. Virtually Complete 1.6-Asymmetric
Induction.
47) D. Enders, W. Dahmen, E. Dederichs, P. Weuster, Synth. Commun. 1983, 3, 1235 -
1242. Spiroacetals from Acetone and Oxiranes. A Simple Route to Optically Active
1,6-Dioxyspiro[4.4]nonane-Pheromones.
48) D. Enders, in Selectivity - a Goal for Synthetic Efficiency, W. Bartmann, B. M.
Trost (Eds.), Verlag Chemie, Weinheim 1984, S. 65 - 86. Asymmetric Synthesis of
Carbonyl Compounds and Primary Amines.
49) D. Enders, H. Eichenauer, U. Baus, H. Schubert, K. A. M. Kremer, Tetrahedron
1984, 40, 1345 - 1359. Asymmetric Synthesis via Metalated Hydrazones. Overall
Enantioselective α-Alkylation of Acyclic Ketones.
50) D. Enders, in Asymmetric Synthesis Vol. 3, J.D. Morrison (Ed.), Academic Press,
Orlando, 1984, P. 275 - 339. Alkylation of Chiral Hydrazones.
51) D. Enders, H. Schubert, Angew. Chem. 1984, 96, 368 - 369; Angew. Chem. Int. Ed.
Engl. 1984, 23, 365 - 366. Enantioselektive Synthese von β-substituierten
primären Aminen-Alkylierung / reduktive Aminierung von Aldehyden via SAMP-
Hydrazone.
52) D. Enders, W. Mies, J.C.S. Chem. Commun. 1984, 1221 - 1223. (S)-(−)-1-Amino-2-
(siloxymethyl)pyrrolidines: Novel and Efficient Reagents for Chromatographic
Resolution of α-Substituted Aldehydes.
53) D. Enders, H. Lotter, N. Maigrot, J.-P. Mazaleyrat, Z. Welvart, Nouv. J. Chim.
1984, 8, 747 - 750. Asymmetric Nucleophilic Acylation via Metalated Chiral
Aminonitriles. Enantioselective Synthesis of α-Hydroxyketones.
6
54) D. Enders, P. Fey, H. Kipphardt, Org. Prep. Proc. Int. 1985, 17, 1 - 9. Efficient
Preparation of the Chiral Auxiliaries SAMP and RAMP. N-Amination via
Hofmann Degradation.
55) R. Kober, K. Papadopoulos, W. Miltz, D. Enders and W. Steglich; H. Reuter, H.
Puff, Tetrahedron 1985, 41, 1693 - 1701. Synthesis of Diastereo- and
Enantiomerically Pure α-Amino-γ-oxo Acid Esters by Reaction of
Acyliminoacetates with Enamines Derived from 6-Membered Ketones.
56) D. Enders, S. Brauer-Scheib, P. Fey, Synthesis 1985, 393 - 396. A Simple and Effi-
cient Synthesis of Lactone-N,N-dialkyl-hydrazones and their Isomeric N-Dialkyl-
amino-lactams.
57) D. Enders, Chem. Scripta 1985, 25, 139 - 147. Recent Developments in
Asymmetric Synthesis via Metalated Chiral Hydrazones.
58) D. Enders, H. Kipphardt, Nachr. Chem. Tech. Lab. 1985, 33, 882 - 888. (S)-2-
Methoxymethyl-pyrrolidin - ein chirales Auxiliar.
59) H. Kipphardt und D. Enders, Kontakte (Darmstadt) 1985 (2), 37 - 45. 8-
Phenylmenthol als chirales Hilfsreagenz in der Asymmetrischen Synthese.
60) D. Enders, R. W. Hoffmann, Chemie in unserer Zeit 1985, 19, 177 - 190.
Asymmetrische Synthese.
61) D. Enders, B. E. M. Rendenbach, Tetrahedron 1986, 42, 2235 - 2242. Asymmetric
Michael Additions via SAMP-/RAMP-Hydrazones. Enantioselective Synthesis of
Pheromones of the Small Forest Ant (Formica Polyctena) and the Red Wood Ant
(F. Rufa).
62) D. Enders, K. Papadopoulos, B. E. M. Rendenbach; R. Appel and F. Knoch,
Tetrahedron Lett. 1986, 27, 3491 - 3494. Asymmetric Michael Additions via SAMP-
/ RAMP-Hydrazones. Anti-Diastereo- and Enantioselective Synthesis of 3,4-Disub-
stituted 5-oxo-alkanoates.
63) D. Enders, H. Schubert, C. Nübling, Angew. Chem. 1986, 98, 1118 -1119; Angew.
Chem. Int. Ed. Engl. 1986, 25, 1109 - 1110. Enantioselektive Synthese von α-
substituierten primären Aminen durch nucleophile Addition an Aldehyd-SAMP-
Hydrazone.
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64) D. Enders, B. E. M. Rendenbach, in Pesticide Science and Biotechnology (R.
Greengalph, T.R. Roberts, Eds.), Blackwell Scientific Publ., Oxford 1987, S. 17 -
24. Enantioselective Synthesis of Bioregulators.
65) D. Enders, B. Bhushan Lohray, Angew. Chem. 1987, 99, 359 - 360; Angew.
Chem. Int. Ed. Engl. 1987, 26, 351 - 352. Enantioselektive Synthese von α-
Trialkylsilylketonen und –aldehyden.
66) D. Enders, P. Fey, H. Kipphardt, Org. Synth. 1987, 65, 173 - 182. (S)-(-)-1-
Amino2-methoxymethylpyrrolidine (SAMP) and (R)-(+)-1- Amino-2-
methoxymethylpyrrolidine (RAMP). Versatile Chiral Auxiliaries.
67) D. Enders, H. Kipphardt, P. Fey, Org. Synth. 1987, 65, 183 - 202. Asymmetric
Synthesis Using the SAMP-/RAMP-Hydrazone Method. (S)-(+)-4-Methyl-3-
heptanone.
68) D. Enders, B. E. M. Rendenbach, Chem. Ber. 1987, 120, 1223 - 1227.
Asymmetric Michael Additions via SAMP-/RAMP-Hydrazones. Enantioselective
Synthesis of β-Substituted δ-Oxopentanoates and δ-Lactones.
69) D. Enders, A. S. Demir, B. E. M. Rendenbach, Chem. Ber. 1987, 120, 1731 -
1735. Asymmetric Michael Additions via SAMP-/RAMP-Hydrazones.
Enantioselective 1.4-Additions of Methylketones to Knoevenagel Acceptors.
70) D. Enders, A. S. Demir, H. Puff, S. Franken, Tetrahedron Lett. 1987, 28, 3795 -
3798. Asymmetric Michael Addition/Lactamization via SAMP-/RAMP-
Hydrazones. Enantioselective Synthesis of Substituted Tetrahydro-quinoline-
2,5-diones.
71) D. Enders, V. Bhushan, Z. Naturforsch. 1987, 42B, 1595 - 1596. Mild and Effi-
cient Oxidative Cleavage of N,N-Dialkylhydrazones to Ketones with Sodium
Perborate.
72) D. Enders, B. B. Lohray, Angew. Chem. 1988, 100, 594 - 596; Angew. Chem. Int.
Ed. Engl. 1988, 27, 581 - 583. Diastereo und enantioselektive Aldol-Reaktionen
via α-Silylketone. Asymmetrische Synthese von Sitophilur, Aggregations-
Pheromon des Reis- und Maiskäfers.
73) W.-Y. Zhang, D. J. Jakiela, A. Maul, C. Knors, J.W. Lauher, P. Helquist, D.
Enders, J. Am. Chem. Soc. 1988, 110, 4652 - 4660. Highly Diastereofacial
Selective Chelation of α-Phosphite-Containing α,β-Unsaturated Ketone System
to the Fe(CO)2 Group.
8
74) D. Enders, V. Bhushan, Tetrahedron Lett. 1988, 29, 2437 - 2440.
Enantioselective Synthesis of Protected α-Hydroxy Aldehydes and Ketones via
Hydroxylation of Metalated Chiral Hydrazones.
75) D. Enders, H. Kipphardt, P. Gerdes, L. J. Breña-Valle, V. Bhushan, Bull. Soc.
Chim. Belg. 1988, 97, 691 - 704. Large Scale Preparation of Versatile Chiral
Auxiliaries Derived from (S)-Proline.
76) D. Enders, G. Bachstädter, K. A. M. Kremer, M. Marsch, K. Harms, G. Boche,
Angew. Chem. 1988, 100, 1580 - 1581; Angew. Chem. Int. Ed. Engl. 1988, 27,
1522 - 1524. Struktur eines chiralen Lithium-ezaenolats: monomeres,
intramolekular chelatisiertes Lithio-2-acetylnaphthalin-SAMP-hydrazon.
77) D. Enders, S. Müller, A. S. Demir, Tetrahedron Lett. 1988, 29, 6437 - 6440.
Enantioselective Hantzsch Dihydropyridine Synthesis via Metalated Chiral
Alkyl Acetoacetate Hydrazones.
78) A. S. Demir, D. Enders, Tetrahedron Lett. 1989, 30, 1705 - 1708. Regioselective
Alkylation of Dianions of Cyclic 1.3-Diketones via their Monodimethyl-
Hydrazones. Synthesis of C-4 Substituted Cyclic 1.3-Diketones.
79) A. S. Demir, D. Enders, Z. Naturforsch. 1989, 44B, 834 - 838. Synthesis of
Bicyclic and Tricyclic Enones via Regioselective Dialkylation of Cyclic 1,3-
Diketonedimethylhydrazones with 4-Chlorobutane -2-one.
80) D. Enders, B. Bockstiegel, Synthesis 1989, 493 - 496. Enantioselective
Alkylation of 2,2-Dimethyl-1,3-dioxan-5-one Using the SAMP-/RAMP-
Hydrazone Method.
81) B. B. Lohray, D. Enders, Helv. Chim. Acta 1989, 72, 980 - 984. Silicon- Directed
Regio- and Enantioselective Synthesis of α-Hydroxy-Ketones.
82) H. Ahlbrecht, D. Enders, L. Santowski, G. Zimmermann, Chem. Ber. 1989, 122,
1995 - 2004. Chirale Homoenolat-Äquivalente II. Asymmetrische Synthese 3-
substituierter Phenylpropionaldehyde über metallierte chirale Cinnamylamine.
83) D. Enders, P. Gerdes, H. Kipphardt, Angew. Chem. 1990, 102, 226 - 228; Angew.
Chem. Int. Ed. Engl. 1990, 29, 179 - 181. Asymmetrische nucleophile Acylierung
via metallierte chirale Aminocyanide; enantioselektive Synthese von 3-
substituierten 4-Oxoestern durch asymmetrische Michael-Addition.
9
84) W. Keim, A. Köhnes, T. Röthel, D. Enders, J. Organomet. Chem. 1990, 382, 295 -
301. Enantioselective Telomerization I. Telomerization of Butadiene with Form-
aldehyde, β-Dicarbonyl-Compounds, Nitroalkanes and Enamines.
85) D. Enders, W. Gatzweiler, E. Dederichs, Tetrahedron 1990, 46, 4757 - 4792. Dia-
stereo- and Enantioselective Synthesis of α,α'-Disubstituted Spiroacetals Using
the SAMP-/RAMP-Hydrazone Method.
86) D. Enders, H. Dyker, Liebigs Ann. Chem. 1990, 1107 - 1110. Synthesis and Proper-
ties of the Two Artificial Fragrances Lilial and Methylundecanal.
87) D. Enders, W. Dahmen, E. Dederichs, W. Gatzweiler, P. Weuster, Synthesis 1990,
1013 - 1019. Synthesis of Spiroacetal Pheromones via Metalated Hydrazones.
88) D. Enders, S. Nakai, Helv. Chim. Acta 1990, 73, 1833 - 1836. Regio-, Diastereo -
and Enantioselective Synthesis of Vicinal Diols via α-Silyl-ketones.
89) D. Enders, A. Plant, Synlett 1990, 725 - 726. Oxidative Cleavage of N,N-Dialkyl-
hydrazones to Ketones with Magnesium Monoperoxyphthalate.
90) D. Enders, T. Schmitz, G. Raabe, C. Krüger, Acta Crist. 1991, C47, 37 - 40. Struc-
ture of (+)-(3S,4R,5R,1'R,2'S,5'R)-Tetracarbonyl-{(3,4-η2)-5-[5'-methyl-2'-(1-
methylethyl)cyclohexyloxy]-2(5H)-furanone}-iron.
91) D. Enders, S. Nakai, Chem. Ber. 1991, 124, 219 - 226. Regio-, Diastereo- and
Enantioselective Synthesis of Vicinal-Diols via α-Silyl-ketones According to the
SAMP-/RAMP-Hydrazone Method.
92) G. Raabe, E. Zobel, J. Fleischhauer, P. Gerdes, D. Mannes, E. Müller, D. Enders,
Z. Naturforsch. 1991, 46a, 275 - 288. The Structure of Lithiated Aminonitriles in
Solution: Interpretation of their Experimental IR Spectra by Means of Ab Initio
Calculations.
93) D. Enders, D. Bartzen, Liebigs Ann. Chem. 1991, 569 - 574. Enantioselective Total
Synthesis of Harmonine, a Defence Alkaloid of Ladybugs (Coleoptera:
Coccinellidae).
94) L. Duhamel, P. Duhamel, D. Enders, W. Karl, F. Leger, J. M. Poirier, G. Raabe,
Synthesis 1991, 649 - 654. β-Lithiated Enamines as Enolate Equivalents in
Michael-Additions to Enoates. A Novel Entry to Mono- and Disubstituted 5-Oxo-
esters.
10
95) D. Enders, W. Gatzweiler, U. Jegelka, Synthesis 1991, 1137 - 1141. Diastereo- and
Enantioselective Synthesis of α,α'-Disubstituted C2-Symmetric Ketones Using the
SAMP-/RAMP-Hydrazone Method.
96) D. Enders, A. Plant, Liebigs Ann. Chem. 1991, 1241 - 1243. Enantioselective Syn-
thesis of (S)-(+)-2-Tridecanol Acetate, an Aggregation Pheromone Component of
Drosophila mulleri.
97) D. Enders, H. J. Scherer, G. Raabe, Angew. Chem. 1991, 103, 1676 - 1678; Angew.
Chem. Int. Ed. Engl. 1991, 30, 1664 - 1666. Diastereo- und enantioselektive, durch
Michael-Addition initiierte Cyclisierungen in trans-substituierten Cyclopentan-
carbonsäureestern.
98) D. Enders, V. N. Pathak, P. Weuster, Chem. Ber. 1992, 125, 515 - 524.
Regioselective Acylations of Ketones to 1,3-Diketones via Metalated
Dimethylhydrazones.
99) D. Enders, H. Dyker, G. Raabe, Angew. Chem. 1992, 104, 649 - 651; Angew. Chem.
Int. Ed. Engl. 1992, 31, 618 - 620. Enantioselektive Synthese 3-substituierter 2-
Ketoester.
100) G. Raabe, W. Karl, D. Enders, J. Fleischhauer, Z. Naturforsch. 1992, 47a, 869 -
876. Conformational Aspects of Substituents in Enamines. X-Ray Structure
Analyses and Quantum Chemical Calculations.
101) D. Enders, D. Mannes, G. Raabe, Synlett 1992, 837 - 839. Asymmetric Nucleophilic
Acylation with Metalated Chiral Amino Nitriles: Enantioselective Synthesis of 1,4-
Diketones via Asymmetric Michael-Addition.
102) D. Enders, O. Meyer, G. Raabe, Synthesis 1992, 1242 - 1244. Diastereo- and
Enantioselective Synthesis of 4-Nitro-Cyclohexanones by [4+2] Cycloaddition of a
Chiral 2-Amino-butadiene to Nitroalkenes.
103) D. Enders, W. Karl, Synlett 1992, 895 - 897. ß-Lithiated Enamines as Enolate
Equivalents in Asymmetric Michael Additions to Enoates. Highly Enantioselective
Synthesis of Mono-and Disubstituted 5-Oxo-Esters.
104) D. Enders, A. Zamponi, G. Raabe, Synlett 1992, 897 - 900. Enantioselective Syn-
thesis of 3-Oxoesters and Carboxylic Acids as Polyfunctional Small Building
Blocks with a Quaternary Stereogenic Center.
11
105) D. Enders, H. Dyker, G. Raabe, J. Runsink, Synlett 1992, 901 - 903. Enantio- and
Diastereoselective Synthesis of 3-Substituted Cyclic Hemiketals of ω-Hydroxy-2-
oxo Esters.
106) D. Enders, U. Jegelka, Synlett 1992, 999 - 1002. Flexible and Stereocontrolled Syn-
thesis of Azasugars with Novel Substitution Patterns.
107) D. Enders, R. Funk, M. Klatt, G. Raabe, E. R. Hovestreydt, Angew. Chem. 1993,
105, 418 - 420; Angew. Chem. Int. Ed. Engl. 1993, 32, 418 - 421. Enantioselektive
Synthese von α-Aminoacetalen und α-Aminosäuren durch nucleophile 1,2-
Addition an Diethoxyacetaldehyd-SAMP-Hydrazon.
108) D. Enders, J. Schankat, Helv. Chim. Acta 1993, 76, 402 - 406. Enantioselektive
Synthese von Allyl- und Propargylaminen durch nucleophile 1,2-Addition an
chirale Aldehydimine.
109) D. Enders, H. Dyker, G. Raabe, Angew. Chem. 1993, 105, 420 - 423; Angew. Chem.
Int. Ed. Engl. 1993, 32, 421 - 423. Enantioselektive Aldolreaktionen mit einem
Phosphoenolpyruvat-Äquivalent. Asymmetrische Synthese von 4-Hydroxy-2-oxo-
carbonsäureestern.
110) D. Enders. U. Jegelka, B. Dücker, Angew. Chem. 1993, 105, 423 - 425; Angew.
Chem. Int. Ed. Engl. 1993, 32, 423 - 425. Diastereo-und enantioselektive Synthese
C2-symmetrischer HIV-1-Protease-Inhibitoren.
111) D. Enders, B. Bockstiegel, H. Dyker, U. Jegelka, H. Kipphardt, D. Kownatka, H.
Kuhlmann, D. Mannes, J. Tiebes, K. Papadopoulos in "Wege zu neuen Verfahren
und Produkten der Biotechnologie", DECHEMA-Monographie 1993, 129, 209 - 222.
112) D. Enders, J. Tiebes, Liebigs Ann. Chem. 1993, 173 - 177. A New Asymmetric Syn-
thesis of Both Enantiomers of Coniine by 1,2-Addition of RLi/YbCl3 to Aldehyde
SAMP-Hydrazones.
113) D. Enders, K. Papadopoulos, E. Herdtweck, Tetrahedron 1993, 49, 1821 - 1830.
Asymmetric Michael Additions via SAMP-/RAMP-Hydrazones. Enantioselective
Synthesis of 2-Substituted 4-Oxosulfones.
114) D. Enders, K.-J. Heider, G. Raabe, Angew. Chem. 1993, 105, 592 - 594; Angew.
Chem. Int. Ed. Engl. 1993, 32, 598 - 601. Diastereo- und enantioselektive Synthese
von 2-substituierten 3-Trialkylzinncyclohexanonen durch Michael-Addition von
Trialkylzinnlithium an Cyclohexenon-SAMP-Hydrazon.
12
115) D. Enders, S. Osborne, J. Chem. Soc. Chem. Commun. 1993, 424 - 426. Determina-
tion of the Relative and Absolute Configuration of Stigmatellin A by Chemical Cor-
relation.
116) D. Enders, M. Klatt, R. Funk, Synlett 1993, 226 - 228. Enantioselective Synthesis
of Protected ß-Amino Acetals and ß-Amino Acids by 1,2-Addition of RM/CeCl3 to
3,3-Ethylenedioxypropanal-SAMP-Hydrazone.
117) D. Enders, A. Zamponi, G. Raabe, J. Runsink, Synthesis 1993, 725 - 728.
Enantioselective Synthesis of 2-Alkyl-2-cyanocycloalkanones with a Quaternary
Stereogenic Center.
118) D. Enders, U. Jegelka, Tetrahedron Lett. 1993, 34, 2453 - 2456. 1,3-Dioxan-5-one
as C3-Building Block for the Diastereo-and Enantioselective Synthesis of C5-to-C9-
De-oxy Sugars Using the SAMP-/ RAMP-Hydrazone Method.
119) D. Enders, M. Finkam, Liebigs Ann. Chem. 1993, 551 - 555. First Synthesis of the
Cytotoxic and Antifungal C14-Amine (2S,3E,5Z)-2-Amino-3,5,13-tetradecatriene
Isolated from the New Zealand Ascidian Pseudodistoma novaezelandiae.
120) D. Enders, M. Finkam, Synlett 1993, 401 - 403. Iron Mediated Synthesis of 4-
Amino Enoates of High Enantiomeric Purity.
121) D. Enders, B. B. Lohray, Synthesis 1993, 1092 - 1094. Enantioselective Siloxybuty-
lation of Aldehydes and Ketones by Lewis Acid Mediated Ring Opening of Tetrahy-
drofuran with Lithiated Hydrazones.
122) D. Enders, H. J. Scherer, J. Runsink, Chem. Ber. 1993, 126, 1929 - 1944.
Diastereo- und enantioselektive Synthese 1,2-trans-substituierter Cycloalkan-
carbonsäureester und Sulfone durch Michael-initiierte Cyclisierungen via SAMP-
/RAMP-Hydrazone.
123) D. Enders, J. Tiebes, N. De Kimpe, M. Keppens, C. Stevens, G. Smagghe, O. Betz,
J. Org. Chem. 1993, 58, 4881 - 4884. Enantioselective Synthesis and
Determination of the Configuration of Stenusine, the Spreading Agent of Beetle
Stenus comma.
124) V. Bhushan, B. B. Lohray, D. Enders, Tetrahedron Lett. 1993, 34, 5067 - 5070.
Efficient Enantioselective Synthesis of Allylsilanes by Wittig Olefination of α-
Silylaldehydes.
13
125) D. Enders in Stereoselective Synthesis, E. Ottow, K. Schöllkopf, B.- G. Schulz (Eds),
Springer-Verlag, Berlin, S. 63 - 90, 1994. Enzymemimetic C-C-and C-N Bond For-
mations.
126) D. Enders, O. Meyer, G. Raabe, J. Runsink, Synthesis 1994, 66 - 72. (S,S)-3,5-Di-
methylmorpholine, a Novel C2-Symmetric Auxiliary. First Appplication in [4+2]-
Cycloadditions Leading to 4-Oxohexahydropyridazine Derivatives.
127) D. Enders, T. Schäfer, O. Piva, A. Zamponi, Tetrahedron 1994, 50, 3349 - 3362.
Enantioselective Synthesis of 2-Sulfenylated Aldehydes: Alkylation of Sulfenylated
Acetaldehyde SAMP-Hydrazones.
128) D. Enders, A. Zamponi, T. Schäfer, C. Nübling, H. Eichenauer, A. S. Demir, G.
Raabe, Chem. Ber. 1994, 127, 1707 - 1721. Enantioselective Synthesis of
Polyfunctional Small Building Blocks with a Quaternary Stereogenic Center.
129) D. Enders, B. Jandeleit, G. Raabe, Angew. Chem. 1994, 106, 2033 -2035; Angew.
Chem. Int. Ed. Engl. 1994, 33, 1949 - 1951. Eisenunterstützte, regio-und
stereoselektive allylische Substitutionen zu 3-substituierten Alkenylsulfonen.
130) D. Enders, D. Backhaus, J. Runsink, Angew. Chem. 1994, 106, 2167 -2170; Angew.
Chem. Int. Ed. Engl. 1994, 33, 2098 - 2100. [2,3]-Sigmatrope Wittig-Umlagerung
chiraler Allyloxyacetaldehyd-Hydrazone zur diastereo-und enantioselektiven Syn-
these von geschützten γ, δ-ungesättigten α-Hydroxyaldehyden und Cyanhydrinen.
131) D. Enders, U. Reinhold, Synlett 1994, 792 - 794. Enantioselective Synthesis of
Protected α-Hydroxy Aldehydes via Alkylation of Metalated Chiral Hydrazones.
132) D. Enders, J. Schankat, M. Klatt, Synlett 1994, 795 - 797. Enantioselective
Synthesis of Homoallylamines and β-Amino Acids via Nucleophilic Allylation of
SAMP/RAMP-Hydrazones.
133) D. Enders, W. Bettray in Proceedings of the Chiral Europe '94 Symposium, 1994,
S. 51 - 60. Recent Advances in the Development of Highly Enantioselective
Synthetic Methods.
134) D. Enders, H. Kempen, Synlett 1994, 969 - 971. Enantioselective Synthesis of
Allylic Alcohols via Asymmetric [2,3]-Sigmatropic Meisenheimer Rearrangement.
135) D. Enders, W. Bettray, G. Raabe, J. Runsink, Synthesis 1994, 1322 - 1326.
Diastereo- and Enantioselective Synthesis of α-Substituted β-Amino Acid Esters
14
by Tandem Michael Addition / α-Alkylation with TMS-SAMP as Chiral Equivalent
of Ammonia.
136) D. Enders, A. Plant, Synlett 1994, 1054 - 1056. Enantioselective Synthesis of α-
Substituted Nitriles by Oxidative Cleavage of Aldehyde SAMP-Hydrazones with
Magnesium Monoperoxyphthalate.
137) D. Enders, B. Jandeleit, Synthesis 1994, 1327 - 1330. Iron-Mediated Complete
Chirality Transfer in Allylic Substitutions. Efficient Synthesis of (−)-(S)-
Myoporone.
138) D. Enders, H. Wahl, W. Bettray, Angew. Chem. 1995, 107, 527 - 529; Angew.
Chem. Int. Ed. Engl. 1995, 34, 455 - 457. Enantioselektive Synthese von β-
Aminosäuren – TMS-SAMP als chirales Ammoniak-Äquivalent in der azaanalogen
Michael-Addition an α,β-ungesättigte Ester.
139) D. Enders, J. Schankat, Helv. Chim. Acta 1995, 78, 970 - 992. Enantioselektive
Synthese von Allyl-, Propargyl- und 1,3-Enin-aminen durch 1,2-Addition von
Organocer-Reagenzien an chirale Aldimine.
140) D. Enders, K. Breuer, G. Raabe, J. Runsink, J. H. Teles, J.-P. Melder, S. Brode,
Angew. Chem. 1995, 107, 1119 - 1112. Angew. Chem. Int. Ed. Engl. 1995, 34, 1021
- 1023. Zur Darstellung, Struktur und Reaktivität von 1,3,4-Triphenyl-4,5-
dihydro-1H-1,2,4-triazol-5-yliden, einem neuen stabilen Carben.
141) D. Enders, Acros Organics Acta 1995, 1, 35 - 36. SADP and SAEP. Novel Chiral
Hydrazine Auxiliaries for Asymmetric Synthesis.
142) D. Enders, Acros Organics Acta 1995, 1, 37 - 38. TMS-SAMP. Novel Chiral Hydra-
zine Auxiliary for Hetero-Michael Additions and Aza-Peterson Olefinations.
143) D. Enders, J. Kirchhoff, D. Mannes, G. Raabe, Synthesis 1995, 659 - 666. Asym-
metric Nucleophilic Acylation with Metalated Aminonitriles: Diastereo- and
Enantioselective Synthesis of 2-Substituted 3-Aroyl-cyclohexanones via Tandem
Michael Addition / α-Alkylation.
144) D. Enders, J. Wiedemann, W. Bettray, Synlett 1995, 369 - 371. Diastereo- and
Enantioselective Synthesis of Trans-2-Amino-cycloalkane-1-carboxylic Acids via
Intramolecular Tandem Michael Addition/ α-Alkylation Using TMS-/SAMP as
Chiral Equivalent of Ammonia.
15
145) D. Enders, B. Jandeleit, Liebigs Ann. Chem. 1995, 1173 - 1176. Efficient and
Convergent Synthesis of (R)-(−)-10-Methyl-tridecane-2-one, the Sex Pheromone of
the Spotted Cucumber Beetle, by Iron-Mediated Chirality Transfer.
146) D. Enders, U. Reinhold, Angew. Chem. 1995, 107, 1332 - 1334; Angew. Chem. Int.
Ed. Engl. 1995, 34, 1219 - 1222. Diastereo- und enantioselektive Synthese von
vicinalen Aminoalkoholen aus Glykolaldehyd-Hydrazonen. Asymmetrische
Synthese von (R,R)-Statin.
147) D. Enders, A. Plant, K. Drechsel, O. F. Prokopenko, Liebigs Ann. Chem. 1995,
1127- 1129. A Convenient Enantioselective Synthesis of (R)-(−)-Phoracantholide I,
a Component of the Defence Secretion of the Eucalypt Longicorn Phoracantha
synonyma.
148) D. Enders, B. Jandeleit, O. F. Prokopenko, Tetrahedron 1995, 51, 6273 - 6284.
Convergent Synthesis of (R,R)-6,12-Dimethylpenta-decan-2-one, the Female Sex
Pheromone of the Banded Cucumber Beetle by Iron Mediated Chirality Transfer.
149) D. Enders, H. Wahl, K. Papadopoulos, Liebigs Ann. Chem. 1995, 1177 - 1184.
Asymmetric Michael Additions via SAMP/RAMP-Hydrazones. Enantioselective
Synthesis of 2-Substituted 4-Oxophosphonates.
150) D. Enders, D. Backhaus, Synlett 1995, 631 - 632. Diastereo- and Enantioselective
Synthesis of β-Substituted γ, δ -Unsaturated α-Hydroxy Ketones via [2,3]- Wittig
Rearrangement of α-Allyloxyketone-Hydrazones.
151) D. Enders, M. Klatt in Encyclopedia of Reagents for Organic Synthesis, L. A.
Paquette, Ed., Wiley, New York, 1995, 3368 - 3370. (S)-2-Methoxymethyl-
pyrrolidine.
152) D. Enders, M. Klatt in Encyclopedia of Reagents for Organic Synthesis, L. A.
Paquette, Ed., Wiley, New York, 1995, 178 - 182. (S)-1-Amino-2-methoxymethyl-
pyrrolidine.
153) D. Enders, O. F.Prokopenko, Liebigs Ann. Chem. 1995, 1185 - 1191. Diastereo- and
Enantioselective Synthesis of the 18-Membered Lichen Macrolide (+)-Aspicilin.
154) D. Enders, R. Gröbner, J. Runsink, Synthesis 1995, 947 - 951. Enantioselective
Synthesis of 3-Substituted 6- and 7-Membered Lactones via α-Alkylation of
Lactone Hydrazones.
16
155) D. Enders, M. Knopp, J. Runsink, G. Raabe, Angew. Chem. 1995, 107, 2442 - 2445;
Angew. Chem. Int. Ed. Engl. 1995, 34, 2278 - 2280. Diastereo- und
enantioselektive Synthese von polyfunktionellen Ketonen mit benachbarten
quartären und tertiären Stereozentren durch asymmetrische Carroll-Umlagerung.
156) D. Enders, B. Jandeleit, Acros Organics Acta 1995, 1, 59 - 60. (S,E)-(–)-Methyl-4-
(phenylmethoxy)-2-pentenoate, a Synthetically Useful Enantiopure Building
Block.
157) D. Enders, M. Bartsch, D. Backhaus, Synlett 1995, 869 - 870. Diastereo- and
Enantioselective Synthesis of (–)-Oudemansin A via [2,3]-Wittig Rearrangement of
Crotyloxyacetaldehyde-SAEP-Hydrazone.
158) D. Enders, D. L. Whitehouse, J. Runsink, Chem. Eur. J. 1995, 1, 382 - 388.
Diastereo- and Enantioselective Synthesis of L-threo and D-erythro-Sphingosine.
159) D. Enders, A. Plant, D. Backhaus, U. Reinhold, Tetrahedron 1995, 51, 10699 -
10714. Asymmetric Synthesis of α-Substituted Nitriles and Cyanohydrins by
Oxidative Cleavage of Chiral Aldehyde Hydrazones with Magnesium
Monoperoxyphthalate.
160) D. Enders, S.-H. Han, R. Maaßen, Tetrahedron Lett. 1995, 36, 8007 - 8010. New
Efficient and Flexible Synthesis of Polysubstituted Pyrroles.
161) D. Enders, J. Kirchhoff, Acros Organics Acta 1996, 2, 10 - 11. (S,S)-(+)-2,2-
Dimethyl- 5 - methylamino-4-phenyl-1,3-dioxan. Novel Chiral Auxiliary for
Asymmetric Michael Additions.
162) D. Enders, R. Syrig, G. Raabe, R. Fernández, C. Gasch, J.-M. Lassaletta, J.- M.
Llera, Synthesis 1996, 48 - 52. Formaldehyde SAMP-Hydrazone as a Neutral
Chiral Formyl Anion and Cyanide Equivalent: Asymmetric Michael Additions to
Nitroalkenes.
163) D. Enders, R. Schiffers, Synthesis 1996, 53 - 58. Enantioselective Synthesis of
Differently Protected 1,2-Diamines via α-Alkylation of Dibenzylamino-Acet-
aldehydeSAMP-Hydrazone.
164) D. Enders, A. Kaiser, Synthesis 1996, 209 - 214. A Short Asymmetric Synthesis of
Both Enantiomers of Ramulosin and Its Analogues.
17
165) D. Enders, U. Reinhold, Liebigs Ann. 1996, 11 - 26. Diastereo- and
Enantioselective Synthesis of 1,2-Amino Alcohols and Protected α-Hydroxy
Aldehydes from Glycol Aldehyde Hydrazones.
166) J. H. Teles, J.-P. Melder, K. Ebel, R. Scheider, S. Brode, D. Enders, K. Breuer, G.
Raabe, Helv. Chim. Acta. 1996, 79, 61 - 83. Benzoin Type Condensations of Form-
aldehyde Catalyzed by Stable Carbenes.
167) D. Enders, P. Fey, T. Schmitz, B. B. Lohray, B. Jandeleit, J. Organomet. Chem.
1996, 514, 227 - 232. Regio- and Stereoselective a4-Umpolung Reactions of α,β-
Unsaturated Esters to 1,6-Dicarbonyl Compounds by Addition of Enantiopure
Nucleophiles to Racemic Tetracarbonyl (η3-allyl)iron(1+) Complexes.
168) D. Enders, D. Backhaus, J. Runsink, Tetrahedron 1996, 52, 1503 - 1528.
Asymmetric [2,3]-Sigmatropic Wittig Rearrangement of Chiral α-Allyloxy-
Hydrazones.
169) D. Enders, T. Berg, G. Raabe, J. Runsink, Helv. Chim. Acta 1996, 79, 118 - 122.
Enantioselektive Synthese von α-Phosphinoketonen.
170) D. Enders, S. v. Berg, B. Jandeleit, Synlett, 1996, 18 - 20. Iron Mediated Allylic
Substitutions with Complete Chirality Transfer. Synthesis of Functionalized γ-
Substituted Alkenylsulfones of High Enantiomeric Purity.
171) D. Enders, U. Frank, P. Fey, B. Jandeleit, B. B. Lohray, J. Organomet. Chem.
1996, 519, 147 - 159. Synthesis of Highly Diastereo- and Enantiomerically
Enriched Tetracarbonyl (η3-allyl)iron(1+) Complexes for Allylic Substitutions with
Silyl Enol Ethers and Silyl Ketene Acetals.
172) D. Enders, D. Ward, J. Adam, G. Raabe, Angew. Chem. 1996, 108, 1059 - 1062. An-
gew. Chem. Int. Ed. Engl. 1996, 35, 981 - 984. Effiziente, regio- und
enantioselektive Mannich- Reaktionen.
173) D. Enders, B. B. Lohray, F. Burkamp, V. Bhushan, R. Hett, Liebigs Ann. 1996, 189
- 200. Regio- and Enantioselective Synthesis of α-Silylaldehydes and Ketones via
SAMP-/RAMP-Hydrazones.
174) D. Enders, O. Piva, F. Burkamp, Tetrahedron 1996, 52, 2893 - 2908. Asymmetric
Synthesis of Vicinal Thioether Alcohols by Diastereoselective 1,2-Addition of
Carbon Nucleophiles to Enantiomerically Enriched α-Sulfenylated Aldehydes.
18
175) D. Enders, F. Burkamp, J. Runsink, J. Chem. Soc. Chem. Commun. 1996, 609 -
610. Diastereo- and Enantioselective Synthesis of 6-Hetero-substituted 3,5-
Dihydroxyesters: Novel Precursors of Mevinolin Analogues.
176) D. Enders, D. L. Whitehouse, Synthesis 1996, 621 - 626. Highly Enantioselective
α-Alkenylation of Aldehydes and Ketones.
177) D. Enders, R. Lochtman, G. Raabe, Synlett 1996, 126 - 128. Enantioselective
Synthesis of 1-Ferrocenylalkylamines via 1,2-Addition of Organolithium
Compounds to Ferrocenecarboxaldehyde-SAMP-Hydrazone.
178) G. Raabe, K. Breuer, D. Enders, Z. Naturforsch. 1996, 51a, 95 - 101. The Role of
Conjugate Interaction in Stable Carbenes of the 1,2,4-Triazol-5-ylidene Type and
Their Energy of Dimerisation. An Ab Initio Study.
179) D. Enders, P. Hecker, O. Meyer, Tetrahedron 1996, 52, 2909 - 2924. A Novel
Approach to 2-Amino-1,3-Dienes by Coupling of α-Chloro Enamines and Alkenyl
Lithium Compounds.
180) D. Enders, W. Bettray, Pure Appl. Chem. 1996, 68, 569 - 580. Recent Advances in
the Development of Highly Enantioselective Synthetic Methods.
181) D. Enders, M. Knopp, Tetrahedron 1996, 52, 5805 - 5818. Novel Asymmetric
Syntheses of (–)-Malingolide and (+)-epi-Malingolide.
182) D. Enders, M. Knopp, J. Runsink, G. Raabe, Liebigs Ann. 1996, 1095 - 1116. The
First Asymmetric Carroll Rearrangement. - Diastereo- and Enantioselective Syn-
thesis of Polyfunctional Ketones with Vicinal Quarternary and Tertiary
Stereogenic Centres.
183) D. Enders, R. Gröbner, G. Raabe, J. Runsink, Synthesis 1996, 941 - 948.
Enantioselective Synthesis of 2-Substituted 5-, 6- and 7-Membered Lactams via α-
Alkylation of their Chiral N-Dialkylamino Derivatives.
184) D. Enders, O. Meyer, Liebigs Ann. 1996, 1023 - 1035. Diastereo- and Enantio-
selective Diels-Alder Reactions with 2-Amino-1,3-dienes.
185) D. Enders, J. Zhu, G. Raabe, Angew. Chem. 1996, 108, 1827 - 1829; Angew. Chem.
Int. Ed. Engl. 1996, 35, 1725 - 1728. Asymmetrische Epoxidierung von Enonen mit
Sauerstoff in Gegenwart von Diethylzink und (R,R)-N-Methylpseudoephedrin.
19
186) D. Enders, O. F. Prokopenko, G. Raabe, J. Runsink, Synthesis 1996, 1095 - 1100.
Highly Diastereoselective Boron Mediated anti-Aldol Reactions of 4-Silyl
Substituted 2,2-Dimethyl-1,3-dioxan-5-one. Diastereo- and Enantioselective
Synthesis of Protected Oxopolyols.
187) D. Enders, K. Breuer, J. H. Teles, Helv.Chim. Acta 1996, 79, 1217 - 1221. A Novel
Asymmetric Benzoin Reaction Catalyzed by a Chiral Triazolium Salt.
188) D. Enders, M. Knopp, R. Schiffers, Tetrahedron: Asymmetry 1996, 7, 1847 - 1882.
Asymmetric [3.3]-Sigmatropic Rearrangements in Organic Synthesis.
189) D. Enders, A. Haertwig, G. Raabe, J. Runsink, Angew. Chem. 1996, 108, 2540 -
2542; Angew. Chem. Int. Ed. Engl. 1996, 35, 2388 - 2390. Enantioselektive
Synthese von vicinalen Aminoalkoholen durch Oxa-Michael-Addition von (–)-N-
Formylnorephedrin an Nitroalkene.
190) D. Enders, M. Meiers, Angew. Chem. 1996, 108, 2391 - 2393; Angew. Chem. Int.
Ed. Engl. 1996, 35, 2261 - 2263. Diastereo- und enantioselektive Synthese von C2-
symmetrischen geschützten 1,n-Diaminen aus Dialdehyden.
191) D. Enders, J. Kirchhoff, V. Lausberg, Liebigs Ann. 1996, 1361 - 1366. Diastereo-
and Enantioselective Synthesis of Lignan Building Blocks via Tandem Michael
Addition / Electrophilic Substitution of Lithiated α-Amino Nitriles to 5H-Furan-2-
one.
192) D. Enders, M. Klatt, Synthesis 1996, 1403 - 1418. Asymmetric Synthesis with (S)-
2-Methoxymethylpyrrolidine (SMP) - a Pioneer Auxiliary.
193) D. Enders, T. Berg, Synlett 1996, 796 - 798. Enantioselective Synthesis of 2-
Phosphino Alcohols via Phosphinylation of Metalated Chiral Aldehyde
Hydrazones.
194) D. Enders, R. Maaßen, S.-H. Han, Liebigs Ann. 1996, 1565 - 1574. New Efficient,
Flexible and Regioselective Synthesis of 2,4-Di-and 2,3,4-Tri-Alkylated and
Arylated 1H-Pyrroles.
195) D. Enders, J. Wiedemann, Synthesis 1996, 1443 - 1450. Diastereo- and
Enantioselective Synthesis of Vicinal Diamines via Aza-Michael Addition to
Nitroalkenes.
196) D. Enders, K. Breuer, J. Runsink, J. H. Teles, Helv. Chim. Acta 1996, 79, 1899 -
1902. The First Asymmetric Intramolecular Stetter Reaction.
20
197) D. Enders, M. Bartsch, D. Backhaus, J. Runsink, G. Raabe, Synthesis 1996, 1438 -
1442. Diastereo- and Enantioselective Synthesis of Polyfunctional Cyclic Ketones
with Neighbouring Quarternary and Tertiary Centers via [2,3]-Wittig Rearrange-
ment.
198) D. Enders, K. Breuer, J. Runsink, J. H. Teles, Liebigs Ann. 1996, 2019 - 2028.
Chemical Reactions of the Stable Carbene 1,3,4-Triphenyl-4,5-dihydro-1H-1,2,4-
triazol-5-ylidene.
199) D. Enders, H. Gielen, G. Raabe, J. Runsink, J. H. Teles, Chem. Ber. 1996, 129,
1483 - 1488. Synthesis and Stereochemistry of the First Chiral Imidazolinylidene-
and Triazolinylidene-Palladium(II) Complexes.
200) D. Enders, W. Bettray, J. Schankat, J. Wiedemann in Enantioselective Synthesis of
β-Amino Acids, E. Juaristi, Ed., Wiley-VCH Publishers, New York 1997, 187 - 210.
Diastereo- and Enantioselective Synthesis of β-Amino Acids via SAMP Hydrazones
and Hetero Michael Addition Using TMS-SAMP as a Chiral Equivalent of
Ammonia.
201) D. Enders, E. Chelain, G. Raabe, Bull. Soc. Chim. Fr. 1997, 134, 299 - 306.
Enantioselective Synthesis of 1,2-Diamines via Nucleophilic 1,2-Addition to
Dibenzylamino-acetaldehyde-SAMP-Hydrazone.
202) D. Enders, A. Kaiser, Liebigs Ann. / Recl. 1997, 485 - 493. Asymmetric Synthesis of
(R,S)-Dehydroiridodial, (R,S)-Dehydroiridodiol and Analogues.
203) D. Enders, B. Jandeleit, S. von Berg, J. Organomet. Chem. 1997, 533, 219 - 236.
„Chirality Transfer“ in Iron Mediated Dienylic Substitutions via Highly Enantio-
merically Enriched Planar Chiral 1-Phenylsulfonyl Substituted Tricarbonyl(η5-
pentadienyl)-iron(1+) Complexes.
204) D. Enders, B. Jandeleit, S. von Berg, Synlett 1997, 421 - 431. Synthesis of Highly
Enantioenriched Compounds via Iron Mediated Allylic Substitutions.
205) D. Enders, T. Berg, G. Raabe, J. Runsink, Liebigs. Ann. / Recl. 1997, 345 - 363.
Enantioselective Synthesis of α-Phosphino Ketones and 2-Phosphino Alcohols.
206) D. Enders, B. Jandeleit, S. von Berg, Synthesis of Highly Enantioenriched Com-
pounds via Iron Mediated Allylic Substitutions in Organic Synthesis via Organo-
metallics (OSM 5), G. Helmchen, Ed., Vieweg, Braunschweig, 1997, 279 - 308.
21
207) D. Enders, J. Wiedemann, Liebigs Ann. / Recl. 1997, 699 - 706. Diastereo- and
Enantioselective Synthesis of Carbocyclic and Heterocyclic β-Amino Acids via
Tandem Aza-Michael-Addition / Intramolecular Cyclization.
208) D. Enders, A. S. Demir, J. Prakt. Chem. / Chem. Ztg. 1997, 339, 553 - 563.
Regioselective Alkylations of Cyclic 1,3-Diketones via Their Metalated Dimethyl-
hydrazones.
209) D. Enders, A. Kaiser, Heterocycles 1997, 46, 631 - 635. A Short Asymmetric
Synthesis of (–)-Neonepetalactone.
210) D. Enders, H. Gielen, K. Breuer, Tetrahedron: Asymmetry 1997, 8, 3571 - 3574.
Catalytic Asymmetric Hydrosilylation with (Triazolinylidene)Rhodium Complexes
Containing an Axis of Chirality.
211) D. Enders, D. Kownatka, T. Hundertmark, O. F. Prokopenko, J. Runsink,
Synthesis 1997, 649 - 652. Asymmetric Michael Additions via 2,2-Dimethyl-1,3-
dioxan-5-one SAMP-Hydrazone. Diastereo- and Enantioselective Synthesis of
Protected 3-Substituted 4,6-Dihydroxy-5-oxoesters.
212) D. Enders, C. Nübling, H. Schubert, Liebigs Ann. / Recl. 1997, 1089 - 1100.
Asymmetric Synthesis of Primary Amines by Nucleophilic Addition of Alkyl-
lithium Compounds to Aldehyde SAMP/RAMP Hydrazones.
213) D. Enders, J. Zhu, L. A. Kramps, Liebigs Ann. / Recl. 1997, 1101 - 1113. Zinc-
mediated Asymmetric Epoxidation of α-Enones.
214) D. Enders, K. Breuer, J. H. Teles, K. Ebel, J. Prakt. Chem. / Chem. Ztg. 1997, 339,
397 - 399. 1,3,4-Triphenyl-4,5-dihydro-1H-1,2,4-triazol-5-ylidene - Applications of a
Stable Carbene in Synthesis and Catalysis.
215) D. Enders, D. Bartzen, Liebigs Ann. / Recl. 1997, 1115 - 1123. Diastereo- and
Enantioselective Synthesis of 4,5,6-Trisubstituted and 6-Monosubstituted
Piperidin-2-ones.
216) D. Enders, K. Breuer, G. Raabe, J. Simonet, A. Ghanimi, H. B. Stegmann, J.-H.
Teles, Tetrahedron Lett. 1997, 38, 2833 - 2836. A Stable Carbene as π-Acceptor.
Electrochemical Reduction to the Radical Anion.
217) D. Enders, R. Lochtman, Synlett 1997, 355 - 356. Diastereo- and Enantioselective
Synthesis of 1,1’-Bis(1-Aminoalkyl)ferrocenes via 1,2-Addition of Organolithium
Compounds to Ferrocene-1,1’-dicarbaldehyde-bis-SAMP-hydrazone.
22
218) D. Enders, H. Gielen, G. Raabe, J. Runsink, J. H. Teles, Chem. Ber. / Recl. 1997,
130, 1253 - 1260. Diastereoselectice Synthesis of the First Enantiomerically Pure
(Triazolin-ylidene)-Ruthenium (II) and Rhodium (III) Chelate Complexes.
219) D. Enders, U. Reinhold, Tetrahedron: Asymmetry 1997, 8, 1895 - 1946.
Asymmetric Synthesis of Amines by Nucleophilic 1,2-Addition of Organometallic
Reagents to the CN-Double Bond.
220) D. Enders, H. Wahl, K. Papadopoulos, Tetrahedron 1997, 53, 12961 - 12978.
Diastereo- and Enantioselective Synthesis of 2,3- and 1,2-Disubstituted 4-
Oxophosphonates via Asymmetric Michael Addition.
221) D. Enders, C. Leriverend, Tetrahedron: Asymmetry 1997, 8, 2787 - 2792.
Diastereo- and Enantioselective Synthesis of Protected Vicinal Silylamines via 1,2-
Addition to α-Silyl-Hydrazones.
222) D. Enders, M. Potthoff, G. Raabe, J. Runsink, Angew. Chem. 1997, 109, 2454 -
2456; Angew. Chem. Int. Ed. Engl. 1997, 36, 2362 - 2364. Regio- und
enantioselektive Synthese von α-Fluorketonen via elektrophile Fluorierung von α-
Silylketonenolaten mit N-Fluorbenzolsulfonimid.
223) D. Enders, B. Bockstiegel, W. Gatzweiler, U. Jegelka, B. Dücker, L. Wortmann,
Chimica Oggi 1997, 15, 20 - 22. 2,2-Dimethyl-1,3-dioxan-5-one. A Dihydroxy-
acetone Equivalent for Asymmetric Synthesis.
224) D. Enders, D. Klein, G. Raabe, J. Runsink, Synlett 1997, 1271 - 1272. Asymmetric
Synthesis of α’-Silylated α-Iodo Ketones via Iodination with Trifluoroiodomethane.
225) D. Enders, R. Peters, R. Lochtman, J. Runsink, Synlett 1997, 1462 - 1464.
Enantioselective Synthesis of Planar Chiral ortho-Functionalised
Ferrocenylketones.
226) D. Enders, J. Kirchhoff, P. Gerdes, D. Mannes, G. Raabe, J. Runsink, G. Boche, M.
Marsch, H. Ahlbrecht, H. Sommer, Eur. J. Org. Chem. 1998, 63 - 72. Structure and
Reactivity of Lithiated α-Amino Nitriles.
227) D. Enders, P. Müller, D. Klein, Synlett 1998, 43 - 44. Diastereo- and
Enantioselective Synthesis of syn-2,3-Disubstituted 1,4-Diketones via Oxidative
Coupling of Metalated Hydrazones.
23
228) D. Enders, U. Baus, P. Müller, K. C. Nicolaou, B. Jandeleit, Molecules Online
1998, 2, 15 - 21. Asymmetric Synthesis of 3-Substituted 4-Oxoesters Using the
SAMP-/ RAMP-Hydrazone Method.
229) D. Enders, H. Dyker, F. R. Leusink, Chem. Eur. J. 1998, 4, 311 - 320.
Enantioselective Synthesis of Protected Isotetronic Acids.
230) D. Enders, T. Schäfer, W. Mies, Tetrahedron 1998, 54, 10239 - 10252.
Enantioselective Synthesis of α-Sulfenylated Ketones and Aldehydes via α-
Thiolation of Metalated SAMP/RAMP Hydrazones.
231) D. Enders, M. Bolkenius, J. Vázquez, J.-M. Lassaletta, R. Fernández, J. Prakt.
Chem. /Chem. Ztg. 1998, 340, 281 - 285. Formaldehyde SAMP-Hydrazone - a
Neutral Chiral Formyl Anion and Cyanide Equivalent.
232) D. Enders, R. Lochtman, Eur. J. Org. Chem. 1998, 689 - 696. Asymmetric
Synthesis of (1-Ferrocenylalkyl)amines and 1,1’-Bis(1-aminoalkyl)ferrocene
Derivatives.
233) D. Enders, M. Kroll, G. Raabe, J. Runsink, Angew. Chem. 1998, 110, 1770 - 1773;
Angew. Chem. Int. Ed. 1998, 37, 1673 - 1675. Diastereoselektive Synthese
hochsubstituierter 5-Ring-Sauerstoff-Heterocyclen via Zirconocen-vermittelte C-C-
Kupplungs-Reaktionen.
234) D. Enders, H. Gielen, J. Runsink, K. Breuer, S. Brode, K. Boehn, Eur. J. Inorg.
Chem. 1998, 913 - 919. Diastereoselective Synthesis of Chiral
(Triazolinylidene)Rhodium Complexes Containing an Axis of Chirality.
235) D. Enders, C. Thomas, G. Raabe, J. Runsink, Helv. Chim. Acta 1998, 81, 1329 -
1336. Enantioselektive Synthese von α-substituierten N-Methyl-Sulfonamiden.
236) D. Enders, M. Kroll, G. Raabe, J. Runsink, Molecules Online 1998, 2, 109 - 113.
Zirkonocene Mediated Diastereoselective Synthesis of 4,5,5-Trisubstituted 2-
Alkoxytetrahydrofurans.
237) J. Fleischhauer, A. Koslowski, A. Wollmer, D. Enders, A. Zamponi, G. Raabe, Z.
Naturforsch. 1998, 53a, 891 - 895. CD-Spectroscopic Confirmation of the Absolute
Configuration of a Conformationally Flexible Aldehyde Ester Containing a
Quarternary Stereogenic Center.
24
238) D. Enders, Th. Hundertmark, R. Lazny, Synlett 1998, 721 - 722. Mild,
Racemization Free Cleavage of Ketone SAMP-Hydrazones with Oxalic Acid -
Recycling of the Chiral Auxiliary.
239) D. Enders, A. Haertwig, G. Raabe, J. Runsink, Eur. J. Org. Chem. 1998, 1771 -
1792. Diastereo- and Enantioselective Synthesis of Vicinal Aminoalcohols via Oxa-
Michael-Addition of N-Formylnorephedrine to Nitroalkenes.
240) D. Enders, A. Haertwig, J. Runsink, Eur. J. Org. Chem. 1998, 1793 - 1802.
Diastereo- and Enantioselective Synthesis of N-Protected 2-Amino-1,4-diols via an
Oxa-Michael-Addition / 1,3-Dipolar Cycloaddition Protocol.
241) D. Enders, R. Maaßen, J. Runsink, Tetrahedron: Asymmetry 1998, 9, 2155 - 2180.
First Asymmetric Nucleophilic Displacement Reactions on Chiral α-Substituted
Aldehyde Hydrazones.
242) D. Enders, H. Gielen, K. Breuer, Molecules Online 1998, 2, 105 - 108. Immobilized
Triazolium Salts as Precursors to Chiral Carbenes - Rhodium-Catalyzed
Asymmetric Hydrosilylation as a First Test Reaction.
243) D. Enders, R. Joseph, C. Poiesz, Tetrahedron 1998, 54, 10069 - 10078. Electrophilic
Amination of Hydrazones: A New Synthetic Route to Protected α-Hydrazino- and
α-Aminoketones.
244) D. Enders, I. Meyer, J. Runsink, G. Raabe, Tetrahedron 1998, 54, 10733 - 10752.
Diastereoselective 1,3-Dipolar Cycloadditions with Enantiopure Azomethin Ylids.
245) D. Enders, H. Gielen, K. Breuer, Z. Naturforsch. 1998, 53b, 1035 - 1038. Axial
Chirality in Square-Planar Metal Complexes.
246) A. A. Birkbeck, D. Enders, Tetrahedron Lett. 1998, 39, 7823 - 7826. The Total
Synthesis of (+)-Pectinatone: An Iterative Alkylation Approach Based on the
SAMP-Hydrazone Method.
247) D. Enders, R. Hett, Synlett 1998, 961 - 962. Asymmetric Synthesis of α’-Silylated
α,β-Epoxy Ketones via Darzens Reaction.
248) D. Enders, T. Hundertmark, C. Lampe, U. Jegelka, I. Scharfbillig, Eur. J. Org.
Chem. 1998, 2839 - 2849. Highly Diastereo- and Enantioselective Synthesis of
Protected anti-1,3-Diols.
25
249) D. Enders, R. Lochtman, M. Meiers, S. F. Müller, R. Lazny, Synlett 1998, 1182 -
1184. Efficient N-N-Bond Cleavage of Chiral Trisubstituted Hydrazines with
BH3.THF.
250) D. Enders, C. Poiesz, R. Joseph, Tetrahedron: Asymmetry 1998, 9, 3709 - 3716.
Enantioselective Synthesis of Protected α-Aminoketones via Electrophilic
Amination of α-Silylketones with an Oxaziridine.
251) D. Enders, L. Kramps, J. Zhu, Tetrahedron: Asymmetry 1998, 9, 3959 - 3962. Zinc-
mediated Asymmetric Epoxidation of Nitro Alkenes with Oxygen.
252) S. Bräse, D. Enders, J. Köbberling, F. Avemaria, Angew. Chem. 1998, 110, 3614 -
3616; Angew. Chem. Int. Ed. Engl. 1998, 37, 3413 - 3415. Ein überraschender
Festphaseneffekt: Entwicklung eines regenerierbaren „spurlosen“ Linker-Systems
für Festphasenreaktionen.
253) D. Enders, S. F. Müller, G. Raabe, Angew. Chem. 1999, 111, 212 - 214; Angew.
Chem. Int. Ed. Engl. 1999, 38, 195 - 197. Enantioselektive Synthese von ß-
Aminosulfonen via azaanaloge Michael-Addition an Alkenylsulfone.
254) J. H. Teles, K. Breuer, D. Enders, H. Gielen, Synth. Commun. 1999, 29, 1 - 9. One
Pot Synthesis of 3,4-Disubstituted 1-Alkyl-4H-1,2,4-Triazol-1-ium Salts.
255) D. Enders, T. Hundertmark, R. Lazny, Synth. Commun. 1999, 29, 27 - 33. Copper
(II) Chloride Mediated Racemization-Free Hydrolysis of α-Alkylated Ketone
SAMP-Hydrazones.
256) D. Enders, P. Teschner, R. Gröbner, G. Raabe, Synthesis 1999, 237 - 242. Asym-
metric Michael Additions via 6- and 7-Membered Lactone SAMP-Hydrazones.
Diastereo- and Enantioselective Synthesis of Substituted Lactone Esters.
257) D. Enders, M. Bartsch, J. Runsink, Synthesis 1999, 243 - 247. Diastereo- and
Enantioselective Formal Synthesis of (+)-Conagenin via Asymmetric [2,3]-Wittig
Rearrangement.
258) D. Enders, I. Meyer, J. Runsink, G. Raabe, Heterocycles 1999, 50, 995 - 1024. Dia-
stereo- and Enantioselective Synthesis of Δ2-1,2,4-Oxadiazolines by 1,3-Dipolar
Cycloaddition of Nitrile Oxides with Chiral Hydrazones.
259) R. Lazny, J. Poplawski, J. Köbberling, D. Enders, S. Bräse, Synlett 1999, 1304 -
1306. Triazenes: A Useful Protecting Strategy for Sensitive Secondary Amines.
26
260) S. Bräse, J. Köbberling, D. Enders, R. Lazny, M. Wang, S. Brandtner, Tetrahedron
Lett. 1999, 40, 2105 - 2108. Triazenes as Robust and Simple Linker for Amines in
Solid-Phase Organic Synthesis.
261) D. Enders, C. R. Thomas, J. Runsink, Tetrahedron: Asymmetry 1999, 10, 323 - 326.
5-Amino-4-aryl-2,2-dimethyl-1,3-dioxans: Application as Chiral NMR Shift
Reagents and Derivating Agents for Acidic Compounds.
262) D. Enders, T. Hundertmark, Eur. J. Org. Chem. 1999, 751 - 756. Asymmetric Syn-
thesis of (+)- and (–)-Streptenol A.
263) D. Enders, J. Vázquez, J. Chem. Soc. Chem. Commun. 1999, 701 -702. Diastereo-
and Enantioselective Synthesis of 2,8-Dioxabicyclo[3.3.0]octan-3-one Derivatives.
264) D. Enders, A. S. Amaya, F. Pierre, New J. Chem. 1999, 23, 261 - 262. Conversion
of Aldehydes to Amides via Dimethylsulfoxide Oxidation of the Corresponding α-
Aminonitriles.
265) D. Enders, J. Vázquez, Synlett 1999, 629 - 631. Asymmetric Synthesis of α-
Substituted β-Formyl δ-Lactones via a Michael Addition / α-Alkylation Protocol.
266) D. Enders, H. Sun, F. R. Leusink, Tetrahedron 1999, 55, 6129 - 6138. Diastereo-
and Enantioselective Synthesis of 4- and 3,4-Substituted 2-Acetoxy-
butyrolactones.
267) D. Enders, S. F. Müller, G. Raabe, Synlett 1999, 741 - 743. Asymmetric Synthesis
of α-Substituted β-Amino Sulfones by aza-Michael Addition / α-Alkylation.
268) D. Enders, J. P. Shilvock, G. Raabe, J. Chem. Soc. Perkin 1. 1999, 1617 - 1620.
Asymmetric Nucleophilic α-Amino-acylation with Metalated Chiral Amino
Nitriles: Enantioselective Synthesis of 3-Substituted 5-Amino-4-oxo-esters via
Asymmetric Michael Addition.
269) D. Enders, D. Klein, Synlett 1999, 719 - 720. A Novel Enantioselective Synthesis of
α-Azido Ketones.
270) D. Enders, T. Otten, Synlett 1999, 747 - 749. α-Silyl Controlled Asymmetric
Michael Additions of Acyclic and Cyclic Ketones to Nitroalkenes.
271) D. Enders, T. Hundertmark, Tetrahedron Lett. 1999, 40, 4169 - 4172. Iterative
Asymmetric Synthesis of Protected anti-1,3-Polyols.
27
272) D. Enders, L. Wortmann, B. Dücker, G. Raabe, Helv. Chim. Acta. 1999, 82, 1195 -
1201. Asymmetric Synthesis of 1,2,3,4,5,6-Hexahydro-5-hydroxypyrimidin-2-ones
as Potential HIV-Protease-Inhibitors.
273) D. Enders, R. Peters, R. Lochtman, G. Raabe, Angew. Chem. 1999, 111, 2579 -
2581; Angew. Chem. Int. Ed. 1999, 38, 2421 - 2423. Asymmetrische Synthese
neuer planar- und zentral-chiraler Ferrocenyl-Liganden.
274) D. Enders, E. Diéz, R. Fernández, E. Martín-Zamora, J. M. Muñoz, R. R.
Pappalardo, J. M. Lassaletta, J. Org. Chem. 1999, 64, 6329 - 6336. Electrophilic
and Nucleophilic Reactivities of the Azomethine Carbon of SAMP-Hydrazones:
Stereoselective Synthesis of γ-Amino Ketone Derivates.
275) F. Pierre, D. Enders, Tetrahedron Lett. 1999, 40, 5301 - 5305. Nucleophilic
Alkenoylation of Aldehydes with Metalated α-Aminonitriles: Regioselective
Synthesis of α-Hydroxyenones.
276) D. Enders in „ Horizonte - Die RWTH auf dem Weg ins 21. Jahrhundert“, R.
Walter, B. Rauhut (Hrsg.), Springer Verlag, Berlin, 1999, S. 111. Asymmetrische
Synthese spiegelbildlicher Moleküle.
277) D. Enders, K. Breuer, Comprehensive Asymmetric Catalysis, Vol. 3, E. N.
Jacobsen, A. Pfaltz, H. Yamamoto (Hrsg.), Springer Verlag, Berlin, 1999, 1093 -
1102. Addition of Acyl Carbanion Equivalents to Carbonyl Groups and Enones.
278) D. Enders, C. Thiebes, J. Indian Chem. Soc. 1999, 76, 561 - 564. Enantioselective
Synthesis of Both Enantiomers of Bgugaine Employing the SAMP-Hydrazone
Method.
279) D. Enders, R. Peters, J. Runsink, J. W. Bats, Org. Lett. 1999, 1, 1863 - 1866. Novel
Ferrocenyl Ligands with Planar and Central Chirality in Pd-Catalyzed Allylic
Substitutions.
280) D. Enders, P. Teschner, G. Raabe, Heterocycles 2000, 52, 733 - 749. Diastereo- and
Enantioselective Synthesis of γ- and δ-Lactams Bearing a Propionic Acid α-Side-
Chain via Michael Addition of N-Dialkylamino Lactams to Enoates.
281) D. Enders, S. F. Müller, G. Raabe, J. Runsink, Eur. J. Org. Chem. 2000, 879 - 892.
Asymmetric Synthesis of α-Substituted β-Amino Sulfones by aza-Michael Addition
to Alkenyl Sulfones and Subsequent α-Alkylation.
28
282) D. Enders, G. Geibel, S. Osborne, Chem. Eur. J. 2000, 6, 1302 - 1309. Diastereo-
and Enantioselective Total Synthesis of Stigmatellin A.
283) D. Enders, L. Wortmann, R. Peters, Acc. Chem. Res. 2000, 33, 157 - 169. Recovery
of Carbonyl Compounds from N,N-Dialkylhydrazones.
284) D. Enders, J. Adam, D. Klein, T. Otten, Synlett 2000, 1371 - 1384. α-Silyl Ketone
Controlled Asymmetric Syntheses.
285) D. Enders, J. Vázquez, G. Raabe, Eur. J. Org. Chem. 2000, 893 - 901.
Formaldehyde SAMP-Hydrazone as a Neutral Formyl Anion Equivalent:
Asymmetric Synthesis of Substituted β-Formyl δ-Lactones and Furofuran
Lactones.
286) D. Enders, A. Nühring, J. Runsink, Chirality 2000, 12, 374 - 377. Efficient Asym-
metric Synthesis of α-Alkylated Cyclohexanedione-1,4-Derivatives - Important
Chiral Building Blocks in the Synthesis of Natural Products.
287) D. Enders, C. Thiebes, Synthesis 2000, 510 - 512. Efficient Synthesis of (2S,12’R)-
2-(12’-Aminotridecyl)pyrrolidine: A Defense Alkaloid of the Mexican Bean Beetle.
288) E. Deniau, D. Enders, Tetrahedron Lett. 2000, 41, 2347 - 2350. A New Simple and
Convenient Synthesis of 3-Substituted Phthalimidines.
289) S. Schunk, D. Enders, Org. Lett. 2000, 2, 907 - 910. Solid-Phase Synthesis of β-
Lactams via the Ester Enolate-Imine Condensation Route.
290) D. Enders, S. Oberbörsch, J. Adam, Synlett 2000, 644 - 646. α-Silyl Controlled
Asymmetric Mannich Reactions of Acyclic Ketones with Imines.
291) A. Job, R. Nagelsdiek, D. Enders, Collect. Czech Chem. Commun. 2000, 65, 524 -
538. Versatile Enantioselective Synthesis of Four Diastereomers of Serricornin, a
Sex Pheromone of the Cigarette Beetle, Using the SAMP/RAMP-Hydrazone
Method.
292) D. Enders, P. Teschner, G. Raabe, Synlett 2000, 637 - 640. Diastereo- and Enantio-
selective Synthesis of α-(β-Aminoalkyl)-Substituted γ-Lactams via Michael
Addition to Nitroalkenes.
293) D. Enders, C. F. Janeck, J. Runsink, Synlett 2000, 641 - 643. Asymmetric
Synthesis of γ-Amino Ketones and Nitriles via β-Amino-ethylation of SAMP-
Hydrazones with Tosylaziridine.
29
294) D. Enders, R. Peters, R. Lochtman, J. Runsink, Eur. J. Org. Chem. 2000, 2839 -
2850. Enantioselective Synthesis of Planar Chiral ortho-Functionalized
Ferrocenylketones.
295) D. Enders, J. P. Shilvock, Chem. Soc. Rev. 2000, 29, 359 - 373. Some Recent
Applications of α-Amino Nitrile Chemistry.
296) D. Enders, R. Peters, R. Lochtman, G. Raabe, J. Runsink, J. W. Bats, Eur. J. Org.
Chem. 2000, 3399 - 3426. Asymmetric Synthesis of Novel Ferrocenyl Ligands with
Planar and Central Chirality and Their Application to Pd-Catalyzed Allylic
Substitutions.
297) D. Enders, C. F. Janeck, G. Raabe, Eur. J. Org. Chem. 2000, 3337 - 3345. Asym-
metric β-Aminoethylation of Ketones and Nitriles with Tosylaziridines Employing
the SAMP-Hydrazone Method.
298) D. Enders, E. Ullrich, Tetrahedron: Asymmetry 2000, 11, 3861 - 3865. Asymmetric
pinacol coupling of aromatic aldehydes with TiCl2/enantiopure amine or hydrazine
reagents.
299) D. Enders, C. Thiebes, Synlett 2000, 1745 - 1748. First Enantioselective Synthesis
of Dendrobatid Alkaloids Indolizidine (–)-209I and (–)-223J.
300) D. Enders, A. Ridder, Synthesis 2000, 1848 - 1851. First Asymmetric Synthesis of
Stigmolone: The Fruiting Body Inducing Pheromone of the Myxobacterium
Stigmatella Aurantiaca.
301) J. Fleischhauer, S. Gabriel, D. Enders, A. Nühring, A. Wollmer, Z. Naturforsch.
2000, 55B, 1011 - 1014. CD-Spectroscopical Investigations for the Determination
of the Absolute Configuration of α-Alkylated 1,4-Cyclohexanedione Derivatives.
302) D. Enders, L. Tedeschi, J. W. Bats, Angew. Chem. 2000, 112, 4774 - 4776; Angew.
Chem. Int. Ed. 2000, 39, 4605 - 4607. Asymmetrische Synthese α-substituierter β-
Nitrophosphonsäuren durch phospha-analoge Michael-Addition an aromatische
Nitroalkene.
303) D. Enders, T. Schüßeler, New. J. Chem. 2000, 24, 973 - 975. First Asymmetric
Synthesis of 6-Methyl-3-nonanone, the Female-produced Sex Pheromone of the
Caddisfly Hesperophylax Occidentalis.
30
304) D. Enders, D. Nguyen, Synthesis 2000, 2092 - 2098. Synthesis of Enantioenriched
Substituted Tetrahydrofurans and Tetrahydropyrans via Iron Mediated Chirality
Transfer and Ring Closure.
305) D. Enders, J. H. Kirchhoff, Synthesis 2000, 2099 - 2105. Asymmetric Total
Synthesis of (+)-2-epi-Deoxoprosopinine.
306) D. Enders, S. von Berg, B. Jandeleit, Org. Synth. 2000, 78, 169 - 176.
Diethyl[(phenylsulfonyl)methyl]phosphonate.
307) D. Enders, S. von Berg, B. Jandeleit, Org. Synth. 2000, 78, 177 - 188. (–)-(E,S)-3-
(Benzyloxy)-1-butenyl phenyl sulfone via a Horner-Wadsworth-Emmons Reaction
of (–)-(S)-2-(Benzyloxy)propanal.
308) D. Enders, S. von Berg, B. Jandeleit, Org. Synth. 2000, 78, 189 - 201. (+)-
(1R,2S,3R) - Tetracarbonyl[(1-3η)-1-(phenylsulfonyl)-but-2-en-1-yl]iron(1+) tetra-
fluoroborate.
309) J. H. Kirchhoff, S. Bräse, D. Enders, J. Comb. Chem. 2001, 3, 71 - 77. A Novel Hy-
drazine Linker Resin and its Application for the Solid-Phase Synthesis of α-
Branched Primary Amines.
310) D. Enders, H. Gielen, J. Organomet. Chem. 2001, 617-618, 70 - 80. Synthesis of
Chiral Triazolinylidene and Imidazolinylidene Transition Metal Complexes and
First Application in Asymmetric Catalysis.
311) E. Deniau, D. Enders, Tetrahedron 2001, 57, 2581 - 2588. Synthesis of 3-Alkyl-1-
isoindolinones by Alkylation of a Benzotriazolyl Substituted N-Dimethylamino-
phthalimidine.
312) D. Enders, C. Thiebes, Pure and Appl. Chem. 2001, 73, 573 - 578. Efficient Stereo-
selective Syntheses of Piperidine, Pyrrolidine and Indolizidine Alkaloids.
313) D. Enders, J. H. Kirchhoff, J. Köbberling, T. H. Peiffer, Org. Lett. 2001, 3, 1241 -
1244. Asymmetric Synthesis of α-Branched Primary Amines on Solid Support via
Novel Hydrazine Resins.
314) D. Enders, V. Braig, G. Raabe, Can. J. Chem. 2001, 79, 1528 - 1535. Asymmetric
Synthesis of 3-Aryl-Substituted 2,3-Dihydro-1H-isoindol-1-ones.
315) D. Enders, T. Klumpen, J. Organomet. Chem. 2001, 637 - 639, 698 - 709.
Asymmetric Synthesis of Planar Chiral 2-Mono- and 2,2'-Disubstituted 1,1'-
Bisbenzoylferrocenes.
31
316) D. Enders, K. Funabiki, Org. Lett. 2001, 3, 1575 - 1577. Efficient Asymmetric
Synthesis of α-Trifluoromethyl Substituted Primary Amines via Nucleophilic 1,2-
Addition to Trifluoroacetaldehyde SAMP- or RAMP-Hydrazone.
317) D. Enders, A. Nühring, J. Runsink, G. Raabe, Synthesis 2001, 1406 - 1414.
Asymmetric Synthesis of Protected 2-Keto-1,3-diol and 1,2,3-Triol Building Blocks
Bearing a Quaternary Stereogenic Center.
318) D. Enders, B. Jandeleit, S. von Berg, G. Raabe, J. Runsink, Organometallics 2001,
20, 4312 - 4332. Iron Mediated Allylic Substitution Reactions with Chirality
Transfer. Stereochemistry of the Formation of Diastereo- and Enantiomerically
Enriched Olefinic and Allylic Tetracarbonyl Iron Complexes.
319) D. Enders, P. Teschner, G. Raabe, J. Runsink, Eur. J. Org. Chem. 2001, 4463 -
4477. Asymmetric Electrophilic Substitutions at the α-Position of γ- and δ-
Lactams.
320) D. Enders, A. Job, M. Wolberg, M. Müller, Synlett 2001, 1796 - 1798. Asymmetric
Synthesis of S-(+)-Argentilactone and S-(–)-Goniothalamin.
321) J. Fleischhauer, S. Gabriel, A. Job, D. Enders, A. Wollmer, Z. Naturforsch. 2001,
56b, 1344 - 1348. CD-Spectroscopic Investigations for the Determination of the
Absolute Configuration of (4R, 6S, 7S)-Serricornin.
322) S. Schunk, D.Enders, Org. Lett. 2001, 3, 3177 - 3180. Solid-Phase Synthesis of β-
Amino ketones and Six-Ring Carbamates via Immobilized α-Alkoxycarbonylamino
Sulfones.
323) N. Vignola, S. Dahmen, D. Enders, S. Bräse, Tetrahedron Lett. 2001, 42, 7833 -
7836. Synthesis of Alkyl Sulfonates from Sulfonic Acids or Sodium Sulfonates
Using Solid-Phase Bound Reagents.
324) D. Enders, O. M. Berner, N. Vignola, J. W. Bats, J. Chem. Soc. Chem. Commun.
2001, 2498 - 2499. Diastereo- and Enantioselective Synthesis of α,β-Disubstituted
γ-Nitro Methyl Sulfonates.
325) D. Enders, S. Faure, M. Potthoff, J. Runsink, Synthesis 2001, 2307 - 2319.
Diastereoselective Electrophilic Fluorination of Enantiopure α-Silylketones Using
N-Fluorobenzosulfonimide. Regio- and Enantioselective Synthesis of α-
Fluoroketones.
32
326) L. Tedeschi, D. Enders, Org. Lett. 2001, 3, 3515 - 3517. Asymmetric Synthesis of β-
Phosphono Malonates via Fe2O3 Mediated phospha-Michael Addition to
Knoevenagel Acceptors.
327) D. Enders, U. Kallfass, B. Nolte, Synlett 2002, 33 - 36. A Short Diastereo- and
Enantioselective Synthesis of cis-4,5-Disubstituted Oxazolidin-2-ones.
328) D. Enders, N. Vignola, O. M. Berner, J. W. Bats, Angew. Chem. 2002, 114, 116 -
119; Angew. Chem. Int. Ed. 2002, 41, 109 - 111. The First Highly Efficient
Asymmetric Synthesis of α-Substituted Methyl Sulfonates.
329) D. Enders, A. Seki, Synlett 2002, 26 - 28. Proline-Catalyzed Enantioselective
Michael Additions of Ketones to Nitrostyrene.
330) D. Enders, M. Voith, Synlett 2002, 29 - 32. Asymmetric Synthesis of Pseudo - C2-
Symmetric 2-Methyl Substituted 1,3-Diols.
331) A. Job, C. F. Janeck, W. Bettray, R. Peters, D. Enders, Tetrahedron 2002, 58, 2253
- 2329. The SAMP/RAMP-Hydrazone Methodology in Asymmetric Synthesis.
332) D. Enders, S. Wallert, Synlett 2002, 304 - 306. Asymmetric Synthesis of β-Amino-
cyclohexyl sulfonates via aza-Michael Addition.
333) D. Enders, S. Oberbörsch, Synlett 2002, 471 - 473. Asymmetric Mannich Reactions
with α-Silylated Trimethylsilyl Enol Ethers and N-Alkoxycarbonyl Imines.
334) O. M. Berner, L. Tedeschi, D. Enders, Eur. J. Org. Chem. 2002, 1877 - 1894.
Asymmetric Michael Additions to Nitroalkenes.
335) D. Enders, U. Kallfass, Angew. Chem. 2002, 114, 1822 – 1824; Angew. Chem. Int.
Ed. 2002, 41, 1743 - 1745. Ein effizienter nucleophiler Carben-Katalysator für die
asymmetrische Benzoinkondensation.
336) D. Enders, A. Schaadt, Synlett 2002, 498 - 500. A Flexible Asymmetric Synthesis
of 1,2-anti tert-Butylsulfanyl Amines.
337) J. Vázquez, A. Prieto, R. Fernández, D. Enders, J. M. Lassaletta, J. Chem. Soc.
Chem. Commun. 2002, 498 - 499. Asymmetric Michael Addition of Formaldehyde
N,N-Dialkylhydrazones to Alkylidene Malonates.
338) D. Enders, V. Lausberg, G. Del Signore, O. M. Berner, Synthesis 2002, 515 - 522. A
General Approach to the Asymmetric Synthesis of Lignans: (–)-Methyl Piperitol, (–
33
)-Sesamin, (–)-Aschantin, (+)-Yatein, (+)-Dihydroclusin, (+)-Burseran, and (–)-Iso-
stegane.
339) J. L. Vicario, A. Job, M. Wolberg, M. Müller, D. Enders, Org. Lett. 2002, 4, 1023 -
1026. Asymmetric Total Synthesis of (–)-Callystatin A Employing the
SAMP/RAMP Hydrazone Alkylation Methodology.
340) D. Enders, B. Nolte, G. Raabe, J. Runsink, Tetrahedron: Asymmetry 2002, 13, 285
- 291. Asymmetric Synthesis and Structural Assignment of (–)-α-Conhydrine.
341) D. Enders, S. Ince, Synthesis 2002, 619 - 624. Chiral Dihydroxyacetone
Equivalents in Synthesis: An Expedient Diastereo- and Enantioselective Synthesis
of Differentially Protected Ketopolyols.
342) D. Enders, S. Ince, M. Bonnekessel, J. Runsink, G. Raabe, Synlett 2002, 962 - 966.
Chiral Dihydroxyacetone Equivalents in Synthesis: Rapid Assembly of Styryl 1,2-
Polyols as an Entry to the Styryllactone Family of Natural Products.
343) D. Enders, B. Nolte, J. Runsink, Tetrahedron: Asymmetry 2002, 13, 587 - 593.
Asymmetric Synthesis of 2-Substituted Piperidin-3-ols.
344) D. Enders, L. Wortmann, Heterocycles 2002, 58, 293 - 299. Asymmetric Synthesis
of 4,6-Disubstituted 1,2,3,4,5,6-Hexahydro-5-hydroxypyrimidin-2-ones as Potential
HIV-Protease Inhibitors.
345) D. Enders, T. Schüßeler, Tetrahedron Lett. 2002, 43, 3467 - 3470. Asymmetric Syn-
thesis of all Stereoisomers of 7,11-Dimethylheptadecane and 7-Methylhepta-
decane, the Female Pheromone Components of the Spring Hemlock Looper and the
Pitch Pine Looper.
346) J. L. Vicario, A. Job, M. Wolberg, M. Müller, D. Enders, Chem. Eur. J. 2002, 8,
4272 - 4284. Asymmetric Total Synthesis of (–)-Callystatin A and (–)-20-epi-
Callystatin A Employing Chemical and Biological Methods.
347) D. Enders, M. Voith, S. J. Ince, Synthesis 2002, 1775 - 1779. Preparation and
Reactions of 2,2-Dimethyl-1,3-dioxan-5-one-SAMP-hydrazone - a Versatile Chiral
Dihydroxyacetone Equivalent.
348) D. Enders, M. Voith, Synthesis 2002, 1571 - 1577. Asymmetric Synthesis of Mono-
protected Double Allylic Alcohols.
349) D. Enders, S. Wallert, Tetrahedron Lett. 2002, 43, 5109 - 5111. Efficient
Asymmetric Synthesis of 3-Substituted β-Sultams.
34
350) D. Enders, T. Schüßeler, Synthesis 2002, 2280 - 2288. First Highly Efficient
Asymmetric Synthesis of the Hyrtios Erectus Diketotriterpenoid.
351) D. Enders, C. R. Thomas, N. Vignola, G. Raabe, Helv. Chim. Acta 2002, 85, 3657 -
3677. Asymmetric Synthesis of α-Substituted N-Methyl-Sulfonamides.
352) S. Schunk, D. Enders, J. Org. Chem. 2002, 67, 8034 - 8042. Solid-Phase Synthesis
of Monocyclic β-Lactam Derivatives.
353) D. Enders, W. Harnying, N. Vignola, Synlett 2002, 1727 - 1729. A Practical
Approach towards the Asymmetric Synthesis of α,γ-Substituted γ-Sultones.
354) D. Enders, O. M. Berner, N. Vignola, W. Harnying, Synthesis 2002, 1945 - 1952.
Asymmetric Michael Addition of Chiral Lithiated Sulfonates to Nitroalkenes. Dia-
stereo- and Enantioselective Synthesis of α,β-Disusbstituted γ-Nitro and β-Alkoxy-
carbonyl Methyl Sulfonates.
355) E. Deniau, D. Enders, Tetrahedron Lett. 2002, 43, 8055 - 8058. A New and
Versatile Synthetic Route to 2-Dimethylamino-3-Alkyl and Arylmethylene-2,3-
Dihydro-1H-Isoindol-1-ones.
356) D. Enders, M. Meiers, Synthesis 2002, 2542 - 2560. Diastereo- and
Enantioselective Synthesis of C2-Symmetric 1,n-Diamines by Nucleophilic
Addition to Dialdehyde-SAMP-Hydrazones.
357) K. Funabiki, N. Nagamori, M. Matsui, D. Enders, Synthesis 2002, 2585 - 2588.
Asymmetric Synthesis of Both Enantiomers of α-Trifluoromethyl Substituted
Homoallylamine.
358) D. Enders, J. Adam, S. Oberbörsch, D. Ward, Synthesis 2002, 2737 - 2748. Asym-
metric Mannich Reactions by α-Silyl Controlled Aminomethylation of Ketones.
359) N. Vignola, S. Dahmen, D. Enders, S. Bräse, J. Comb. Chem. 2003, 5, 138 - 144.
Efficient Synthesis of Sulfonic, Phosphoric and Phosphinic Esters Employing
Alkylating Polymer-Bound Reagents.
360) D. Enders, G. Del Signore, O. M. Berner, Chirality 2003, 15, 510 - 513. First
Asymmetric Synthesis of (–)-Lintetralin via Intramolecular Friedel-Crafts-Type
Cyclization.
361) D. Enders, F. Burkamp, Coll. Czech. Chem. Commun. 2003, 68, 975 - 1006. α-
Heterosubstituted Aldehydes in Organic Synthesis. Enantioselective Approaches
to New Analogues of Mevinic Acids.
35
362) J. M. Lassaletta, J. Vázquez, A. Prieto, R. Fernández, G. Raabe, D. Enders, J. Org.
Chem. 2003, 68, 2698 - 2703. Asymmetric Synthesis of Succinic Semialdehyde
Derivatives.
363) D. Enders, K. Breuer, U. Kallfass, T. Balensiefer, Synthesis 2003, 1292 -1295.
Preparation and Application of 1,3,4-Triphenyl-4,5-dihydro-1H-1,2,4-triazol-5-
ylidene, a Stable Carbene.
364) E. Deniau, D. Enders, A. Couture, P. Grandclaudon, Tetrahedron: Asymmetry
2003, 14, 2253 - 2258. A New Synthetic Route to Highly Enantioenriched 3-
Substituted 2,3-Dihydro-1H-isoindol-1-ones.
365) D. Enders, T. Klumpen, G. Raabe, Synlett 2003, 1198 – 1200. Asymmetric
Synthesis of Planar Chiral 2-Monosubstituted Diferrocenyl Ketones.
366) D. Enders, A. Moll, A. Schaadt, G. Raabe, J. Runsink, Eur. J. Org. Chem. 2003,
3923 - 3938. A Flexible Asymmetric Synthesis of anti-1,2-Sulfanyl Amines.
367) D. Enders. S. Wallert, Synthesis 2003, 1856 - 1868. Asymmetric Synthesis of β-
Amino-cyclohexyl sulfonates, β-Sultams and γ-Sultones.
368) D. Enders, W. Harnying, N. Vignola, Eur. J. Org. Chem. 2003, 3939 - 3947.
Allylation of Chiral Lithiated Sulfonates. Asymmetric Synthesis of α, γ-Substituted
γ-Sultones.
369) D. Enders, A. Lenzen, Synlett 2003, 2185 - 2187. Asymmetric Total Synthesis of
Attenol A and B.
370) D. Enders, M. Moser, Tetrahedron Lett. 2003, 44, 8479 - 8481. Asymmetric
Strecker Synthesis by Addition of Trimethylsilyl Cyanide to Aldehyde SAMP-
Hydrazones.
371) D. Enders, D. Steinbusch, Eur. J. Org. Chem. 2003, 4450 - 4454. An Efficient
Asymmetric Synthesis of Tarchonanthuslactone.
372) D. Enders, M. Haas, Synlett, 2003, 2182 - 2184. Asymmetric Synthesis of 4,5-Di-
substituted 3-Hydroxy δ-Lactones – Prelactone B and Prelactone V.
373) D. Enders, W. Harnying, Arkivoc 2004, (ii) 181 - 188. Asymmetric Synthesis of α,γ-Substituted γ-Alkoxy Methyl Sulfonates via Diastereospecific Ring-Opening of
Sultones.
36
374) D. Enders, L. Wortmann, G. Raabe, B. Dücker, Heterocycles 2004, 62, 559 - 581. A
Highly Flexible Route to 1,2,3,4,5,6-Hexahydro-5-hydroxypyrimidin-2-ones as
Potential HIV Protease Inhibitors.
375) D. Enders, T. Balensiefer, Acc. Chem. Res. 2004, 37, 534 - 541. Nucleophilic Carbe-
nes in Asymmetric Organocatalysis.
376) D. Enders, M. Backes in Enzyclopedia of Reagents for Organic Synthesis, L. A. Pa-
quette, Ed., Wiley, New York, 2004. Tetramethylguanidinium Azide.
377) D. Enders, G. Del Signore, Tetrahedron: Asymmetry 2004, 15, 747 – 751. Efficient
Asymmetric Synthesis of α- (Heteroaryl)alkylamines by 1,2-Addition of Lithiated
Hetarenes to Aldehyde SAMP-Hydrazones.
378) D. Enders, C. Rijksen, E. Bremus-Köbberling, A. Gillner, J. Köbberling,
Tetrahedron Lett. 2004, 45, 2839 - 2841. A Triazene-based New Photolabile Linker
in Solid Phase Chemistry.
379) D. Enders, W. Harnying, G. Raabe, Synthesis 2004, 590 - 594. Diastereoselective
Hydrolysis of α,γ-Substituted γ-Sultones in the Asymmetric Synthesis of γ-Hydroxy
Sulfonates.
380) D. Enders, A. Müller-Hüwen, Eur. J. Org. Chem. 2004, 1732 - 1739. Asymmetric
Synthesis of 2-Amino-1,3-diols and D-erythro-Sphinganine.
381) D. Enders, G. Del Signore, Heterocycles 2004, 64, 101 - 120. Asymmetric Synthesis
of Heterocyclic β-Aminosulfones via Nucleophilic 1,2-Addition of 2-Lithiobenzothio-
phene to Aldehyde-SAMP-Hydrazones.
382) D. Enders, A. Lenzen, M. Müller, Synthesis 2004, 1486 - 1496. Efficient
Asymmetric Syntheses of (+)-Strictifolione.
383) D. Enders, M. Backes, Tetrahedron: Asymmetry 2004, 15, 1813 - 1817. First Asym-
metric Synthesis of Both Enantiomers of Tropional® and their Olfactorial
Evaluation.
384) D. Enders, M. Moser, G. Geibel. M. C. Laufer, Synthesis 2004, 2040 - 2046.
Diastereo- and Enantioselective Synthesis of Differently N,O-Protected 1,3-Amino
Alcohols with Three Neighbouring Stereogenic Centers.
385) D. Enders, O. Niemeier, Synlett 2004, 2111 - 2114. Thiazol-2-ylidene Catalysis in
Intramolecular Crossed Aldehyde-Ketone Benzoin Reactions.
37
386) D. Enders, J. Gries, Z.-S. Kim, Eur. J. Org. Chem. 2004, 4471 - 4482. Asymmetric
Synthesis of 2-Mono- and 2,3-trans-Disubstituted Azetidines.
387) L. Doszczak, T. Gasperi, A. Saint-Dizier, M. A. Loreto, D. Enders, Chem. &
Biodiversity 2004, 1, 1921 - 1935. Silylating Reagents – a Powerful Tool in
Constructing Isosteric Analogues of Highly Branched Odorants.
388) D. Enders, W. Harnying, Synthesis 2004, 2910 - 2918. A Highly Efficient
Asymmetric Synthesis of Homotaurine Derivatives via Diastereoselective Ring
Opening of γ-Sultones.
389) D. Enders, V. Braig, M. Boudou, G. Raabe, Synthesis 2004, 2980-2990.
Asymmetric Synthesis of 3-Substituted Dihydro-2H-isoquinolin-1-ones, Dihydro-
and Tetrahydroisoquinolines via 1,2-Addition/Ring Closure.
390) D. Enders, N. Vignola, O. M. Berner, W. Harnying, Tetrahedron 2005, 61, 3231 -
3243. Efficient Asymmetric Synthesis of α-Alkylated Benzylic Methyl Sulfonates.
391) D. Enders, Z.-X. Chen, Lett. Org. Chem. 2005, 2, 156 - 159. Synthesis of β-Benzyl-
sulfanyl-β-trifluoromethyl-α-amino acids via Michael Addition in the Presence of
Et3N/LiBr.
392) E. Deniau, D. Enders, A. Couture, P. Grandclaudon, Tetrahedron: Asymmetry,
2005, 16, 875 - 881. Asymmetric Synthesis of 3-Hetero-substituted 2,3-Dihydro-
1H-isoindol-1-ones.
393) D. Enders, Z.-X. Chen, G. Raabe, Synthesis 2005, 306 - 310. Stereoselective
Synthesis of 3-Substituted Ethyl (Z)-4,4,4-Trifluoro-2-formylamino-2-butenoates.
394) D. Enders, M. Voith, A. Lenzen, Angew. Chem. 2005, 117, 1330 – 1351; Angew.
Chem. Int. Ed. 2005, 44, 1304 – 1325. The Dihydroxyacetone Unit - a Versatile C3-
Building Block in Organic Synthesis.
395) D. Enders, C. Grondal, Angew. Chem. 2005, 117, 1235 – 1238. Angew. Chem. Int.
Ed. 2005, 44, 1210 – 1212. Direkte organokatalytische de novo-Synthese von
Kohlenhydraten.
396) R. Kumar, M. Raclaru, T. Schüßeler, J. Gruber, R. Sadre, W. Lühs, K. M. Zarhoul,
W. Friedt, D. Enders, M. Frentzen, D. Weier, FEBS Letters 2005, 579, 1357 –
1364. Characterisation of Plant Tocopherol Cyclases and their Overexpression in
Transgenic Brassica napus Seeds.
38
397) D. Enders, M. Milovanovic, E. Voloshina, G. Raabe, J. Fleischhauer, Eur. J. Org.
Chem. 2005, 1984 - 1990. First Asymmetric Synthesis and Determination of the
Absolute Configuration of a Lignan Isolated from Virola sebifera.
398) D. Enders, A. Moll, Synthesis 2005, 1807 - 1816. Asymmetric Synthesis of cis-3,4-
Disubstituted β-Sultams.
399) D. Enders, M. R. M. Hüttl, Synlett 2005, 991 - 993. Direct Organocatalytic α-Fluor-
ination of Aldehydes and Ketones.
400) D. Enders, I. Breuer, A. Nühring, Eur. J. Org. Chem. 2005, 2677 - 2683. First
Asymmetric Synthesis of (+)-Sordidin and (–)-7-epi-Sordidin, Aggregation
Pheromones of the Banana Weevil Cosmopolites sordidus.
401) D. Enders, M. Boudou, J. Gries in New Methods for the Asymmetric Synthesis of
Nitrogen Heterocycles, J. L. Vicario, D. Badia, L. Carrillo (Eds.), Research
Signpost, Trivandrum, India, 2005, 1 - 31. Asymmetric Syntheses of Four-, Five-
and Six-Membered N-Heterocycles Employing the SAMP/RAMP-Hydrazone
Methodology.
402) D. Enders, A. Lenzen, G. Raabe, Angew. Chem. 2005, 117, 3832 – 3835; Angew.
Chem. Int. Ed. 2005, 44, 3766 - 3769. Asymmetrische Synthese des Grundgerüsts
der Cripowelline A und B – das 1-epi-Aglycon.
403) D. Enders, C. Grondal, M. Vrettou, G. Raabe, Angew. Chem. 2005, 117, 4147 –
4151; Angew. Chem. Int. Ed. 2005, 44, 4079 - 4083. Asymmetrische Synthese von
selektiv geschützten Aminozucker-Derivaten via direkte organokatalytische
Mannich-Reaktion.
404) D. Enders, J.-C. Adelbrecht, W. Harnying, Synthesis 2005, 2962 - 2968.
Asymmetric Synthesis of α- and α,β-Substituted β-Alkoxycarbonyl Sulfonates.
405) D. Enders, I. Breuer, G. Raabe, Synthesis 2005, 3517 - 3530. Asymmetric
Synthesis of 2-Keto-1,3-diols and Protected 1,2,3-Triols Bearing Two Quaternary
Stereocenters.
406) D. Enders, J. Gries, Synthesis 2005, 3508 - 3516. Asymmetric Synthesis of
Substituted Azetidine Type α- and β-Amino Acids.
407) D. Enders, A. Lenzen, M. Backes, C. Janeck, K. Catlin, M.-I. Lannou, J. Runsink,
G. Raabe, J. Org. Chem. 2005, 70, 10538 - 10551. Asymmetric Total Synthesis of
the 1-epi-Aglycon of the Cripowellins A and B.
39
408) D. Enders, A. Hieronymi, A. Ridder, Synlett 2005, 2391 - 2393. Asymmetric
Synthesis of 4’-Quaternary 2’-Deoxy-3’-epi-β-C-Nucleosides.
409) M. Boudou, D. Enders, J. Org. Chem. 2005, 70, 9486 - 9494. Asymmetric Synthesis
of Tetrahydropalmatine via Tandem 1,2-Addition/Cyclisation.
410) D. Enders, O. Niemeier, Heterocycles 2005, 66, 385 - 403. Asymmetric Synthesis of
β-Substituted γ-Lactams Employing the SAMP-/RAMP-Hydrazone Methodology.
Application to the Synthesis of (R)-(–)-Baclofen.
411) D. Enders, I. Breuer, E. Drosdow, Synthesis 2005, 3239 - 3244. Asymmetric
Synthesis of 4’-epi-Trachycladines A and B.
412) D. Enders, S. Noll, J. W. Bats, Synlett 2005, 2679 - 2681. Efficient Entry to
Diastereo- and Enantiomerically Pure α-Branched [2.2]Paracyclophanyl-
alkylamines.
413) D. Enders, A. Saint-Dizier, M. I. Lannou, A. Lenzen, Eur. J. Org. Chem. 2006, 29 -
49. The Phospha-Michael Addition in Organic Synthesis.
414) C. Grondal. D. Enders, Tetrahedron 2006, 62, 329 - 337. Direct Asymmetric
Organocatalytic de novo Synthesis of Carbohydrates.
415) D. Enders, W. Bettray in Asymmetric Synthesis – The Essentials, S. Bräse, M.
Christmann, Eds., Wiley-VCH, Weinheim, 2006, 21 - 26. Asymmetric Syntheses
with SAMP-/RAMP-Hydrazones.
416) D. Enders, A. Moll, J. W. Bats, Eur. J. Org. Chem. 2006, 1271 - 1284. Asymmetric
Synthesis of 3-Substituted γ- and δ-Sultams.
417) D. Enders, J. Pale�ek, C. Grondal, Chem. Commun. 2006, 655 - 657. A Direct
Organocatalytic Entry to Sphingoids: Asymmetric Synthesis of D-arabino- and L-
ribo-Phytosphingosine.
418) D. Enders, O. Niemeier, T. Balensiefer, Angew. Chem. 2006, 118, 1491 - 1495;
Angew. Chem. Int. Ed. 2006, 45, 1463 – 1467. Asymmetric Intramolecular
Crossed-Benzoin Reactions by N-Heterocyclic Carbene Catalysis.
419) D. Enders, L. Tedeschi, D. Förster, Synthesis 2006, 1447 - 1460. Asymmetric
Michael Additions of a Chiral Phosphite to Nitroalkenes and Knoevenagel
Acceptors.
40
420) B. Karimi, D. Enders, Org. Lett. 2006, 8, 1237 - 1240. A New N-Heterocyclic
Carbene Palladium Complex/Ionic Liquid Matrix Immobilized on Silica:
Application as Recoverable Catalyst for the Heck Reaction.
421) D. Enders, M. R. M. Hüttl, C. Grondal, G. Raabe, Nature 2006, 441, 861 - 863.
Control of Four Stereocentres in a Triple Cascade Organocatalytic Reaction.
422) D. Enders, M. Vrettou, Synthesis 2006, 2155 - 2158. Asymmetric Synthesis of (+)-
Polyoxamic Acid via an Efficient Organocatalytic Mannich Reaction as the Key
Step.
423) D. Enders, O. Niemeier, G. Raabe, Synlett 2006, 2431 - 2434. Asymmetric
Synthesis of Chromanones via N-Heterocyclic Carbene Catalyzed Intramolecular
Crossed-Benzoin Reactions.
424) D. Enders, C. Grondal, M. Vrettou, Synthesis 2006, 3597 - 3604. Efficient Entry to
Amino Sugars and Derivatives via Asymmetric Organocatalytic Mannich
Reactions.
425) D. Enders, S. Chow, Eur. J. Org. Chem. 2006, 4578 - 4584. Organocatalytic
Asymmetric Michael Addition of 2,2-Dimethyl-1,3-dioxan-5-one to Nitroalkenes
Employing Proline-based Catalysts.
426) C. Grondal, D. Enders, Synlett 2006, 3507-3509. A Direct Entry to Carbasugars.
Asymmetric Synthesis of 1-epi-(+)-MK7607.
427) D. Enders, O. Niemeier, L. Straver, Synlett 2006, 3399-3402. Asymmetric Organo-
catalytic Synthesis of cis-Substituted Dihydrobenzofuranols via Intramolecular
Aldol Reactions.
428) K. Funabiki, M. Nagamori, M. Matsui, G. Raabe, D. Enders in Current
Fluoroorganic Chemistry. New Synthetic Directions, Technologies, Materials and
Biological Applications. ACS Symposium Series Book 949, T. Yamazaki, J. T.
Welch, J. F. Honak, Eds., 2006, 447 - 461. Asymmetric Synthesis of β-
Trifluoromethylated β-Amino Carbonyl Compounds Based on the 1,2-Addition to
Trifluoroacetaldehyde SAMP/RAMP-Hydrazone.
429) D. Enders, T. Balensiefer, O. Niemeier, M. Christmann in Enantioselective
Organocatalysis. Reactions and Experimental Procedures, P. I. Dalko, Ed., Wiley-
VCH, Weinheim, 2007, 331 - 355. Nucleophilic N-Heterocyclic Carbenes in Asym-
metric Organocatalysis.
41
430) D. Enders, M. Milovanovi�, Z. Naturforsch. 2007, 62b, 117 - 120. Asymmetric
Synthesis of (+)-Hinokinin, (+)-Dihydrocubebin and Cubebin Dimethyl Ether, a
New Lignan from Phyllantis niruri.
431) D. Enders, M. R. M. Hüttl, J. Runsink, G. Raabe, B. Wendt, Angew. Chem. 2007,
119, 471 - 473; Angew. Chem. Int. Ed. 2007, 46, 467-469. Organocatalytic One Pot
Asymmetric Synthesis of Functionalized Tricyclic Carbon Skeletons via a Triple
Cascade/Diels-Alder Sequence.
432) D. Enders, T. Gasperi, Chem. Commun. 2007, 88-90. Proline Organocatalysis as a
New Tool for the Asymmetric Synthesis of Ulosonic Acid Precursors.
433) D. Enders, C. Grondal, M. R. M. Hüttl, Angew. Chem. 2007, 119, 1590 - 1601;
Angew. Chem. Int. Ed. 2007, 46, 1570 - 1581. Asymmetric Organocatalytic Domino
Reactions.
434) D. Enders, C. Herriger, Eur. J. Org. Chem. 2007, 1085 - 1090. Asymmetric
Synthesis of 2-Trifluoromethyl-1,2,3-triols.
435) C. Grondal, D. Enders, Adv. Synth. Catal. 2007, 349, 694 - 702. A Direct
Organocatalytic Entry to Selectively Protected Aldopentoses and Derivatives.
436) D. Enders, S. Dhulut, D. Steinbusch, A. Herrbach, Chem. Eur. J. 2007, 13, 3942 -
3949. Asymmetric Total Synthesis of (–)-Pironetin Employing the SAMP/RAMP
Hydrazone Methodology.
437) D. Enders, M. H. Bonten, G. Raabe, Angew. Chem. 2007, 119, 2364 - 2367; Angew.
Chem. Int. Ed. 2007, 46, 2314 - 2216. Asymmetric Nucleophilic Gloyxylation via a
Metalated α-Aminonitrile Derivative in Michael Additions to Nitroalkenes.
438) D. Enders, W. Bettray in Asymmetric Synthesis with Chemical and Biological
Methods, D. Enders, K.-E. Jaeger, Eds., Wiley-VCH, Weinheim, 2007, p. 1 - 37.
Development of Novel Enantioselective Synthetic Methods.
439) D. Enders, W. Bettray in Asymmetric Synthesis with Chemical and Biological
Methods, D. Enders, K.-E. Jaeger, Eds., Wiley-VCH, Weinheim, 2007, p. 38 - 75.
Asymmetric Synthesis of Natural Products Employing the SAMP/RAMP-
Hydrazone Methodology.
440) M. Albrecht, S. Mirtschin, O. Osetska, S. Dehn, D. Enders, R. Fröhlich, T. Pape, E.
F. Hahn, Eur. J. Inorg. Chem. 2007, 3276 - 3287. Pentadentate Ligands for the 1:1
Coordination of Lanthanide(III) Salts.
42
441) D. Enders, M. H. Bonten, G. Raabe, Synlett 2007, 885 - 888. Organocatalytic
Asymmetric Conjugate Nucleophilic Glyoxylation.
442) D. Enders, E. Peiffer, G. Raabe, Synthesis 2007, 1021 - 1026. Asymmetric
Synthesis of (S, S)- and (R, R)-2-Methylthreitol.
443) D. Enders, K. Lüttgen, A. A. Narine, Synthesis 2007, 959 - 980. Asymmetric Sulfa-
Michael Additions.
444) D. Enders, O. Niemeier, A. Henseler, Chem. Rev. 2007, 107, 5606 - 5655.
Organocatalysis by N-Heterocyclic Carbenes.
445) D. Enders, A. A. Narine, T. R. Benninghaus, G. Raabe, Synlett 2007, 1667 - 1670.
Asymmetric Organocatalytic Domino Reactions of γ-Nitroketones and Enals.
446) D. Enders, D. Iffland, Synthesis 2007, 1837 - 1840. Asymmetric Synthesis of α-
Phenyl-γ-Hetero-Substituted Isopropyl Sulfonates via Diastereoselective Ring-
Opening of γ-Sultones.
447) W. Harnying, W. Kitisriworaphan, M. Pohmakotr, D. Enders, Synlett 2007, 2529 -
2532. Stereoselective Aldol Reactions: Asymmetric Synthesis of α,β-Substituted β-
Hydroxy Sulfonates.
448) R. Brehme, D. Enders, R. Fernandez, J. M. Lassaletta, Eur. J. Org. Chem. 2007,
5629 - 5660. Aldehyde N,N-Dialkylhydrazones as Neutral Acyl Anion Equivalents.
Umpolung of the Imine Reactivity.
449) D. Enders, M. R. M. Hüttl. G. Raabe, J. W. Bats, Adv. Synth. Catal. 2008, 350, 267
- 279. Asymmetric Synthesis of Polyfunctionalized Mono-, Bi-, and Tricyclic
Carbon Frameworks via Organocatalytic Domino Reactions.
450) D. Enders, J. Barbion, Chem. Eur. J. 2008, 14, 2842 - 2849. Asymmetric Synthesis
of (+)-Altholactone, a Styryllactone Isolated from Various Goniothalamus Species.
451) D. Enders, M. R. M. Hüttl, O. Niemeier, Ernst Schering Foundation Symposium
Proceedings: Organocatalysis, M. T. Reetz, B. List, S. Jaroch, H. Weinmann (Eds.),
Springer-Verlag, Berlin, 2008, 45 - 124. Biomimetic Organocatalytic C-C-Bond
Formations.
452) N. Gassler, A. Reinartz, E. Kämmerer, D. Enders, W. Bettray, Nutrition for the
Middle-Aged and Elderly, N. E. Bernhardt, A. M. Kasko, Eds., Nova Science
Publishers, Hauppauge, 2008, 447 - 458. The Role of Dietary Fatty Acids and Acyl-
CoA Synthetases in the Development of Colorectal Cancer.
43
453) D. Enders, S. Noll, G. Raabe, J. Runsink, Synthesis 2008, 1288 - 1296. Synthesis of
All Possible Stereoisomers of α-Branched [2.2]Paracyclophanyl-alkylamines.
454) D. Enders, A. Hieronymi, G. Raabe, Synthesis 2008, 1545 - 1558. Asymmetric
Synthesis of 4’-Quaternary 2’-Deoxy-3’- and 4’-epi-β-C- and N- Nucleosides.
455) D. Enders, V. Terteryan, J. Pale�ek, Synthesis 2008, 2278 - 2282. Asymmetric
Synthesis of Jaspine B (Pachastrissamine) via an Organocatalytic Aldol Reaction
as Key Step.
456) D. Enders, A. A. Narine, F. Toulgoat, T. Bisschops, Angew. Chem. 2008, 120, 5744
- 5748. Angew. Chem. Int. Ed. 2008, 47, 5661-5665. Asymmetric Brønsted Acid-
Catalyzed Isoindoline Synthesis: Enhancement of Enantiomeric Ratio by
Stereoablative Kinetic Resolution.
457) D. Enders, J. Han, Tetrahedron: Asymmetry 2008, 19, 1367 - 1371. Synthesis of
Enantiopure Triazolium Salts from Pyroglutamic Acid and Their Evaluation in the
Benzoin Condensation.
458) D. Enders, C. Wang, J. W. Bats, Angew. Chem. 2008, 120, 7649 - 7653; Angew.
Chem. Int. Ed. 2008, 47, 7539 - 7542. Organocatalytic Asymmetric Domino
Reactions: A Cascade Consisting of a Michael Addition and an Aldehyde α-
Alkylation.
459) D. Enders, J. Han, A. Henseler, Chem. Commun. 2008, 3989 - 3991. Asymmetric
Intermolecular Stetter Reactions Catalyzed by a Novel Triazolium Derived N-
Heterocyclic Carbene.
460) D. Enders, A. A. Narine, J. Org. Chem. 2008, 73, 7857 - 7870. Lessons from
Nature: Biomimetic Organocatalytic Carbon-Carbon Bond Formations.
461) D. Enders, D. Förster, G. Raabe, J. W. Bats, J. Org. Chem. 2008, 73, 9641 - 9646.
Asymmetric Synthesis of β-Nitroketones via Michael Addition of Lithiated α-
Amino Nitriles to Nitroalkenes.
462) D. Enders, J. Han, Synthesis 2008, 3864 - 3868. Asymmetric Intermolecular
Stetter Reactions of Aromatic Heterocyclic Aldehydes with Arylidenemalonates.
463) D. Enders, K. Hoffman, Eur. J. Org. Chem. 2009, 1665 - 1668. Organocatalytic
Asymmetric Sulfa-Michael Additions to �,�-Unsaturated Sulfonates.
464) D. Enders, E. A. Jonas, T. Klumpen, Eur. J. Org. Chem. 2009, 2149 - 2162.
Efficient Asymmetric Synthesis of Planar-Chiral Bisferrocenes.
44
465) D. Enders, D. Iffland, G. Raabe, Synthesis 2009, 1683 - 1688. Asymmetric
Synthesis of 1,2-anti-Disubstituted Taurine Derivatives.
466) D. Enders, C. Wang, J. W. Bats, Synlett 2009, 1777 - 1780. Asymmetric Synthesis
of Functionalized 3,4-Dihydronaphthalenes via an Organocatalytic Domino
Nitroalkane-Michael/Aldol Condensation Reaction.
467) D. Enders, A. Henseler, Adv. Synth. Catal. 2009, 351, 1749 - 1752. A Direct
Intermolecular Cross-Benzoin Type Reaction: N-Heterocyclic Carbene Catalyzed
Coupling of Aromatic Aldehydes with Trifluoromethyl Ketones.
468) D. Enders, C. Wang, G. Raabe, Synthesis 2009, 4119 - 4124. Enantioselective
Synthesis of 3H-Pyrrolo[1,2-a]indole-2-carbaldehydes via an Organocatalytic
Domino aza-Michael/Aldol Condensation Reaction.
469) D. Enders, H. Saeidian, Z. Mirjafary, D. Iffland, G. Raabe, J. Runsink, Synlett
2009, 2872 - 2874. Diastereo- and Enantioselective Synthesis of α,β-Disubstituted
γ- Bisalkoxycarbonyl Sulfonates.
470) D. Enders, C. Wang, J. X. Liebich, Chem. Eur. J. 2009, 15, 11058 - 11076.
Organocatalytic Asymmetric Aza-Michael Additions.
471) D. Enders, A. Henseler, S. Lowins, Synthesis 2009, 4125 - 4128. N-Heterocyclic
Carbene-catalyzed Nucleophilic Acylation of Trifluoromethyl Ketimines.
472) D. Enders, M. Mirjafary, H. Saeidian, Tetrahedron: Asymmetry 2009, 20, 2429 -
2431. Efficient Diastereo- and Enantioselective Synthesis of α,β-Disubstituted γ-
Phosphono Sulfonates.
473) D. Enders, M. Jeanty, J. W. Bats, Synlett 2009, 3175 - 3178. Organocatalytic
Asymmetric Triple Domino Reactions of Nitromethane with α,β-Unsaturated
Aldehydes.
474) D. Enders, R. Krüll, W. Bettray, Synthesis 2010, 567 - 572. Microwave Assisted
Organocatalytic Quadruple Domino Reactions of Acetaldehyde and Nitroalkenes.
475) C. Grondal, M. Jeanty, D. Enders, Nature Chemistry 2010, 2, 167 - 178.
Organocatalytic Cascade Reactions as a New Tool in Total Synthesis.
476) D. Enders, C. Wang, A. Greb, Adv. Synth. Catal. 2010, 352, 987 - 992. Asymmetric
Synthesis of 2,3,4-Trisubstituted Functionalized Tetrahydrofurans via an
Organocatalytic Michael Addition as Key Step.
45
477) D. Enders, C. Wang, M. Mukanova, A. Greb, Chem. Commun. 2010, 46, 2447 -
2449. Organocatalytic Asymmetric Synthesis of Polyfunctionalized 3-
(Cyclohexenyl-methyl)-indoles via a Quadruple Domino Friedel-Crafts-type /
Michael/Michael/ Aldol Condensation Reaction.
478) D. Enders, M. Seppelt, T. Beck, Adv. Synth. Catal. 2010, 352, 1413 - 1418.
Enantioselective Organocatalytc Synthesis of Arylglycines via Friedel-Crafts
Alkylation of Arenes with a Glyoxylate Imine.
479) D. Enders, B. Schmid, N. Erdmann, G. Raabe, Synthesis 2010, 2271 - 2277.
Asymmetric Synthesis of Thiadecalines via an Organocatalytic Triple
Cascade/Sulfa-Michael Sequence.
480) D. Enders, V. Terteryan, J. Pale�ek, Synthesis 2010, 2979 - 2984. Asymmetric
Synthesis of the α-D-Galactosyl Ceramide KRN7000 via an Organocatalytic Aldol
Reaction as Key Step.
481) D. Enders, J. X. Liebich, G. Raabe, Chem. Eur. J. 2010, 16, 9763 - 9766.
Organocatalytic Asymmetric Synthesis of trans-1,3-Disubstituted
Tetrahydroisoquinolines via a Reductive Amination / Aza-Michael Sequence.
482) D. Enders, A. Grossmann, J. Fronert, G. Raabe, Chem. Commun. 2010, 46, 6282 -
6284. N-Heterocyclic Carbene Catalysed Asymmetric Cross-Benzoin Reactions of
Heteroaromatic Aldehydes with Trifluoromethyl Ketones.
483) D. Enders, C. Wang, X. Yang, G. Raabe, Adv. Synth. Catal. 2010, 352, 2869 - 2874.
Asymmetric Synthesis of cis-3,4-Disubstituted Chromans and Dihydrocoumarins
via an Organocatalytic Michael/Hemiacetalization Reaction.
484) D. Enders, D. P. Göddertz, C. Beceño, G. Raabe, Adv. Synth. Catal. 2010, 352,
2863 - 2868. Asymmetric Synthesis of Polyfunctionalized Pyrrolidines via a
Thiourea Catalyzed Domino Mannich/Aza-Michael Reaction.
485) D. Enders, K. Gottfried, G. Raabe, Adv. Synth. Catal. 2010, 352, 3147 - 3152.
Organocatalytic Enantioselective Strecker-Synthesis of α-Quaternary α-
Trifluoromethyl Amino Acids.
486) M. W. Alachraf, P. P. Handayani, M. R. M. Hüttl, C. Grondal, D. Enders, W.
Schrader, Org. Biomol. Chem. 2011, 9, 1047 - 1053. Electrospray Mass
Spectrometry for Detailed Mechanistic Studies of a Complex Organocatalyzed
Triple Cascade Reaction.
46
487) D. Enders, C. Wang, X. Yang, G. Raabe, Synlett 2011, 469 - 472. One Pot
Organocatalytic Asymmetric Synthesis of 1H-Pyrrolo[1.2a]indol-3(2H)-ones via a
Michael/Hemiaminalization/Oxidation Sequence.
488) D. Enders, J. X. Liebich, A. Rembiak, Synthesis 2011, 281 - 286. Direct
Organocatalytic α-Sulfenylation of Aldehydes and Ketones with
Tetramethylthiuram Disulfide.
489) D. Enders, S. Mangelinckx in Electronic Encyclopedia of Reagents for Organic
Synthesis, P. L. Fuchs, Ed. Wiley, Chichester, 2011. Dimethylthexylsilyl
Trifluoromethanesulfonate.
490) D. Enders, M. Seppelt, Synlett 2011, 402 - 404. Catalytic Enantioselective
Synthesis of 3-Substituted Benzosultams via Corey-Bakshi-Shibata Reduction of
Cyclic N-Sulfonylimines.
491) D. Enders, G. Urbanietz, G. Raabe, Synthesis 2011, 1905 - 1911. Organocatalytic
Asymmetric Synthesis of Functionalized 4H-Chromenes via a One Pot Domino
Michael-Hemiacetalization and Dehydration Sequence.
492) D. Enders, X. Yang, C. Wang, G. Raabe, J. Runsink, Chem. Asian J. 2011, 6, 2255-
2259. Dienamine Activation in the Organocatalytic Asymmetric Synthesis of cis-
3,4-Difunctionalized Chromans and Dihydrocoumarins.
493) D. Enders, A. Grossmann, H. Huang, G. Raabe, Eur. J. Org. Chem. 2011, 4298 -
4301. Dual Secondary Amine/N-Heterocyclic Carbene Catalysis in the Asymmetric
Michael − Cross-Benzoin Cascade Reaction of ß-Ketosulfones with Enals.
494) C. C. J. Loh, J. Badorrek, G. Raabe, D. Enders, Chem. Eur. J. 2011, 17, 13409 -
13414. Merging Organocatalysis and Gold Catalysis: Enantioselective Synthesis of
Tetracyclic Indole Derivatives Through a Sequential Double Friedel-Crafts-Type
Reaction.
495) C. C. J. Loh, D. Enders, Angew. Chem. 2012, 124, 46 - 49; Angew. Chem. Int. Ed.
2012, 51, 46 - 48. Exploiting the Electrophilic Properties of Indole Intermediates –
New Options in Asymmetric Reaction Design.
496) D. Enders, M. Ludwig, G. Raabe, Chirality 2012, 24, 215 - 222. Synthesis and
Application of the First Planar-Chiral Strong Brønsted Acid Organocatalysts.
497) A. Grossmann, D. Enders, Angew. Chem. 2012, 124, 320 - 332; Angew. Chem. Int.
Ed. 2012, 51, 314 - 325. N-Heterocyclic Carbene Catalyzed Domino Reactions.
47
498) D. Enders, G. Urbanietz, R. Hahn, G. Raabe, Synthesis 2012, 44, 773 - 782.
Asymmetric Synthesis of Functionalized Chromans via a One Pot Organocatalytic
Domino Michael-Hemiacetalization or Lactonization and Dehydration Sequence.
499) D. Enders, T. V. Nguyen, Tetrahedron Lett. 2012, 53, 2091 - 2095. Secondary
Amine Catalyzed Retro-Aldol Reactions of Enals and Enones: One-Pot Conversion
of Enals to α-Substituted Derivatives.
500) C. Wang, X. Yang, D. Enders, Chem. Eur. J. 2012, 18, 4832 - 4835. Asymmetric
Michael Addition of N-Boc-Protected Oxindindols to Nitroalkenes Catalyzed by a
Chiral Secondary Amine.
501) D. Enders, G. Urbanietz, E. Cassens-Sasse, S. Keeß, G. Raabe, Adv. Synth. Catal.
2012, 354, 1481 - 1488. Control of Six Contiguous Stereocenters in an Asymmetric
Organocatalytic One-Pot Michael/Michael/Aldol Addition Sequence.
502) C. C. J. Loh, D. Enders, Chem. Eur. J. 2012, 18, 10212 - 10225. Merging
Organocatalysis and Gold Catalysis – A Critical Evaluation of the Underlying
Concepts.
503) S. Takizawa, T. M.-N. Nguyen, A. Grossmann, D. Enders, H. Sasai, Angew. Chem.
2012, 124, 5519 - 5522; Angew. Chem. Int. Ed. 2012, 51, 5423 - 5426.
Enantioselective Synthesis of α-Alkylidene-γ-butyrolactones via Intramolecular
Rauhut-Currier Reaction Promoted by Acid-Base Organocatalysts.
504) D. Enders, S. Breukers, L. F. Reichenbach in Electronic Encyclopedia of Reagents
for Organic Synthesis, T. Rovis, Ed. Wiley, Chichester, 2012. 2,2-Dimethyl-1,3-
dioxan-5-one.
505) D. Enders, A. Greb, K. Deckers, P. Selig, C. Merkens, Chem. Eur. J. 2012, 18,
10226 - 10229. Quadruple Domino Organocatalysis: An Asymmetric aza-
Michael/Michael/Michael/Aldol Reaction Sequence Leading to Tetracyclic Indole
Structures with Six Stereocenters.
506) C. Wang, X. Yang, C. C. J. Loh, G. Raabe, D. Enders, Chem. Eur. J. 2012, 18,
11531 - 11535. Organocatalytic Asymmetric Synthesis of 3-Sulfenylated N-BOC-
Protected Oxindoles.
507) D. Enders, J. Fronert, T. Bisschops, F. Boeck, Beilstein J. Org. Chem. 2012, 8,
1112 - 1117. Asymmetric Total Synthesis of Smyrindiol Employing an
Organocatalytic Aldol Key Step.
48
508) N. Erdmann, I. Atodiresei, D. Enders, Synthesis 2012, 44, 2107 - 2113.
Asymmetric Synthesis of 3-Substituted Hexahydro-3H-Isochromenes via an
Organocatalytic Triple Cascade/Yb-Catalyzed Hetero-Diels-Alder Sequence.
509) V. Nguyen, D. Enders, Org. Biomol. Chem. 2012, 10, 5327 - 5331. Chiral
Quaternary Phosphonium Salts: A New Class of Organocatalysts.
510) X. Yang, C. Wang, Q. Ni, D. Enders, Synthesis 2012, 44, 2601 - 2606. Secondary
Amine-Catalyzed Asymmetric Michael Addition of N-tert-Butoxycarbonyl-
Protected Oxindoles to Maleimides.
511) C. Wang, X. Yang, G. Raabe, D. Enders, Adv. Synth. Catal. 2012, 354, 2629 - 2634.
A Short Asymmetric Synthesis of the Benzopyrano[3,4-c]pyrrolidine Core via an
Organocatalytic Domino oxa-Michael/Michael Reaction.
512) D. Enders, A. Grossmann, B. Gieraths, M. Düzdemir, C. Merkens, Org. Lett. 2012,
14, 4254 - 4257. Organocatalytic One Pot Asymmetric Synthesis of 4H,5H-
Pyrano[2,3-c]pyrazoles.
513) C. C. J. Loh, G. Raabe, D. Enders, Chem. Eur. J. 2012, 18, 13250- 13254.
Enantioselective Synthesis of Tetrahydrocarbazoles Through a Michael Addition /
Ciamician-Plancher Rearrangement Sequence. Asymmetric Synthesis of a Potent
Constrained Analog of MS-245.
514) J.-P. Wan, C. C. J. Loh, F. Pan, D. Enders, Chem. Commun. 2012, 48, 10049 -
10051. Enantioselective Organocatalytic Domino Synthesis of Tetrahydropyridin-
2-ols.
515) D. Enders, S. David, K. Deckers, A. Greb, G. Raabe, Synthesis 2012, 44, 3483 -
3488. Asymmetric Synthesis of Gonioheptolide A Analogues via an Organocatalytic
Aldol Reaction as the Key Step.
516) D. Enders, A. Grossmann, D. Van Craen, Org. Biomol. Chem. 2013, 11, 138 - 141.
N-Heterocyclic Carbene Catalyzed Synthesis of Oxime Esters.
517) D. Enders, A. Rembiak, M. Seppelt, Tetrahedron Lett. 2013, 54, 470 - 473.
Asymmetric Organocatalytic Reduction of Ketimines with Catecholborane
Employing an N-Triflyl Phosphoramide Brønsted Acid as Catalyst.
49
518) S. Takizawa, T. M.-N. Nguyen, A. Grossmann, M. Suzuki, D. Enders, H. Sasai,
Tetrahedron 2013, 69, 1202 - 1209. Facile Synthesis of α-Alkylidene-γ-
butyrolactones: Intramolecular Rauhut-Currier Reaction Promoted by Chiral Acid-
Base Organocatalysts.
519) T. V. Nguyen, J. Hartmann, D. Enders, Synthesis 2013, 45, 845 - 873. Recent
Synthetic Strategies to Access Seven-Membered Carbocycles in Natural Product
Synthesis.
520) S. Ansari, G. Raabe, D. Enders, Monatsh. Chem. 2013, 144, 641 - 646. Asymmetric
Michael Addition of 1,3-Bis(phenylthio)propan-2-one to Nitroalkenes Employing
Takemoto’s Thiourea Catalyst.
521) X. Zeng, Q. Ni, G. Raabe, D. Enders, Angew. Chem. 2013, 125, 3050 – 3054;
Angew. Chem. Int. Ed. 2013, 52, 2977 - 2980. A Branched Domino Reaction: Two
Component Quadruple Organocatalytic Asymmetric Synthesis of
Polyfunctionalized Cyclohexene Derivatives.
522) N. Erdmann, A. R. Philipps, I. Atodiresei, D. Enders, Adv. Synth. Catal. 2013, 355,
847 - 857. An Asymmetric Organocatalytic Quadruple Cascade Initiated by a
Friedel-Crafts-Type Reaction with Electron-Rich Arenes.
523) D. Enders, R. Hahn, I. Atodiresei, Adv. Synth. Catal. 2013, 355, 1126 - 1136.
Asymmetric Synthesis of Functionalized Tetrahydronaphthalenes via an
Organocatalytic Nitroalkane-Michael/Henry Domino Reaction.
524) B. Karimi, E. Jafari, D. Enders, Chem. Eur. J. 2013, 19, 10142 - 10145. Highly
Efficient Catalytic Enantioselective Mannich Reaction of Malonates with N-tert-
Butoxycarbonyl Imines by Using Yb(OTf)3/Pybox Catalysts at Room Temperature.
525) D. Enders, L. F. Reichenbach, Synthesis 2013, 45, 959 - 965. Asymmetric
Synthesis of Synargentolide A and Its 3-Epimer Using the RAMP-Hydrazone
Methodology.
526) D. Enders, G. Del Signore, G. Raabe, Turk. J. Chem. 2013, 37, 492 - 518.
Asymmetric Synthesis of �-(Heteroaryl)alkylamines and �-Amino Acids via
Nucleophilic 1,2-Addition of Lithiated Heterocycles to Aldehyde SAMP-
Hydrazones.
527) B. Karimi, D. Enders, E. Jafari, Synthesis 2013, 45, 2769 - 2812. Recent Advances
in Metal-Catalyzed Asymmetric Mannich Reactions.
50
528) C. C. J. Loh, I. Atodiresei, D. Enders, Chem. Eur. J. 2013, 19, 10822 - 10826.
Asymmetric Organocatalytic Michael/Henry Domino Reactions through Hydrogen
Bonding Activation: A Kinetic Access into Indane Scaffolds Bearing cis-Vicinal
Substituents.
529) J. Fronert, T. Bisschops, E. Cassens-Sasse, I. Atodiresei, D.Enders, Synthesis
2013, 45, 1708 - 1712. Asymmetric Organocatalytic Synthesis of trans-3,4-
Disubstituted Isochromanones via an Intramolecular Aldol Reaction.
530) D. Enders, A. Rembiak, B. A. Stöckel, Adv. Synth. Catal. 2013, 355, 1937 - 1942.
Chemo- and Enantioselective Brønsted Acid Catalyzed Reduction of α-Imino
Esters with Catecholborane.
531) D. Enders, C. Joie, K. Deckers, Chem. Eur. J. 2013, 19, 10818 - 10821.
Organocatalytic Asymmetric Synthesis of Tetracyclic Pyridocarbazole Derivatives
by Using a Diels-Alder/aza-Michael/Aldol Condensation Domino Reaction.
532) Q. Ni, H. Zhang, A. Grossmann, C. C. J. Loh, C. Merkens, D. Enders, Angew.
Chem. 2013, 125, 13806 – 13811; Angew. Chem. Int. Ed. 2013, 52, 13562 - 13566.
Asymmetric Synthesis of Pyrroloindolones via N-Heterocyclic Carbene Catalyzed
[2+3] Annulation of α-Chloroaldehydes with Nitrovinylindoles.
533) D. Hack, D. Enders, Synthesis 2013, 45, 2904 - 2912. Asymmetric Organocatalytic
Michael Addition of Pyrroles to Enones Catalyzed by Cinchona Alkaloid-Derived
Primary Amines.
534) X. Song, Q. Ni, A. Grossmann, D. Enders, Chem. Asian J. 2013, 8, 2965 - 2969. N-
Heterocyclic Carbene Catalyzed One-Pot Synthesis of Hydroxamic Esters.
535) C. C. J. Loh, D. Hack, D. Enders, Chem. Comm. 2013, 49, 10230 - 10232.
Asymmetric Domino Synthesis of Indanes Bearing Four Contiguous Stereocentres
Catalyzed by Sub-mol% Loadings of a Squaramide in Minutes.
536) P. Chauhan, D. Enders, Angew. Chem. 2014, 126, 1509 – 1511; Angew. Chem. Int.
Ed. 2014, 53, 1485 - 1487. N-Heterocyclic Carbene Catalyzed Activation of Esters:
A New Option for Asymmetric Domino Reactions.
537) C. Joie, K. Deckers, D. Enders, Synthesis 2014, 46, 799 - 808. Organocatalytic
Asymmetric Synthesis of Functionalized 1,3,5-Triaryl 2-Pyrrolidinones via an aza-
Michael/Aldol Domino Reaction.
51
538) S. Takizawa, J. Kodera, Y. Yoshida, M. Sako, S. Breukers, D. Enders, H. Sasai,
Tetrahedron 2014, 70, 1786 - 1793. Enantioselective Oxidative Coupling of
Polycyclic Phenols.
539) G. Urbanietz, I. Atodiresei, D. Enders, Synthesis 2014, 46, 1261 - 1269.
Asymmetric Synthesis of Functionalized Dihydro- and Tetrahydropyrans via an
Organocatalytic Domino Michael-Hemiacetalization Reaction.
540) D. Enders, B. Stöckel, A. Rembiak, Chem. Commun. 2014, 50, 4489 - 4491.
Enantio- and Chemoselective Brønsted-Acid/Mg(nBu)2 Catalysed Reduction of α-
Ketoesters with Catecholborane.
541) D. Hack, C. C. J. Loh, J. M. Hartmann, G.Raabe, D. Enders, Chem. Eur. J. 2014,
20, 3917 - 3921. Merging Gold and Organocatalysis: A Facile Asymmetric
Synthesis of Annulated Pyrroles.
542) H. Saeidian, D. Enders, Z. Mirjafary, Iran. Chem. Commun. 2014, 2, 137 - 146.
The SAMP-/RAMP-Hydrazone Methodology in Asymmetric Synthesis of 4S-
Ferrugineone and 4S,5S-Ferrugineol: The Pheromones of Palm Weevils.
543) C. Joie, K. Deckers., G. Raabe, D. Enders, Synthesis 2014, 46, 1539 - 1546. An
Asymmetric Organocatalytic Quadruple Cascade to Tetraaryl-Substituted 2-
Azabicyclo[3.3.0]octadienones.
544) Q. Ni, X. Song, G. Raabe, D. Enders, Chem. Asian J. 2014, 9, 1535 - 1538. N-
Heterocyclic Carbene-Catalyzed Enantioselective Annulation of Indolin-3-ones
with Bromoenals.
545) P. Chauhan, G. Urbanietz, G. Raabe, D. Enders, Chem. Commun. 2014, 50, 6853 -
6855. Asymmetric Synthesis of Functionalised Cyclohexanes Bearing Five
Stereocenters via a One-Pot Organocatalytic Michael/Michael/1,2-Addition
Sequence.
546) P. Chauhan, S. Mahajan, C. C. J. Loh, G. Raabe, D. Enders, Org. Lett. 2014, 16,
2954 - 2957. Stereocontrolled Construction of Six Vicinal Stereogenic Centers on
Spiropyrazolones via Organocascade Michael/Michael/1,2-Addition Reactions.
547) C. C. Loh, P. Chauhan, D. Hack, C. Lehmann, D. Enders, Adv. Synth. Catal. 2014,
356, 3181 - 3186. Rapid Asymmetric Synthesis of Highly Functionalized Indanols
via a Michael/Henry Organocascade with Sub-mol% Squaramide Catalyst
Loadings.
52
548) P. Chauhan, S. Mahajan, D. Enders, Chem. Rev. 2014, 114, 8807 - 8864.
Organocatalytic Carbon-Sulfur Bond Forming Reactions.
549) R. Hahn, G. Raabe, D. Enders, Org. Lett. 2014, 16, 3636 - 3639. Asymmetric Syn-
thesis of Highly Functionalized Tetrahydropyrans via a One-Pot Organocatalytic
Michael/Henry/Ketalization Sequence.
550) B. Karimi, E. Jafari, D. Enders, Eur. J. Org. Chem. 2014, 7253 - 7258. Asymmetric
Mannich Reaction of Malonates with Aldimines Using YbIII-Pybox Complexes
Supported on Self-Assembled Organic-Inorganic Hybrid Silica with an
Imidazolium Framework.
551) D. Hack, P. Chauhan, K. Deckers, G. N. Hermann, L. Mertens, G. Raabe, D.
Enders, Org. Lett. 2014, 16, 5188 - 5191. Combining Silver- and Organocatalysis: A
Sequential Michael-Addition/Hydroalkoxylation One-Pot Approach to Annulated
Coumarins.
552) M. Blümel, P. Chauhan, R. Hahn, G. Raabe, D. Enders, Org. Lett. 2014, 16, 6012 -
6015. Asymmetric Synthesis of Tetrahydropyridines via an Organocatalytic One-
Pot Multicomponent Michael/aza-Henry/Cyclization Triple Domino Reaction.
553) X. Song, Q. Ni, C. Zhu, G. Raabe, D. Enders, Synthesis 2015, 47, 421 - 428.
Asymmetric NHC-Catalyzed Annulation of 2-Alkenyl-Benzothiazoles with α-
Chloroaldehydes.
554) R. Hahn, E. Jafari, G. Raabe, D. Enders, Synthesis, 2015, 47, 472 - 480.
Organocatalytic Asymmetric Synthesis of Dihydroisoquinolinones via a One-Pot
aza-Henry/Hemiaminalization/Oxidation Sequence.
555) L.-H. Zou, A. R. Philipps, G. Raabe, D. Enders, Chem. Eur. J. 2015, 21, 1004 -
1008. Asymmetric Synthesis of Fully Substituted Cyclopentane-Oxindoles via an
Organocatalytic Triple Michael Domino Reaction.
556) P. Chauhan, S. Mahajan, U. Kaya, D. Hack, D. Enders, Adv. Synth. Catal. 2015,
357, 253 –281. Bifunctional Amine-Squaramides: Powerful Hydrogen-Bonding
Organocatalysts for Asymmetric Domino/Cascade Reactions.
557) Q. Ni, X. Song, J. Xiong, G. Raabe, D. Enders, Chem. Commun. 2015, 51, 1263 -
1266. Regio- and Stereoselective Synthesis of Benzothiazolo-Pyrimidinones via an
NHC-Catalyzed Mannich/Lactamization Domino Reaction.
53
558) D. Hack, P. Chauhan, K. Deckers, Y. Mizutani, G. Raabe, D. Enders, Chem.
Commun. 2015, 51, 2266 - 2269. Combining Silver- and Organocatalysis: an
Enantioselective Sequential Catalytic Approach Towards Pyrano-Annulated
Pyrazoles.
559) S. Mahajan, P. Chauhan, C. F. J. Loh, S. Uzungelis, G. Raabe, D. Enders,
Synthesis 2015, 47, 1024 - 1031. Organocatalytic Asymmetric Domino
Michael/Henry Reaction of Indolin-3-ones with o-Formyl-β-nitrostyrenes.
560) P. Chauhan, S. Mahajan, G. Raabe, D. Enders, Chem. Commun. 2015, 51, 2270 -
2272. Organocatalytic One-Pot 1,4-/1,6-/1,2-Addition Sequence for the
Stereocontrolled Formation of Six Consecutive Stereocenters.
561) K. Zhao, T. Shu, J.Jia, G. Raabe, D. Enders, Chem. Eur. J. 2015, 21, 3933- 3936.
An Organocatalytic Mannich/Denitration Reaction for the Asymmetric Synthesis
of 3-Ethylacetate-Substitued 3-Amino-2-Oxindoles. Formal Synthesis of AG-041R.
562) C. Beceño, P. Chauhan, A. Rembiak, A. Wang, D. Enders, Adv. Synth. Catal. 2015,
357, 672 - 676. Brønsted Acid Catalyzed Enantioselective Synthesis of Isatin
Derived N,S-Acetals.
563) L. Wang, Q. Ni, M. Blümel, T. Shu, G. Raabe, D. Enders, Chem. Eur. J. 2015, 21,
8033 - 8037. NHC-Catalyzed Asymmetric Synthesis of Functionalized
Succinimides from Enals and α-Ketoamides.
564) D. Hack, M. Blümel, P. Chauhan, A. Philipps, D. Enders, Chem. Soc. Rev. 2015,
44, 6059 - 6093. Catalytic Conia-Ene and Related Reactions.
565) A. R. Philipps, L. Fritze, N. Erdmann, D. Enders, Synthesis 2015, 47, 2377 - 2384.
An Asymmetric Organocatalytic Quadruple Domino Reaction Employing a
Vinylogous Friedel-Crafts/Michael/Michael/Aldol Condensation Sequence.
566) Q. Ni, X. Song, J. Xiong, G. Raabe, D. Enders, Synlett 2015, 26, 1465 - 1469. NHC-
Catalyzed Enantioselective Annulation of Benzothiazolyl Ethyl Acetates with 2-
Bromoenals.
54
567) P. Chauhan, D. Enders, The TAKASAGO Times 2015, 176, 46 - 50.
Organocatalytic Quadruple Domino Reactions: an Efficient Strategy for the
Asymmetric Synthesis of Complex Molecules.
568) M. Blümel, P. Chauhan, C. Vermeeren, A. Dreier, C. Lehmann, D. Enders,
Synthesis. 2015, 47, 3618 - 3628. Asymmetric Organocatalytic Synthesis of Highly
Functionalized Spirocyclohexane-Indandiones via a One-Pot Michael/ Michael/ Al-
dol Sequence.
569) P. Chauhan, S. Mahajan, D. Enders, Chem. Commun. 2015, 51, 12890 - 12907.
Asymmetric Synthesis of Pyrazoles and Pyrazolones Employing the Reactivity of
Pyrazolin-5-one Derivatives.
570) C. Beceño, T. Krappitz, G. Raabe, D. Enders, Synthesis 2015, 47, 3813 - 3821.
Asymmetric Synthesis of Tetrahydropyridines via a Brønsted Acid Catalyzed aza-
Diels-Alder Reaction.
571) Q. Ni, J. Xiong, X. Song, G. Raabe, D. Enders, Chem. Commun. 2015, 51, 14628 –
14631. NHC-Catalyzed Activation of α,β-Unsubstituted N-Acyltriazoles: An Easy
Access to Dihydropyranones.
572) Y. Zhi, K. Zhao, T. Shu, D. Enders, Synthesis 2016, 48, 238 - 244. Synthesis of
Benzotriazepine Derivatives via [4+3]Cycloaddition of aza-ortho-Quinone Methide
Intermediates and Azomethine Imines.
573) K. Zhao, Y. Zhi, A. Wang, D. Enders, ACS Catalysis 2016, 6, 657 - 660.
Asymmetric Organocatalytic Synthesis of 3-Diarylmethine-Substituted Oxindoles
Bearing a Quaternary Stereocenter via 1,6-Conjugate Addition to para-Quinone
Methides.
574) T. Shu, Q. Ni, X. Song, K. Zhao, T. Wu, R. Puttreddy, K. Rissanen, D. Enders,
Chem. Commun. 2016, 52, 2609 - 2611. Asymmetric Synthesis of Cyclopentanes
Bearing Four Contiguous Stereocenters via an NHC-Catalyzed Michael/Michael/
Esterification Domino Reaction.
575) D. Hack, A. Dürr, K. Deckers, P. Chauhan, N. Seling, L. Rübenach, L. Mertens, G.
Raabe, F. Schoenebeck, D. Enders, Angew. Chem. 2016, 128, 1829 - 1832; Angew.
Chem. Int. Ed. 2016, 55, 1797 - 1800. Asymmetric Synthesis of Spiropyrazolones
by Sequential Organo- and Silver Catalysis.
55
576) U. Kaya, P. Chauhan, D. Hack, K. Deckers, R. Puttreddy, K. Rissanen, D. Enders,
Chem. Commun. 2016, 52, 1669 - 1672. Enantioselective Synthesis of 4H-
Pyranonaphthochinones via a Sequential Squaramide and Silver Catalysis.
577) K. Zhao, Y. Zhi, X. Li, R. Puttreddy, K. Rissanen, D. Enders, Chem. Commun.
2016, 52, 2249 - 2252. Asymmetric Synthesis of 3,3’-Pyrrolidinyl-Dispirooxindoles
via a One-Pot Organocatalytic Mannich/Deprotection/aza-Michael Sequence.
578) J. Wang, L. Gibbert, S. Djudjaj, C. Alidousty, T. Rauen, U. Kunter, A. Rembiak, D.
Enders, V. Jankowski, G. S. Braun, J. Floege, T. Ostendorf, U. Raffetseder, Kidney
Int. 2016, 90, 1226 - 1237. Therapeutic Nuclear Shuttling of YB-1 Reduces Renal
Damage and Fibrosis.
579) L. Wang, S. Li, P. Chauhan, D. Hack, A. R. Philipps, R. Puttreddy, K. Rissanen, G.
Raabe, D. Enders, Chem. Eur. J. 2016, 22, 5123 - 5127. Asymmetric Three
Component One-Pot Synthesis of Spiropyrazolones and 2,5-Chromene-diones via
Aldol Condensation/NHC-Catalyzed Annulation Reactions.
580) S. Mahajan, P. Chauhan, M. Blümel, G. Raabe, R. Puttreddy, K. Rissanen, D.
Enders, Synthesis 2016, 48, 1131 - 1138. Asymmetric Synthesis of Spiro-
Tetrahydrothiophene Indane-1,3-Diones via a Squaramide-Catalyzed sulfa-
Michael/Aldol Domino Reaction.
581) M. Blümel, J.-M. Noy, D. Enders, M. H. Stenzel, T. V. Nguyen, Org. Lett. 2016, 18,
2208 - 2211. Development and Applications of Transesterification Reactions
Catalyzed by N-Heterocyclic Olefins.
582) L. Wang, S. Li, M. Blümel, A. R. Philipps, A. Wang, R. Puttreddy, K. Rissanen, D.
Enders, Angew. Chem. 2016, 128, 11276 – 11280. Angew. Chem. Int. Ed. 2016, 55,
11110 – 11114. Asymmetric Synthesis of Spirobenzazepinones with
Atroposelectivity and Spiro-1,2-Diazepinones via NHC-Catalyzed [3+4] Annulation
Reactions.
583) P. Chauhan, S. Mahajan, U. Kaya, A. Valkonen, K. Rissanen, D. Enders Adv.
Synth. Catal. 2016, 358, 3173 - 3178. Asymmetric Synthesis of Spiro β-Lactams via
a Squaramide Catalyzed sulfa-Michael Addition/Desymmetrization Protocol.
584) U. Kaya, P. Chauhan, K. Deckers, R. Puttreddy, K. Rissanen, G. Raabe, D. Enders,
Synthesis 2016, 48, 3207 - 3216. Asymmetric Synthesis of Tetrahydrobenzofurans
and Annulated Dihydropyrans via a One-Pot Cooperative Organo- and Silver
Catalysis.
56
585) M. Blümel, R. D. Crocker, J. B. Harper, D. Enders, T. V. Nguyen, Chem. Commun.
2016, 52, 7958 - 7961. N-Heterocyclic Olefins as Efficient Phase-Transfer Catalysts
for Base-Promoted Alkylation Reactions.
586) F. Vetica, J. Fronert, R. Puttreddy, K. Rissanen, D. Enders, Synthesis 2016, 48,
4451 - 4458. Asymmetric Organocatalytic Synthesis of 4-Amino-Isochromanones
via a Direct One-Pot Intramolecular Mannich Reaction.
587) U. Kaya, S. Mahajan, J.-H. Schöbel, A. Valkonen, K. Rissanen, D. Enders,
Synthesis 2016, 48, 4091 - 4098. Diastereoselective Synthesis of Spiro-Tetrahydro-
thiophene Pyrazolones via a Sulfa-Michael/Aldol Domino Reaction.
588) K. Zhao, Y. Zhi, T. Shu, A. Valkonen, K. Rissanen, D. Enders, Angew. Chem. 2016,
128,12283 – 12287; Angew. Chem. Int. Ed. 2016, 55, 12104 - 12108.
Organocatalytic Domino Oxa-Michael/1,6- Addition Reactions: A Strategy for the
Asymmetric Synthesis of Chromans Bearing Oxindole Scaffolds.
589) Y. Zhi, K. Zhao, Q. Liu, A. Wang, D. Enders, Chem. Commun. 2016, 52, 14011 –
14014. Asymmetric Synthesis of Functionalized Trifluoromethyl-Substituted
Pyrrolidines via an Organocatalytic Domino Michael/Mannich [3+2]Cycloaddition.
590) S. Dochain, F. Vetica, R. Puttreddy, K. Rissanen, Angew. Chem. 2016, 128, 16387 -
16389; Angew. Chem. Int. Ed. 2016, 55, 16153 - 16155. Combining Organocatalysis
and Lanthanide Catalysis: A Sequential One-Pot Quadruple Domino/Diels-Alder
Asymmetric Synthesis of Functionalized Tricycles.
591) F. Bröhl, D. S. Kundu, G. Raabe, D. Enders, Synthesis 2017, 49, 1243 - 1254. One-
Pot Synthesis of 1-Substituted 1H-Isochromenes by Combining Brønsted Acid with
Silver Catalysis.
592) A. R. Philipps, M, Blümel, S. Dochain, D.Hack, D. Enders, Synthesis 2017, 49,
1538 - 1546. Enantioselective Catalytic One-Pot Synthesis of Functionalized
Methyleneindanes and Methylindenes via a Michael/Conia-Ene Sequence.
593) S. Li, L. Wang, P. Chauhan, A. Peuronen, K. Rissanen, D. Enders, Synthesis 2017,
49, 1808 - 1815. Asymmetric Synthesis of Five-Membered Spiropyrazolones via N-
Heterocyclic (NHC)-Carbene Catalyzed [3+2]Annulations.
594) U. Kaya, U. P. N. Tran, D. Enders, T. V. Nguyen, Org. Lett. 2017, 19, 1398 - 1401.
N-Heterocyclic Olefin Catalyzed Silylation and Hydrosilylation Reactions of
Hydroxyl and Carbonyl Compounds.
57
595) P. Chauhan, U. Kaya, D. Enders, Adv. Synth. Catal. 2017, 359, 888 - 912.
Advances in Organocatalytic 1,6-Addition Reactions: Enantioselective
Construction of Remoted Stereogenic Centres.
596) F. Vetica, P. Chauhan, S. Dochain, D. Enders, Chem. Soc. Rev. 2017, 46, 1661 -
1674. Asymmetric Organocatalytic Methods for the Synthesis of Tetrahydropyrans
and Their Application in Total Synthesis.
597) Q. Liu, K. Zhao, Y. Zhi, G. Raabe, D. Enders, Org. Chem. Frontiers 2017, 4, 1416 -
1419. Squaramide-Catalyzed Domino Michael/aza-Henry [3+2]Cycloaddition:
Asymmetric Synthesis of Functionalized 5-Trifluoromethyl and 3-Nitro- Sub-
stituted Pyrrolidines.
598) K. Zhao, D. Enders, Angew. Chem. 2017, 129, 3808 – 3810; Angew. Chem. Int. Ed.
2017, 56, 3754 - 3756. Merging N-Heterocyclic Carbene Catalysis and Single
Electron Transfer: A New Strategy for Asymmetric Transformations.
599) X.-Y. Chen, Q. Liu, P. Chauhan, S. Li, A. Peuronen, K. Rissanen, E. Jafari, D.
Enders, Angew. Chem. 2017, 129, 6337 – 6341; Angew. Chem. Int. Ed. 2017, 56,
6241 - 6245. N-Heteocyclic Carbene Catalyzed [4+2]Annulation of Enals via a
Double Vinylogous Michael Addition: Asymmetric Synthesis of 3,5-Diaryl
Cyclohexenones.
600) M. Blümel, D. Hack, L. Ronkartz, C. Vermeeren, D. Enders, Chem. Commun.
2017, 53, 3956 - 3959. Development of an Enantioselective Amine-Silver Co-
catalyzed Conia-Ene Reaction.
601) P. Chauhan, S. Mahajan, U. Kaya, A. Peuronen, K. Rissanen, D. Enders, J. Org.
Chem. 2017, 82, 7050 - 7058. Asymmetric Synthesis of Amino-Bis-Pyrazolone
Derivatives via an Organocatalytic Mannich Reaction.
602) Y. Zhi, K. Zhao, A. Wang, U. Englert, G. Raabe, D. Enders, Adv. Synth. Catal.
2017, 359, 1867 - 1871. Asymmetric Synthesis of Cyclopentane-Substituted
Oxindoles via Organocatalytic Desymmetrization of Cyclopent-4-ene-1,3-diones.
603) M. Kumar, P. Chauhan, A. Valkonen, K. Rissanen, D. Enders, Org. Lett. 2017, 19,
3025 - 3028. Asymmetric Synthesis of Functionalized Tricyclic Chromanes via an
Organocatalytic Triple Domino Reaction.
604) S. Mahajan, P. Chauhan, U. Kaya, K. Deckers, K. Rissanen, D. Enders, Chem.
Commun. 2017, 53, 6633 - 6636. Enantioselective Synthesis of Pyrazolone α-
Aminonitrile Derivatives via an Organocatalytic Strecker Reaction.
58
605) V. P. Reddy Gajulapalli, E. Jafari, D. S. Kundu, S. Mahajan, A. Peuronen, K.
Rissanen, D. Enders, Synthesis 2017, 49, 4986 - 4995. Organocatalytic Asymmetric
Synthesis of 2,3’-Connected Bis-Indolinones by Mannich Reactions of N-
Acetylindolin-3-ones with Isatin N-BOC Ketimines.
606) L. Wang, S. Li, M. Blümel, R. Puttreddy, A. Peuronen, K. Rissanen, D. Enders,
Angew. Chem. 2017, 129, 8636 – 8641; Angew. Chem. Int. Ed. 2017, 56, 8516 -
8521. Switchable Access to Different Spirocyclopentane Oxindoles by N-Hetero-
cyclic Carbene Catalyzed Reactions of Isatin-Derived Enals and N-Sulfonyl
Ketimines.
607) D. J. M. Lyons, R. D. Crocker, D. Enders, T. V. Nguyen, Green Chem. 2017, 19,
3993 - 3996. Tropylium Salts as Efficient Organic Lewis Acid Catalysts for
Acetalization and Transacetalization Reactions in Batch and Flow.
608) Y. Zhi, K. Zhao, C. von Essen, K. Rissanen, D. Enders, Synlett 2017, 28, 2876 -
2880. Thiourea-Catalyzed Domino Michael-Mannich[3+2]Cycloadditions: A
Strategy for the Asymmetric Synthesis of 3,3‘-Pyrrolidinyl-dispirooxindoles.
609) S. Li, X.-Y. Chen, Q. Liu, A. Peuronen, K. Risanen, D. Enders, Synthesis 2017, 49,
4861 - 4868. N-Heterocyclic Carbene-Catalyzed Activation of α-Chloro-aldehydes:
Asymmetric Synthesis of 5-Cyano-Substituted Dihydropyranones.
610) F. Vetica, S. Bailey, P. Chauhan, M. Turberg, A. Ghaur, G. Raabe, D. Enders, Adv.
Synth. Catal. 2017, 359, 3729 - 3734. Desymmetrization of Cyclopentendiones via
Organocatalytic Cross-Dehydrogenative Coupling.
611) X.-Y. Chen, S. Li, H. Sheng, Q. Liu, E. Jafari, C. von Essen, K. Rissanen, D.
Enders, Chem. Eur. J. 2017, 23, 13042 - 13045. N-Heterocyclic Carbene Catalyzed
[3+2]Cycloaddition of Enals with Masked Cinnamates for the Asymmetric One-Pot
Synthesis of Adipic Acid Derivatives.
612) P. Chauhan, S. Mahajan, D. Enders, Acc.Chem. Res. 2017, 50, 2809 - 2821.
Achieving Molecular Complexity via Stereoselective Multiple Domino Reactions
Promoted by a Secondary Amine Organocatalyst.
613) Q. Liu, X.-Y. Chen, S. Li, E. Jafari. G. Raabe, D. Enders, Chem. Commun. 2017,
53, 11342 - 11344. N-Heterocyclic Carbene Catalyzed [4+2]Annulation of β-Methyl
Enals and Cyclic Trifluoromethyl Ketimines for the Asymmetric Synthesis of
Dihydroquinazolinone Derivatives.
59
614) U. Kaya, P. Chauhan, S. Mahajan, K. Deckers, A. Valkonen, K. Rissanen, D.
Enders, Angew. Chem. 2017, 129, 15560 – 15564; Angw. Chem. Int. Ed. 2017, 56,
15358 - 15362. Asymmetric Squaramide Catalyzed Domino aza-Friedel-
Crafts/N,O-Acetalization Reactions Between Naphthols and Pyrazolinone
Ketimines.
615) Q. Liu, X.-Y. Chen, S. Li, F. Vetica, G. Raabe, D. Enders, Synthesis 2018, 50, 127 -
133. Two-Step Synthesis of α,β- Unsaturated γ-Amino Acid Esters via N-
Heterocyclic Carbene Catalyzed [4+2]Cycloadditions of Enals and Nitroso
Compounds.
616) K. Zhao, Y. Zhi, A. Wang, D. Enders, Synthesis. 2018, 50, accepted. Synthesis of
Malononitrile-Substituted Diarylmethines via 1,6-Addition of Masked Acyl
Cyanides to para-Quinone Methides.
617) E. Jafari, D. S. Kundu, P. Chauhan, V. P. Reddy Gajulapalli, C. von Essen, K.
Rissanen, D. Enders, Synthesis 2018, 50, 323 - 329. Organocatalytic Enantio-
selective Vinylogous Henry Reaction of 3,5-Dimethyl-4-Nitroisoxazole with
Trifluoromethyl Ketones.
618) X.-Y. Chen, J. Xiong, Q. Liu, S. Li, H. Sheng, C. von Essen, K. Rissanen, D.
Enders, Angew. Chem. 2018, 130, 306 - 310; Angew. Int. Ed. 2018, 57, 300 - 304.
Control of N-Heterocyclic Carbene Catalyzed Reactions of Enals: Asymmetric
Synthesis of Oxindole-γ-Amino Acid Derivatives.
619) X.-Y. Chen, Q. Liu, P. Chauhan, D. Enders, Angew. Chem. 2018, accepted. N-
Heterocyclic Carbene Catalysis via Azolium Dienolates: An Efficient Strategy for
Enantioselective Remote Functionalizations.
620) Q. Li, K. Zhao, A. Peuronen, K. Rissanen, D. Enders, Y. Tang, J. Am. Chem. Soc.
2018, accepted. Enantioselelctive Total Syntheses of (+)-Hippolachnin A, (+)-
Gracilioether A, (−)-Gracilioether E and (−)-Gracilioether F.
621) F. Vetica, P. Chauhan, S. Mahajan, G. Raabe, D. Enders, Synthesis 2018, 50,
accepted. Asymmetric Organocatalytic Friedel-Crafts Hydroxyalkylation of Indoles
Using Electrophilic Pyrazole-4,5-diones.
622) S. Li, X.-Y. Chen, H. Sheng, C. von Essen, K. Rissanen, D. Enders, Synthesis 2018,
50, accepted. N-Heterocyclic Carbene Catalyzed Asymmetric Synthesis of
Dihydropyranothiazoles via Azolium Enolate Intermediates.
60
623) E. Jafari, P. Chauhan, M. Kumar, X.-Y. Chen, S. Li, C. von Essen, K. Rissanen, D.
Enders, Eur. J. Org. Chem. 2018, submitted. Organocatalytic Asymmetric
Synthesis of Trifluoromethylated Tetrahydrocarbazoles via a Vinylogous
Michael/Aldol Formal [4+2] Annulation.
624) X.-C. Chen, D. Enders, Chem. 2018, 4, accepted. Multisubstituted Unnatural
Prolines for Asymmetric Catalytic Domino Reactions.
625) L. Zhao, L. Wang, S. Li, G. Raabe, D. Enders, Synthesis 2018, 50, submitted.
Asymmetric Synthesis of Cyclopenta[c]quinoline Derivatives via N-Heterocyclic
Carbene Catalyzed 1,4- and 1,2-Addition Domino Reactions.
626) Y. Zhi, K. Zhao, C. von Essen, K. Rissanen, D. Enders, Org. Chem. Frontiers 2018,
submitted. Synthesis of trans-2,3-Dihydrobenzofurans by a Formal
[4+1]Annulation Between para-Quinone Methides and Sulfonium Salts.
627) M. Kumar, P. Chauhan, S. J. Bailey, E. Jafari, C. von Essen, K. Rissanen, D.
Enders, Org.Lett. 2018, 20, submitted. Organocatalytic Oxa-
Michael/Michael/Michael/Aldol Condensation Quadruple Domino Sequence:
Asymmetric Synthesis of Tricyclic Chromanes.
628)
629)
