2003-2004 Antineoplastics 1 February 2016 3:08 AM.

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2003-2004 Antineoplastics May 12, 2022 06:13 PM

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Aminoglutethimide Antineoplastic Immunosuppressive Glucocorticoid antagonist Aromatase inhibitor (decreases steroid synthesis)

Transcript of 2003-2004 Antineoplastics 1 February 2016 3:08 AM.

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2003-2004Antineoplastics

May 3, 202306:01 PM

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Alemtuzumab

Antineoplastic

Anti-CD52 antibody

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Aminoglutethimide

AntineoplasticImmunosuppressive

Glucocorticoid antagonistAromatase inhibitor

(decreases steroid synthesis)

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Amsacrine

Antineoplastic

Miscellaneous

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Anastrozole

AntineoplasticAntiestrogen

Aromatase inhibitor

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L-asparaginase

Antineoplastic

Protein synthesis inhibitor

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Azathioprine

ImmunosuppressiveAntineoplastic

Antimetabolite(“pseudofeedback inhibition” of

HGPRT and PRP)

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Bleomycin

Antineoplastic

Natural productAntibiotic

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Busulfan

Antineoplastic

Alkylating Agent

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Carmustine (BCNU)

Antineoplastic

Alkylating Agent

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Cisplatin

Antineoplastic

MiscellaneousCross-linking agent

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Cyclophosphamide

Antineoplastic

Alkylating Agent

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Cyclosporine

ImmunosuppressiveAntineoplastic

Binds cyclophilinInhibits calcineurin

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Cyproterone acetate

AntiandrogenAntineoplastic

androgen receptor antagonist

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Cytarabine (AraC)

Antineoplastic

Antimetabolite

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Dacarbazine

Antineoplastic

Alkylating Agent

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Dactinomycin

Antineoplastic

Natural productAntibiotic

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Daunorubicin

Antineoplastic

Anthracycline antibiotic Natural product

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Dexamethasone

AdrenocorticosteroidGlucocorticoidAntineoplastic

Anti-inflammatory steroidNot by inhalation

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Doxorubicin

Antineoplastic

Anthracycline antibioticNatural product

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Etoposide

Antineoplastic

Natural productPlant alkaloid

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Exemestane

AntineoplasticAntiestrogen

Aromatase Inhibitor

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5-Fluorouracil

Antineoplastic

AntimetaboliteThymidylate synthase inhibitor

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Fulvestrant

AntineoplasticAntiestrogen

Estrogen receptor antagonist

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Gemtuzumab

Antineoplastic

Anti-CD33 antibody

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Goserelin

AntineoplasticGonadotropin releasing

hormone(GnRH) agonist

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Hydroxyurea

Antineoplastic

MiscellaneousRibonucleotide reductase

inhibitor

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Ibritumomab

Antineoplastic

Anti-CD20 antibody

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Imatinib

Antineoplastic

MiscellaneousTyrosine kinase inhibitor

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Interleukin 2

Cytokine Antineoplastic

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Interleukin 11

Cytokine Antineoplastic (supporting

agent)

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Iressa

Antineoplastic

MiscellaneousTyrosine kinase inhibitor

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Letrozole

AntineoplasticAntiestrogen

Aromatase Inhibitor

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Leucovorin

Antineoplastic (supporting agent)

Folic acid analogue(used in methotrexate rescue)

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Leuprolide

AntineoplasticGonadotropin releasing hormone (GnRH) agonist

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Lomustine (CCNU)

Antineoplastic

Alkylating Agent

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Mechlorethamine

Antineoplastic

Alkylating Agent

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Melphalan

Antineoplastic

Alkylating Agent

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6-Mercaptopurine

Antineoplastic

Antimetabolite(“pseudofeedback inhibition” of

HGPRT and PRP – purine synthesis)

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Mesna

Antineoplastic (supporting agent)

Prevent hemorrhagic cystitisdue to cyclophosphamide

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Methotrexate

ImmunosuppressiveAntineoplastic

Folic acid antagonistDihydrofolate reductase

inhibitor

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Mitomycin C

Antineoplastic

Natural productAntibiotic

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Paclitaxel

Antineoplastic

Natural productPlant alkaloid (taxane)

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Pentostatin

Antineoplastic

MiscellaneousEnzyme inhibitor

(blocks purine synthesis)

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Rituxumab

Antineoplastic

Anti-CD20 antibody

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Tacrolimus

ImmunosuppressiveAntineoplastic

Binds FKBP (FK506 binding protein)

Inhibits calcineurin

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Thalidomide

Antineoplastic

Anti-angiogenicAnti-TNF

Leprosy (not antibiotic)

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6-Thioguanine

Antineoplastic

Antimetabolite (“pseudofeedback inhibition” of

HGPRT and PRP – purine synthesis)

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Thiotepa

Antineoplastic

Alkylating agent

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Trastuzumab

Antineoplastic

Anti-HER2 antibody

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Tumor necrosis factor

CytokineAntineoplastic

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Vinblastine

Antineoplastic

Vinca alkaloidNatural product

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Vincristine

Antineoplastic

Vinca alkaloidNatural product